IT1190914B - Tiazolo (3,2-a)pirimidine sostituite e procedimento per la loro preparazione - Google Patents

Tiazolo (3,2-a)pirimidine sostituite e procedimento per la loro preparazione

Info

Publication number
IT1190914B
IT1190914B IT22353/82A IT2235382A IT1190914B IT 1190914 B IT1190914 B IT 1190914B IT 22353/82 A IT22353/82 A IT 22353/82A IT 2235382 A IT2235382 A IT 2235382A IT 1190914 B IT1190914 B IT 1190914B
Authority
IT
Italy
Prior art keywords
pyrimides
thiazol
replaced
procedure
preparation
Prior art date
Application number
IT22353/82A
Other languages
English (en)
Other versions
IT8222353A1 (it
IT8222353A0 (it
Inventor
Doria Gianfederico
Carlo Passarotti
Giuliana Arcari
Ada Buttinoni
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of IT8222353A0 publication Critical patent/IT8222353A0/it
Publication of IT8222353A1 publication Critical patent/IT8222353A1/it
Application granted granted Critical
Publication of IT1190914B publication Critical patent/IT1190914B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT22353/82A 1981-07-15 1982-07-12 Tiazolo (3,2-a)pirimidine sostituite e procedimento per la loro preparazione IT1190914B (it)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB8121979 1981-07-15
GB8201621 1982-01-20
GB8212430 1982-04-29

Publications (3)

Publication Number Publication Date
IT8222353A0 IT8222353A0 (it) 1982-07-12
IT8222353A1 IT8222353A1 (it) 1984-01-12
IT1190914B true IT1190914B (it) 1988-02-24

Family

ID=27261230

Family Applications (1)

Application Number Title Priority Date Filing Date
IT22353/82A IT1190914B (it) 1981-07-15 1982-07-12 Tiazolo (3,2-a)pirimidine sostituite e procedimento per la loro preparazione

Country Status (25)

Country Link
US (2) US4444773A (it)
KR (1) KR880002301B1 (it)
AT (1) AT384614B (it)
AU (1) AU551718B2 (it)
CA (1) CA1208635A (it)
CH (1) CH653036A5 (it)
DE (1) DE3226516A1 (it)
DK (1) DK156222C (it)
ES (2) ES513808A0 (it)
FI (1) FI71940C (it)
FR (1) FR2509734B1 (it)
GB (1) GB2103608B (it)
GR (1) GR76208B (it)
HU (1) HU186951B (it)
IE (1) IE53426B1 (it)
IL (1) IL66316A (it)
IT (1) IT1190914B (it)
LU (1) LU84262A1 (it)
NL (1) NL8202706A (it)
NO (1) NO822441L (it)
NZ (1) NZ201194A (it)
PT (1) PT75240B (it)
SE (2) SE453295B (it)
SU (1) SU1358786A3 (it)
YU (1) YU151582A (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8202706A (nl) * 1981-07-15 1983-02-01 Erba Farmitalia Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.
US4537962A (en) * 1982-02-04 1985-08-27 Farmitalia Carlo Erba, S.P.A. Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
US4546101A (en) * 1982-09-10 1985-10-08 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds useful for treating infectious diseases in human being and animals and processes for preparation thereof
GB8300728D0 (en) * 1983-01-12 1983-02-16 Erba Farmitalia Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
DE10112197A1 (de) * 2001-03-14 2002-09-19 Gruenenthal Gmbh Substituierte Pyrazolo- und Thiazolopyrimidine
EA018133B1 (ru) * 2008-01-11 2013-05-30 Гленмарк Фармасьютикалс, С.А. Конденсированные пиримидиновые производные как модуляторы trpv3
US8119647B2 (en) * 2008-04-23 2012-02-21 Glenmark Pharmaceuticals S.A. Fused pyrimidineone compounds as TRPV3 modulators
ES2408654T3 (es) * 2008-07-02 2013-06-21 Avexa Limited Tiazopirimidinonas y uso de las mismas
CN106916168B (zh) * 2017-03-13 2019-08-27 牡丹江医学院 一种治疗重症胰腺炎的化合物及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3594378A (en) * 1969-10-24 1971-07-20 Ayerst Mckenna & Harrison Thiazolopyrimidine derivatives and preparation thereof
US3888983A (en) * 1970-08-14 1975-06-10 Seperic Derivatives of thiazolino-pyrimidin-6-ones, in inducing analgesia
GB2084568A (en) * 1980-08-16 1982-04-15 Beecham Group Ltd Imidazothiazole derivatives
NL8202706A (nl) * 1981-07-15 1983-02-01 Erba Farmitalia Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.

