IL135331A - Crystalline antifungal polymorph form i and pharmaceutical compositions comprising the same - Google Patents
Crystalline antifungal polymorph form i and pharmaceutical compositions comprising the sameInfo
- Publication number
- IL135331A IL135331A IL13533198A IL13533198A IL135331A IL 135331 A IL135331 A IL 135331A IL 13533198 A IL13533198 A IL 13533198A IL 13533198 A IL13533198 A IL 13533198A IL 135331 A IL135331 A IL 135331A
- Authority
- IL
- Israel
- Prior art keywords
- same
- pharmaceutical compositions
- polymorph form
- antifungal
- crystalline
- Prior art date
Links
- 230000000843 anti-fungal effect Effects 0.000 title 1
- 229940121375 antifungal agent Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US94618397A | 1997-10-07 | 1997-10-07 | |
| PCT/US1998/020476 WO1999018097A1 (en) | 1997-10-07 | 1998-10-05 | Crystalline antifungal polymorph |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL135331A0 IL135331A0 (en) | 2001-05-20 |
| IL135331A true IL135331A (en) | 2005-08-31 |
Family
ID=25484068
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL13533198A IL135331A (en) | 1997-10-07 | 1998-10-05 | Crystalline antifungal polymorph form i and pharmaceutical compositions comprising the same |
Country Status (30)
| Country | Link |
|---|---|
| EP (1) | EP1021439B1 (de) |
| JP (4) | JP2001519346A (de) |
| KR (1) | KR100626109B1 (de) |
| CN (1) | CN1125067C (de) |
| AR (1) | AR015947A1 (de) |
| AT (1) | ATE263163T1 (de) |
| AU (1) | AU759982B2 (de) |
| BR (1) | BR9812866A (de) |
| CA (1) | CA2305803C (de) |
| CO (1) | CO4970829A1 (de) |
| CZ (1) | CZ299835B6 (de) |
| DE (1) | DE69822859T2 (de) |
| DK (1) | DK1021439T3 (de) |
| ES (1) | ES2217594T3 (de) |
| HU (1) | HU225233B1 (de) |
| ID (1) | ID29290A (de) |
| IL (1) | IL135331A (de) |
| IN (1) | IN1998CH02232A (de) |
| MX (1) | MX225999B (de) |
| MY (1) | MY130126A (de) |
| NO (1) | NO318827B1 (de) |
| NZ (1) | NZ503662A (de) |
| PE (1) | PE120499A1 (de) |
| PH (1) | PH11998002606B1 (de) |
| PL (1) | PL189317B1 (de) |
| PT (1) | PT1021439E (de) |
| SK (1) | SK285190B6 (de) |
| TW (1) | TW589310B (de) |
| WO (1) | WO1999018097A1 (de) |
| ZA (1) | ZA989063B (de) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2130540A1 (de) * | 2008-06-02 | 2009-12-09 | Sandoz AG | Pharmazeutische Zusammensetzungen mit einer kristallinen Form von Posaconazol |
| EP2141159A1 (de) | 2008-07-03 | 2010-01-06 | Sandoz AG | Kristalline Form von Posaconazol |
| CA2767489A1 (en) | 2009-07-09 | 2011-01-13 | Sandoz Ag | A crystalline form of posaconazole |
| AU2011254654B2 (en) | 2010-05-19 | 2016-01-07 | Sandoz Ag | Process for the preparation of chiral triazolones |
| RU2588570C2 (ru) | 2010-05-19 | 2016-07-10 | Сандоз Аг | Способ получения хиральных гидразидов |
| CA2798007C (en) | 2010-05-19 | 2018-10-23 | Sandoz Ag | Preparation of posaconazole intermediates |
| EP2571869B1 (de) | 2010-05-19 | 2015-09-23 | Sandoz AG | Reinigung von posaconazol und posaconazol-zwischenprodukten |
| US9493428B2 (en) | 2011-06-16 | 2016-11-15 | Sandoz Ag | Process for the preparation of a chiral compound |
| US9102664B2 (en) | 2011-09-19 | 2015-08-11 | Msn Laboratories Private Limited | Process for the preparation of triazole antifungal drug, its intermediates and polymorphs thereof |
| CA2919290A1 (en) | 2013-07-25 | 2015-01-29 | Sandoz Ag | Improved process for the preparation of crystalline form iv of posaconazole |
| ITMI20132117A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| ITMI20132114A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| ITMI20132118A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| ITMI20132115A1 (it) * | 2013-12-18 | 2015-06-19 | Djada Pharmaceutical Sa | Una forma cristallina di posaconazolo |
| CN104370894A (zh) * | 2014-10-21 | 2015-02-25 | 江苏恒盛药业有限公司 | 无定型泊沙康唑的制备工艺 |
| CN104387374A (zh) * | 2014-10-21 | 2015-03-04 | 江苏恒盛药业有限公司 | 泊沙康唑晶型i的制备工艺 |
| MX2017005120A (es) | 2014-10-21 | 2018-02-12 | Ariad Pharma Inc | Formas cristalinas de 5-cloro-n4-[-2-(dimetilfosforil) fenil]-n2-{2-metoxi-4-[4-(4-metilpiperazin-1-il)piperidin-1-il] pirimidin-2,4-diamina. |
| PL3331501T3 (pl) | 2015-08-08 | 2020-03-31 | Alfred E. Tiefenbacher (Gmbh & Co. Kg) | Preparat o zwiększonej odporności na warunki przewodu pokarmowego zawierający pozakonazol |
