HU186951B - Process for producing substitited thizaolo-bracket-3,2-a-bracket closed-parimidines and pharmaceutical compositions containing them - Google Patents
Process for producing substitited thizaolo-bracket-3,2-a-bracket closed-parimidines and pharmaceutical compositions containing them Download PDFInfo
- Publication number
- HU186951B HU186951B HU822289A HU228982A HU186951B HU 186951 B HU186951 B HU 186951B HU 822289 A HU822289 A HU 822289A HU 228982 A HU228982 A HU 228982A HU 186951 B HU186951 B HU 186951B
- Authority
- HU
- Hungary
- Prior art keywords
- formula
- alkyl
- group
- pyridyl
- thiazolo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Biochemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Molecular Biology (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Rheumatology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8121979 | 1981-07-15 | ||
| GB8201621 | 1982-01-20 | ||
| GB8212430 | 1982-04-29 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HU186951B true HU186951B (en) | 1985-10-28 |
Family
ID=27261230
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU822289A HU186951B (en) | 1981-07-15 | 1982-07-14 | Process for producing substitited thizaolo-bracket-3,2-a-bracket closed-parimidines and pharmaceutical compositions containing them |
Country Status (25)
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL8202706A (nl) * | 1981-07-15 | 1983-02-01 | Erba Farmitalia | Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan. |
| AU553266B2 (en) * | 1982-02-04 | 1986-07-10 | Farmitalia Carlo Erba S.P.A. | Substituted 1,3,4-thiadiazolo(3,2-a) pyrimidines |
| US4546101A (en) * | 1982-09-10 | 1985-10-08 | Fujisawa Pharmaceutical Co., Ltd. | New cephem compounds useful for treating infectious diseases in human being and animals and processes for preparation thereof |
| GB8300728D0 (en) * | 1983-01-12 | 1983-02-16 | Erba Farmitalia | Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives |
| DE10112197A1 (de) * | 2001-03-14 | 2002-09-19 | Gruenenthal Gmbh | Substituierte Pyrazolo- und Thiazolopyrimidine |
| EP2229388A4 (en) * | 2008-01-11 | 2012-03-07 | Glenmark Pharmaceuticals Sa | CONDENSED PYRIMIDINE DERIVATIVES AS TRPV3 MODULATORS |
| US8119647B2 (en) * | 2008-04-23 | 2012-02-21 | Glenmark Pharmaceuticals S.A. | Fused pyrimidineone compounds as TRPV3 modulators |
| JP5539978B2 (ja) * | 2008-07-02 | 2014-07-02 | アベキサ・リミテッド | チアゾピリミジノンおよびその使用 |
| CN106916168B (zh) * | 2017-03-13 | 2019-08-27 | 牡丹江医学院 | 一种治疗重症胰腺炎的化合物及其制备方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3594378A (en) * | 1969-10-24 | 1971-07-20 | Ayerst Mckenna & Harrison | Thiazolopyrimidine derivatives and preparation thereof |
| US3888983A (en) * | 1970-08-14 | 1975-06-10 | Seperic | Derivatives of thiazolino-pyrimidin-6-ones, in inducing analgesia |
| GB2084568A (en) * | 1980-08-16 | 1982-04-15 | Beecham Group Ltd | Imidazothiazole derivatives |
| NL8202706A (nl) * | 1981-07-15 | 1983-02-01 | Erba Farmitalia | Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan. |
-
1982
- 1982-07-06 NL NL8202706A patent/NL8202706A/nl not_active Application Discontinuation
- 1982-07-06 AU AU85648/82A patent/AU551718B2/en not_active Ceased
- 1982-07-07 NZ NZ201194A patent/NZ201194A/en unknown
- 1982-07-07 LU LU84262A patent/LU84262A1/xx unknown
- 1982-07-08 AT AT0266182A patent/AT384614B/de not_active IP Right Cessation
- 1982-07-08 ES ES513808A patent/ES513808A0/es active Granted
- 1982-07-12 YU YU01515/82A patent/YU151582A/xx unknown
- 1982-07-12 IT IT22353/82A patent/IT1190914B/it active
- 1982-07-12 FI FI822468A patent/FI71940C/fi not_active IP Right Cessation
- 1982-07-12 SE SE8204292D patent/SE8204292L/xx not_active Application Discontinuation
- 1982-07-12 SE SE8204292A patent/SE453295B/sv not_active IP Right Cessation
- 1982-07-13 CH CH4272/82A patent/CH653036A5/de not_active IP Right Cessation
- 1982-07-13 PT PT75240A patent/PT75240B/pt unknown
- 1982-07-13 SU SU823466583A patent/SU1358786A3/ru active
- 1982-07-14 IL IL66316A patent/IL66316A/xx unknown
- 1982-07-14 NO NO822441A patent/NO822441L/no unknown
- 1982-07-14 GB GB08220385A patent/GB2103608B/en not_active Expired
- 1982-07-14 HU HU822289A patent/HU186951B/hu not_active IP Right Cessation
- 1982-07-14 US US06/398,302 patent/US4444773A/en not_active Expired - Fee Related
- 1982-07-14 GR GR68755A patent/GR76208B/el unknown
- 1982-07-14 CA CA000407223A patent/CA1208635A/en not_active Expired
- 1982-07-14 DK DK314682A patent/DK156222C/da not_active IP Right Cessation
- 1982-07-14 IE IE1692/82A patent/IE53426B1/en unknown
- 1982-07-15 DE DE19823226516 patent/DE3226516A1/de not_active Ceased
- 1982-07-15 KR KR8203145A patent/KR880002301B1/ko not_active Expired
- 1982-07-15 FR FR8212391A patent/FR2509734B1/fr not_active Expired
-
1983
- 1983-03-16 ES ES520642A patent/ES8404363A1/es not_active Expired
-
1984
- 1984-05-30 US US06/615,346 patent/US4551457A/en not_active Expired - Fee Related
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| HU90 | Patent valid on 900628 | ||
| HMM4 | Cancellation of final prot. due to non-payment of fee |