IL85609A - Pharmaceutical compositions containing phenyl carbamates for systemic transdermal applications,(s)-n-ethyl-3-((1-dimethylamino)ethyl)-n-methyl-phenyl-carbamate and salts thereof and their preparation - Google Patents

Pharmaceutical compositions containing phenyl carbamates for systemic transdermal applications,(s)-n-ethyl-3-((1-dimethylamino)ethyl)-n-methyl-phenyl-carbamate and salts thereof and their preparation

Info

Publication number
IL85609A
IL85609A IL85609A IL8560988A IL85609A IL 85609 A IL85609 A IL 85609A IL 85609 A IL85609 A IL 85609A IL 8560988 A IL8560988 A IL 8560988A IL 85609 A IL85609 A IL 85609A
Authority
IL
Israel
Prior art keywords
ethyl
phenyl
carbamate
dimethylamino
salts
Prior art date
Application number
IL85609A
Other languages
English (en)
Other versions
IL85609A0 (en
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6322236&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL85609(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IL85609A0 publication Critical patent/IL85609A0/xx
Publication of IL85609A publication Critical patent/IL85609A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C271/00Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C271/06Esters of carbamic acids
    • C07C271/40Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings
    • C07C271/42Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C271/44Esters of carbamic acids having oxygen atoms of carbamate groups bound to carbon atoms of six-membered aromatic rings with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/325Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
IL85609A 1987-03-04 1988-03-02 Pharmaceutical compositions containing phenyl carbamates for systemic transdermal applications,(s)-n-ethyl-3-((1-dimethylamino)ethyl)-n-methyl-phenyl-carbamate and salts thereof and their preparation IL85609A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3706914 1987-03-04

Publications (2)

Publication Number Publication Date
IL85609A0 IL85609A0 (en) 1988-08-31
IL85609A true IL85609A (en) 1992-07-15

Family

ID=6322236

Family Applications (1)

Application Number Title Priority Date Filing Date
IL85609A IL85609A (en) 1987-03-04 1988-03-02 Pharmaceutical compositions containing phenyl carbamates for systemic transdermal applications,(s)-n-ethyl-3-((1-dimethylamino)ethyl)-n-methyl-phenyl-carbamate and salts thereof and their preparation

Country Status (29)

Country Link
US (1) US5602176A (fr)
JP (3) JP2625478B2 (fr)
KR (1) KR0133686B1 (fr)
AT (1) AT394190B (fr)
AU (1) AU618949B2 (fr)
BE (1) BE1001467A3 (fr)
CA (1) CA1307003C (fr)
CH (1) CH675720A5 (fr)
CS (1) CS411091A3 (fr)
CY (1) CY1735A (fr)
DK (1) DK175762B1 (fr)
ES (1) ES2010527A6 (fr)
FI (1) FI89165C (fr)
FR (1) FR2611707B1 (fr)
GB (1) GB2203040C (fr)
GR (1) GR1000023B (fr)
HK (1) HK110093A (fr)
HU (1) HU201906B (fr)
IE (1) IE61714B1 (fr)
IL (1) IL85609A (fr)
IT (1) IT1219853B (fr)
LU (2) LU87150A1 (fr)
MY (1) MY103225A (fr)
NL (1) NL195004C (fr)
NZ (1) NZ223714A (fr)
PT (1) PT86875B (fr)
SA (1) SA93140384B1 (fr)
SE (1) SE8800731L (fr)
ZA (1) ZA881584B (fr)

Families Citing this family (88)