| EA039213B1 (ru) | 2015-12-24 | 2021-12-17 | Такеда Фармасьютикал Компани Лимитед | Сокристалл, способ его получения и лекарственное средство, содержащее сокристалл |
| EP4424308A3 (de) | 2016-02-26 | 2024-12-04 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Magenresistente formulierung mit posaconazol und einem polymeren fällungshemmer |
| CN105949278B (zh) * | 2016-03-30 | 2019-12-06 | 南京曼杰生物科技有限公司 | 一种取代的四氢呋喃水溶性衍生物及其应用 |
| WO2017032908A1 (en) | 2016-07-08 | 2017-03-02 | Synthon B.V. | Pharmaceutical composition comprising amorphous posaconazole |
| TR201620462A2 (tr) | 2016-12-31 | 2018-07-23 | Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi | POSAKONAZOL İÇEREN FARMASÖTİK BİLEŞİMLER ve ÜRETİM YÖNTEMİ |
| TR201722493A2 (tr) | 2017-12-28 | 2019-07-22 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Posakonazol i̇çeren kati farmasöti̇k kompozi̇syon |
| EP4196096A1 (de) | 2020-08-13 | 2023-06-21 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Magenresistente hochfeste formulierung mit posaconazol |
| AU2022324717A1 (en) | 2021-11-25 | 2024-06-13 | Alfred E. Tiefenbacher (Gmbh Und Co. Kg) | Granules containing posaconazole |
| EP4091604B1 (de) | 2021-11-25 | 2024-04-03 | Alfred E. Tiefenbacher (GmbH & Co. KG) | Posaconazol-haltige granulate |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL103558A0 (en) * | 1991-10-30 | 1993-03-15 | Schering Corp | Tri-substituted tetrahydrofuran antifungals |
| ZA9410142B (en) * | 1993-12-21 | 1996-05-02 | Schering Corp | Tetrahydrofuran antifungals |
| KR100352147B1 (ko) * | 1994-01-24 | 2002-11-11 | 얀센 파마슈티카 엔.브이. | 수용성아졸항진균제 |
| US5625064A (en) * | 1995-04-19 | 1997-04-29 | Schering Corporation | Process for the preparation of triazolones |
| ATE240319T1 (de) * | 1995-06-02 | 2003-05-15 | Schering Corp | Antifungale tetrahydrofurane |
-
1998
- 1998-10-05 WO PCT/US1998/020476 patent/WO1999018097A1/en not_active Ceased
- 1998-10-05 CZ CZ20001264A patent/CZ299835B6/cs not_active IP Right Cessation
- 1998-10-05 ES ES98951994T patent/ES2217594T3/es not_active Expired - Lifetime
- 1998-10-05 HU HU0004899A patent/HU225233B1/hu unknown
- 1998-10-05 CA CA002305803A patent/CA2305803C/en not_active Expired - Lifetime
- 1998-10-05 JP JP2000514908A patent/JP2001519346A/ja not_active Withdrawn
- 1998-10-05 PT PT98951994T patent/PT1021439E/pt unknown
- 1998-10-05 CN CN98811886A patent/CN1125067C/zh not_active Expired - Lifetime
- 1998-10-05 AT AT98951994T patent/ATE263163T1/de active
- 1998-10-05 AR ARP980104957A patent/AR015947A1/es not_active Application Discontinuation
- 1998-10-05 CO CO98057733A patent/CO4970829A1/es unknown
- 1998-10-05 SK SK512-2000A patent/SK285190B6/sk not_active IP Right Cessation
- 1998-10-05 EP EP98951994A patent/EP1021439B1/de not_active Expired - Lifetime
- 1998-10-05 DE DE69822859T patent/DE69822859T2/de not_active Expired - Lifetime
- 1998-10-05 ZA ZA989063A patent/ZA989063B/xx unknown
- 1998-10-05 NZ NZ503662A patent/NZ503662A/xx not_active IP Right Cessation
- 1998-10-05 IL IL13533198A patent/IL135331A/xx not_active IP Right Cessation
- 1998-10-05 BR BR9812866-3A patent/BR9812866A/pt not_active Application Discontinuation
- 1998-10-05 DK DK98951994T patent/DK1021439T3/da active
- 1998-10-05 ID IDW20000632A patent/ID29290A/id unknown
- 1998-10-05 PE PE1998000942A patent/PE120499A1/es not_active IP Right Cessation
- 1998-10-05 AU AU97803/98A patent/AU759982B2/en not_active Expired
- 1998-10-05 KR KR20007003709A patent/KR100626109B1/ko not_active Expired - Lifetime
- 1998-10-05 PL PL98339659A patent/PL189317B1/pl unknown
- 1998-10-06 MY MYPI98004576A patent/MY130126A/en unknown
- 1998-10-06 TW TW087116562A patent/TW589310B/zh not_active IP Right Cessation
- 1998-10-06 IN IN2232CH1998 patent/IN1998CH02232A/en unknown
- 1998-10-06 PH PH11998002606A patent/PH11998002606B1/en unknown
-
2000
- 2000-04-06 MX MXPA00003404 patent/MX225999B/es active IP Right Grant
- 2000-04-06 NO NO20001779A patent/NO318827B1/no not_active IP Right Cessation
-
2008
- 2008-01-04 JP JP2008000110A patent/JP2008106075A/ja not_active Withdrawn
-
2012
- 2012-05-18 JP JP2012114724A patent/JP2012153729A/ja active Pending
- 2012-05-18 JP JP2012114725A patent/JP2012153730A/ja active Pending
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| EXP | Patent expired |