HRP20030635A2 - Crystal modification of a cyclic depsipeptide having improved strength - Google Patents

Crystal modification of a cyclic depsipeptide having improved strength Download PDF

Info

Publication number
HRP20030635A2
HRP20030635A2 HR20030635A HRP20030635A HRP20030635A2 HR P20030635 A2 HRP20030635 A2 HR P20030635A2 HR 20030635 A HR20030635 A HR 20030635A HR P20030635 A HRP20030635 A HR P20030635A HR P20030635 A2 HRP20030635 A2 HR P20030635A2
Authority
HR
Croatia
Prior art keywords
spp
depsipeptide
formula
crystalline form
animals
Prior art date
Application number
HR20030635A
Other languages
English (en)
Croatian (hr)
Inventor
Kalbe Jochen
Traeubel Michael
Harder Achim
Von Samson-Himmelstjerna Georg
Original Assignee
Bayer Aktiengesellschaft
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft
Publication of HRP20030635A2 publication Critical patent/HRP20030635A2/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
HR20030635A 2001-02-01 2002-01-21 Crystal modification of a cyclic depsipeptide having improved strength HRP20030635A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10104362A DE10104362A1 (de) 2001-02-01 2001-02-01 Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
PCT/EP2002/000541 WO2002066048A1 (de) 2001-02-01 2002-01-21 Kristallmodifikation eines cyclischen depsipeptids mit besserer wirksamkeit

Publications (1)

Publication Number Publication Date
HRP20030635A2 true HRP20030635A2 (en) 2005-10-31

Family

ID=7672376

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20030635A HRP20030635A2 (en) 2001-02-01 2002-01-21 Crystal modification of a cyclic depsipeptide having improved strength

Country Status (27)

Country Link
US (1) US20040115483A1 (enExample)
EP (1) EP1357932B1 (enExample)
JP (1) JP2004525111A (enExample)
KR (2) KR20030081378A (enExample)
CN (1) CN1278735C (enExample)
AT (1) ATE284703T1 (enExample)
AU (1) AU2002226415B2 (enExample)
BR (1) BRPI0206841B8 (enExample)
CA (1) CA2436832C (enExample)
CR (1) CR7039A (enExample)
CZ (1) CZ299564B6 (enExample)
DE (2) DE10104362A1 (enExample)
EE (1) EE05490B1 (enExample)
ES (1) ES2233805T3 (enExample)
HR (1) HRP20030635A2 (enExample)
HU (1) HU229229B1 (enExample)
IL (2) IL157026A0 (enExample)
MX (1) MXPA03006866A (enExample)
NO (1) NO331289B1 (enExample)
NZ (1) NZ527230A (enExample)
PL (1) PL213106B1 (enExample)
PT (1) PT1357932E (enExample)
RU (1) RU2300390C2 (enExample)
SK (1) SK286280B6 (enExample)
UA (1) UA74623C2 (enExample)
WO (1) WO2002066048A1 (enExample)
ZA (1) ZA200305864B (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080003546A1 (en) * 2006-06-29 2008-01-03 Dunbar Kimberly L Animated digital charted yarncraft instruction
RS62130B1 (sr) 2015-05-20 2021-08-31 Boehringer Ingelheim Animal Health Usa Inc Antihelmintička depsipeptidna jedinjenja
EP3397638B1 (en) 2015-12-28 2023-08-23 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
BR112019009977A2 (pt) 2016-11-16 2019-08-27 Boehringer Ingelheim Animal Health Usa Inc compostos depsipeptídicos anti-helmínticos
CN114262303A (zh) * 2022-01-04 2022-04-01 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型ii及其制备方法
CN114195732A (zh) * 2022-01-04 2022-03-18 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型iii及其制备方法
CN115010680A (zh) * 2022-07-13 2022-09-06 丽珠集团福州福兴医药有限公司 单晶型i的艾默德斯及其制备方法
CN114989110A (zh) * 2022-07-13 2022-09-02 丽珠集团福州福兴医药有限公司 单晶型ⅳ的艾默德斯及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2096907A (en) * 1981-04-22 1982-10-27 Exxon Research Engineering Co Distillation column with steam stripping
DK0634408T3 (da) * 1992-03-17 2002-04-22 Fujisawa Pharmaceutical Co Depsipeptidderivater, fremstilling og anvendelse deraf
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE4400464A1 (de) * 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
EP0872481B1 (en) * 1995-06-30 2009-03-18 Astellas Pharma Inc. Depsipeptide derivative, process for production thereof, and novel intermediate therefor
DE69634961T2 (de) * 1995-09-22 2006-04-20 Bayer Ag Neue zyklische depsipeptid pf1022 derivate
KR100551651B1 (ko) * 1997-11-10 2006-02-13 아스텔라스세이야쿠 가부시키가이샤 뎁시펩티드 유도체의 신규 결정 및 그의 제조 방법
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere

