FR2509734B1 - Thiazolo(3,2-a)pyrimidines substituees et procedes pour leur preparation - Google Patents

Thiazolo(3,2-a)pyrimidines substituees et procedes pour leur preparation

Info

Publication number
FR2509734B1
FR2509734B1 FR8212391A FR8212391A FR2509734B1 FR 2509734 B1 FR2509734 B1 FR 2509734B1 FR 8212391 A FR8212391 A FR 8212391A FR 8212391 A FR8212391 A FR 8212391A FR 2509734 B1 FR2509734 B1 FR 2509734B1
Authority
FR
France
Prior art keywords
thiazolo
processes
preparation
substituted pyrimidines
pyrimidines
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR8212391A
Other languages
English (en)
Other versions
FR2509734A1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of FR2509734A1 publication Critical patent/FR2509734A1/fr
Application granted granted Critical
Publication of FR2509734B1 publication Critical patent/FR2509734B1/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR8212391A 1981-07-15 1982-07-15 Thiazolo(3,2-a)pyrimidines substituees et procedes pour leur preparation Expired FR2509734B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB8121979 1981-07-15
GB8201621 1982-01-20
GB8212430 1982-04-29

Publications (2)

Publication Number Publication Date
FR2509734A1 FR2509734A1 (fr) 1983-01-21
FR2509734B1 true FR2509734B1 (fr) 1985-07-19

Family

ID=27261230

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8212391A Expired FR2509734B1 (fr) 1981-07-15 1982-07-15 Thiazolo(3,2-a)pyrimidines substituees et procedes pour leur preparation

Country Status (25)

Country Link
US (2) US4444773A (fr)
KR (1) KR880002301B1 (fr)
AT (1) AT384614B (fr)
AU (1) AU551718B2 (fr)
CA (1) CA1208635A (fr)
CH (1) CH653036A5 (fr)
DE (1) DE3226516A1 (fr)
DK (1) DK156222C (fr)
ES (2) ES513808A0 (fr)
FI (1) FI71940C (fr)
FR (1) FR2509734B1 (fr)
GB (1) GB2103608B (fr)
GR (1) GR76208B (fr)
HU (1) HU186951B (fr)
IE (1) IE53426B1 (fr)
IL (1) IL66316A (fr)
IT (1) IT1190914B (fr)
LU (1) LU84262A1 (fr)
NL (1) NL8202706A (fr)
NO (1) NO822441L (fr)
NZ (1) NZ201194A (fr)
PT (1) PT75240B (fr)
SE (2) SE453295B (fr)
SU (1) SU1358786A3 (fr)
YU (1) YU151582A (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8202706A (nl) * 1981-07-15 1983-02-01 Erba Farmitalia Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.
US4537962A (en) * 1982-02-04 1985-08-27 Farmitalia Carlo Erba, S.P.A. Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
US4546101A (en) * 1982-09-10 1985-10-08 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds useful for treating infectious diseases in human being and animals and processes for preparation thereof
GB8300728D0 (en) * 1983-01-12 1983-02-16 Erba Farmitalia Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
DE10112197A1 (de) * 2001-03-14 2002-09-19 Gruenenthal Gmbh Substituierte Pyrazolo- und Thiazolopyrimidine
EA018133B1 (ru) * 2008-01-11 2013-05-30 Гленмарк Фармасьютикалс, С.А. Конденсированные пиримидиновые производные как модуляторы trpv3
US8119647B2 (en) * 2008-04-23 2012-02-21 Glenmark Pharmaceuticals S.A. Fused pyrimidineone compounds as TRPV3 modulators
ES2408654T3 (es) * 2008-07-02 2013-06-21 Avexa Limited Tiazopirimidinonas y uso de las mismas
CN106916168B (zh) * 2017-03-13 2019-08-27 牡丹江医学院 一种治疗重症胰腺炎的化合物及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3594378A (en) * 1969-10-24 1971-07-20 Ayerst Mckenna & Harrison Thiazolopyrimidine derivatives and preparation thereof
US3888983A (en) * 1970-08-14 1975-06-10 Seperic Derivatives of thiazolino-pyrimidin-6-ones, in inducing analgesia
GB2084568A (en) * 1980-08-16 1982-04-15 Beecham Group Ltd Imidazothiazole derivatives
NL8202706A (nl) * 1981-07-15 1983-02-01 Erba Farmitalia Gesubstitueerde thiazolo3,2-apyrimidinen en werkwijzen ter bereiding ervan.