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US5712282A (en) * 1994-04-15 1998-01-27 Masaomi Iyo Method for therapeutically treating tardive dyskinesia and uses thereof
US6251938B1 (en) 1996-12-18 2001-06-26 Teva Pharmaceutical Industries, Ltd., Phenylethylamine derivatives
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HU229507B1 (en) 1996-12-18 2014-01-28 Technion Res & Dev Foundation 1,2,3,4-tetrahydro-amino-naphtalenyl- and aminoindan derivatives and pharmaceutical compositions comprising them
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NZ510683A (en) 1998-10-01 2003-09-26 Novartis Ag Sustained release oral formulations of rivastigmine
US20040209849A1 (en) * 1998-11-27 2004-10-21 Sanochemia Pharmazeutika Aktiengesellschaft Use of effectors of the central cholinergic nervous system for treatment of delirium
WO2000033840A1 (fr) * 1998-12-11 2000-06-15 Bonnie Davis Utilisation d'inhibiteurs d'acetylcholine esterase pour la modulation de l'axe hypothalamo-hypophyso-gonadique
GB9923045D0 (en) * 1999-09-29 1999-12-01 Novartis Ag New oral formulations
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US20040010038A1 (en) * 2002-02-27 2004-01-15 Eran Blaugrund Propargylamino indan derivatives and propargylamino tetralin derivatives as brain-selective MAO inhibitors
CZ293014B6 (cs) 2002-10-24 2004-01-14 Léčiva, A.S. Způsob výroby (-)-(S)-3-[1-(dimethylamino)ethyl]fenyl-N-ethyl-N-methylkarbamátu
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EP1603548A4 (fr) * 2003-02-05 2007-10-10 Myriad Genetics Inc Composition et methode de traitement de troubles neurodegeneratifs
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AU2004311577A1 (en) * 2003-07-11 2005-07-21 Myriad Genetics, Inc. Pharmaceutical methods, dosing regimes and dosage forms for the treatment of Alzheimer's disease
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ES2267399B1 (es) 2005-08-04 2008-02-01 Ragactives, S.L. Procedimiento para la obtencion de carbamatos de fenilo.
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IL74497A (en) * 1985-03-05 1990-02-09 Proterra Ag Pharmaceutical compositions containing phenyl carbamate derivatives and certain phenyl carbamate derivatives
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Also Published As

Publication number Publication date
DK112588A (da) 1988-09-05
FI89165C (fi) 1993-08-25
FR2611707B1 (fr) 1990-04-20
JPH09165362A (ja) 1997-06-24
SE8800731A0 (sv) 1988-09-05
NL195004B (nl) 2003-07-01
KR0133686B1 (ko) 1998-04-21
GB2203040B (en) 1990-10-24
AU1255488A (en) 1988-09-08
CH675720A5 (fr) 1990-10-31
JPH09118617A (ja) 1997-05-06
NL8800436A (nl) 1988-10-03
SE8800731L (sv) 1988-09-05
ATA55188A (de) 1991-08-15
IE880583L (en) 1988-09-04
BE1001467A3 (fr) 1989-11-07
SA93140384B1 (ar) 2006-04-04
HUT49325A (en) 1989-09-28
GR880100125A (en) 1989-01-31
SE8800731D0 (sv) 1988-03-02
NZ223714A (en) 1994-05-26
LU87150A1 (fr) 1988-11-17
CY1735A (en) 1994-06-03
IL85609A0 (en) 1988-08-31
FI880972A0 (fi) 1988-03-02
AU618949B2 (en) 1992-01-16
IT8847693A0 (it) 1988-03-04
PT86875A (pt) 1988-04-01
PT86875B (pt) 1992-05-29
GB2203040A (en) 1988-10-12
US5602176A (en) 1997-02-11
IE61714B1 (en) 1994-11-30
DK175762B1 (da) 2005-02-14
HU201906B (en) 1991-01-28
DK112588D0 (da) 1988-03-02
CA1307003C (fr) 1992-09-01
MY103225A (en) 1993-05-29
GR1000023B (el) 1990-01-31
IT1219853B (it) 1990-05-24
FI89165B (fi) 1993-05-14
KR880011088A (ko) 1988-10-26
ES2010527A6 (es) 1989-11-16
JP2859225B2 (ja) 1999-02-17
NL195004C (nl) 2003-11-04
FI880972A (fi) 1988-09-05
GB8804888D0 (en) 1988-03-30
GB2203040C (en) 2014-07-30
HK110093A (en) 1993-10-29
AT394190B (de) 1992-02-10
ZA881584B (en) 1989-11-29
JP2625478B2 (ja) 1997-07-02
JPS63238054A (ja) 1988-10-04
CS411091A3 (en) 1992-12-16
LU90297I2 (fr) 1998-12-07
FR2611707A1 (fr) 1988-09-09

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