Also Published As

Publication number Publication date
PL213106B1 (pl) 2013-01-31
HUP0302880A2 (hu) 2003-12-29
NO20033413D0 (no) 2003-07-30
NZ527230A (en) 2005-04-29
BR0206841A (pt) 2004-02-25
BRPI0206841B1 (pt) 2018-02-14
RU2003126589A (ru) 2005-02-27
HUP0302880A3 (en) 2005-05-30
CZ20032063A3 (cs) 2003-11-12
EE05490B1 (et) 2011-12-15
AU2002226415B2 (en) 2007-03-22
CA2436832C (en) 2013-06-11
CN1592631A (zh) 2005-03-09
SK286280B6 (sk) 2008-06-06
KR20090041451A (ko) 2009-04-28
DE50201777D1 (de) 2005-01-20
CA2436832A1 (en) 2002-08-29
PL362389A1 (en) 2004-11-02
US20040115483A1 (en) 2004-06-17
MXPA03006866A (es) 2004-05-31
PT1357932E (pt) 2005-04-29
EP1357932B1 (de) 2004-12-15
WO2002066048A8 (de) 2003-11-20
IL157026A (en) 2010-11-30
BRPI0206841B8 (pt) 2021-05-25
HK1075013A1 (en) 2005-12-02
IL157026A0 (en) 2004-02-08
WO2002066048A1 (de) 2002-08-29
DE10104362A1 (de) 2002-08-08
NO20033413L (no) 2003-09-26
KR20030081378A (ko) 2003-10-17
ATE284703T1 (de) 2005-01-15
CN1278735C (zh) 2006-10-11
CR7039A (es) 2004-06-08
SK9882003A3 (en) 2003-12-02
EP1357932A1 (de) 2003-11-05
RU2300390C2 (ru) 2007-06-10
ZA200305864B (en) 2004-08-27
HU229229B1 (en) 2013-09-30
ES2233805T3 (es) 2005-06-16
NO331289B1 (no) 2011-11-21
EE200300365A (et) 2003-10-15
CZ299564B6 (cs) 2008-09-03
UA74623C2 (en) 2006-01-16
JP2004525111A (ja) 2004-08-19

Similar Documents

Publication Publication Date Title
AU703048B2 (en) Endoparasiticidal compositions
HU218569B (hu) Eljárás ciklusos depszipeptidek szulfonilezésére, az így előállított új vegyületek és parazitaellenes szerkénti alkalmazásuk
US5036069A (en) Anthelmintic active compound combinations
HU226207B1 (en) Endoparaziticide compositions
KR100372348B1 (ko) 내부기생충구제를위한곤충의니코틴효능성아세틸콜린수용체에대한길항물질및효능물질
MXPA96006179A (en) Agonists and antagonists of the receptors of the nicotinic acid acetilcoline of insects for the control of endoparasi
CA2436832C (en) Crystal form of a cyclic depsipeptide having improved activity
KR100485149B1 (ko) 경구 투여가능한 헥사하이드로피라진 유도체 과립
RU2250779C2 (ru) Эндопаразитицидное средство
HUP0102476A2 (hu) Szubsztituált ciklooktadepszipeptidek
WO2003082836A1 (en) New dioxomorpholines for combating endoparasites
DE19515297A1 (de) Endoparasitizide Mittel
MXPA00011972A (en) Substituted cyclooctadepsipeptides

Legal Events

Date Code Title Description
A1OB Publication of a patent application
ARAI Request for the grant of a patent on the basis of the submitted results of a substantive examination of a patent application
PPPP Transfer of rights

Owner name: BAYER ANIMAL HEALTH GMBH, DE

ODRP Renewal fee for the maintenance of a patent

Payment date: 20110120

Year of fee payment: 10

ODBI Application refused