Also Published As

Publication number Publication date
GB2103608B (en) 1985-01-30
US4444773A (en) 1984-04-24
IE53426B1 (en) 1988-11-09
AU551718B2 (en) 1986-05-08
PT75240A (en) 1982-08-01
ES8307827A1 (es) 1983-08-01
SE8204292L (sv) 1983-03-14
DK156222B (da) 1989-07-10
KR840000569A (ko) 1984-02-25
PT75240B (en) 1984-07-23
DK314682A (da) 1983-01-16
LU84262A1 (fr) 1983-02-07
US4551457A (en) 1985-11-05
SE453295B (sv) 1988-01-25
FR2509734A1 (fr) 1983-01-21
HU186951B (en) 1985-10-28
IT1190914B (it) 1988-02-24
IL66316A (en) 1986-04-29
GB2103608A (en) 1983-02-23
SE8204292D0 (sv) 1982-07-12
NL8202706A (nl) 1983-02-01
FI822468L (fi) 1983-01-16
YU151582A (en) 1985-04-30
GR76208B (fr) 1984-08-03
CH653036A5 (de) 1985-12-13
ES8404363A1 (es) 1984-05-01
IT8222353A1 (it) 1984-01-12
FI71940C (fi) 1987-03-09
FI822468A0 (fi) 1982-07-12
IL66316A0 (en) 1982-11-30
FI71940B (fi) 1986-11-28
SU1358786A3 (ru) 1987-12-07
ES520642A0 (es) 1984-05-01
AT384614B (de) 1987-12-10
ATA266182A (de) 1987-05-15
IE821692L (en) 1983-01-15
DE3226516A1 (de) 1983-02-03
IT8222353A0 (it) 1982-07-12
CA1208635A (fr) 1986-07-29
DK156222C (da) 1989-12-04
NZ201194A (en) 1985-02-28
NO822441L (no) 1983-01-17
ES513808A0 (es) 1983-08-01
AU8564882A (en) 1983-01-20
KR880002301B1 (ko) 1988-10-22

Similar Documents

Publication Publication Date Title
FI822266L (fi) Nya imidazo/1,2-a/pyridiner och pyraziner
FI822605L (fi) Apparat foer tillverkning av glaskaerl
BR8202208A (pt) Conjunto de diferencial
FI821444L (fi) Apparat foer maetning av bandmaterials tjockleksprofil
FR2509734B1 (fr) Thiazolo(3,2-a)pyrimidines substituees et procedes pour leur preparation
DE3376324D1 (de) Imidazo(1,5-a)pyridine derivatives
MA19438A1 (fr) Nouveaux derives de piperazino-2 pyrimidine et procedes pour leur preparation
FI821035A0 (fi) Imidazo/1,2-a/pyrimidinderivat, deras framstaellning och anvaendning vid sjukvaord
GB2050353B (en) Substituted pyrido(1,2-a) pyrimidines
GB2114129B (en) Substituted 1,3,4-thiadiazolo(3,2-a) pyrimidines and process for their preparation
BR8203910A (pt) Filtro envolvido
GB2112776B (en) New heterocyclic anti-tumor substances
AU8531482A (en) Imidazo (1,2-a)pyrimidines
FI822329A0 (fi) Foerfarande foer framstaellning av substituerade pyrrolo/2,1-b/ kinazoliner och pyrido /2,1-b/ kinatsoliner
ZA824797B (en) Substituted thiazolo(3,2-a)pyrimidines and process for their preparation
DE3276808D1 (de) Pyrido (2,3-d) pyrimidines
DK133782A (da) 1,2-dihydropyrido(3,4-b)pyraziner samt fremgangsmaade til fremstilling af samme
BR8207164A (pt) Conjunto de filtro
PH20432A (en) Novel imidazo 1,2-a pyridines
ZA815026B (en) 2,3,6,7-tetrahydrothiazolo(3,2-a)-pyrimidine derivatives
FI811890L (fi) Apparat foer hantering av boerdor
IT8101902A0 (it) Gruppo livellatore
IE810695L (en) Pyrimidone derivatives
IT8129516V0 (it) Occhiale multiuso
IT8123833A0 (it) Apparecchiatura perl'arrotondamento di corpi di vetro.

Legal Events

Date Code Title Description
ST Notification of lapse