Also Published As

Publication number Publication date
GB2103608B (en) 1985-01-30
US4444773A (en) 1984-04-24
IE53426B1 (en) 1988-11-09
AU551718B2 (en) 1986-05-08
PT75240A (en) 1982-08-01
ES8307827A1 (es) 1983-08-01
SE8204292L (sv) 1983-03-14
DK156222B (da) 1989-07-10
KR840000569A (ko) 1984-02-25
PT75240B (en) 1984-07-23
DK314682A (da) 1983-01-16
LU84262A1 (fr) 1983-02-07
US4551457A (en) 1985-11-05
SE453295B (sv) 1988-01-25
FR2509734A1 (fr) 1983-01-21
HU186951B (en) 1985-10-28
IL66316A (en) 1986-04-29
GB2103608A (en) 1983-02-23
SE8204292D0 (sv) 1982-07-12
NL8202706A (nl) 1983-02-01
FI822468L (fi) 1983-01-16
YU151582A (en) 1985-04-30
GR76208B (it) 1984-08-03
CH653036A5 (de) 1985-12-13
ES8404363A1 (es) 1984-05-01
IT8222353A1 (it) 1984-01-12
FI71940C (fi) 1987-03-09
FI822468A0 (fi) 1982-07-12
IL66316A0 (en) 1982-11-30
FI71940B (fi) 1986-11-28
SU1358786A3 (ru) 1987-12-07
ES520642A0 (es) 1984-05-01
AT384614B (de) 1987-12-10
ATA266182A (de) 1987-05-15
IE821692L (en) 1983-01-15
DE3226516A1 (de) 1983-02-03
IT8222353A0 (it) 1982-07-12
CA1208635A (en) 1986-07-29
DK156222C (da) 1989-12-04
NZ201194A (en) 1985-02-28
NO822441L (no) 1983-01-17
ES513808A0 (es) 1983-08-01
AU8564882A (en) 1983-01-20
KR880002301B1 (ko) 1988-10-22
FR2509734B1 (fr) 1985-07-19

Similar Documents

Publication Publication Date Title
MX6983E (es) Procedimiento de preparacion de derivados 1,3-dihidro-6-metil-7-hidroxifuro-(3,4-c)-piridina
IT8322837A0 (it) Cefem-derivati e procedimenti per la loro preparazione.
IT1194555B (it) 1h-pirazolo (1,5-a) pirimidine sostituite e procedimento per la loro preparazione
IT8122083A0 (it) Chinossalin-2-il-etenil-chetoni eprocedimento per la loro preparazione.
IT1166756B (it) 1,3-diaril-2-imino-imidazolidine e 2-imino-esaidro-pirimidine sostituite e procedimento per la loro preparazione
ES511220A0 (es) "procedimiento de preparacion de nuevos derivados 4-aminoetoxi-5-isopropil-2-metil".
AR229519A1 (es) Procedimiento de preparacion de derivados de 2,3-dihidro-9-fenil-1h-pirazolo(1,2-a)-indazolio
AR229367A1 (es) Procedimiento para la preparacion de 1,2-dicloroetano
IT1190914B (it) Tiazolo (3,2-a)pirimidine sostituite e procedimento per la loro preparazione
IT8423392A0 (it) Cefem composti e procedimenti per la loro preparazione.
MX159288A (es) Procedimiento para la preparacion de derivados de 3,7-diazabisiclo(3,3-1)nonano
IT1193604B (it) 1,3,4-tiadiazolo (3,2-a) pirimidine sostituite e procedimento per la loro preparazione
IT1185050B (it) Carbossi derivati di tiazolo (3,2-a) pirimidine sostituite e procedimento per la loro preparazione
IT1149020B (it) Composti fenetilpiperidinici antiaritmici e procedimento per la loro preparazione
IT8423805A0 (it) Composti azabiciclici e procedimenti per la loro preparazione.
IT1210971B (it) Composti biciclici eprocedimento per la loro preparazione.
IT1148404B (it) 2-fenil-2h-1,2,3-triazoli,procedimenti per la loro produzione e loro impiego
IT8322500A0 (it) 2-pirimidilalcansolfonati procedimenti per la loro preparazione e il loro impiego.
IT8322499A0 (it) Cianalchilpiperazine procedimenti per la loro preparazione e loro impiego.
IT8224818A0 (it) Procedimento per la preparazione del7-metil-3-metilen-7-otten-1-il-propionato.
IT1201442B (it) Alchilsolfonipropeni,procedimento per la loro preparazione e loro impiego
IT8220637A0 (it) Cefem derivati e procedimento per la loro preparazione.
MX155775A (es) Procedimiento mejorado para la preparacion de 2,3,-dicloropropionitrilo
AR228084A1 (es) Procedimiento para la preparacion de 1,2-dicloroetano
ES517636A0 (es) Procedimiento de preparacion de haloalcohil-8-4h-(1)-benzo-piran-4-onas.