CN1278735C - 具有改进活性的环缩酚肽的晶型 - Google Patents

具有改进活性的环缩酚肽的晶型 Download PDF

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Publication number
CN1278735C
CN1278735C CNB028044843A CN02804484A CN1278735C CN 1278735 C CN1278735 C CN 1278735C CN B028044843 A CNB028044843 A CN B028044843A CN 02804484 A CN02804484 A CN 02804484A CN 1278735 C CN1278735 C CN 1278735C
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CN
China
Prior art keywords
spp
sheep
activity
animals
epg
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CNB028044843A
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English (en)
Chinese (zh)
Other versions
CN1592631A (zh
Inventor
J·卡尔贝
M·特拉厄贝尔
A·哈尔德
G·冯萨姆森-希梅斯特杰纳
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Pharma AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of CN1592631A publication Critical patent/CN1592631A/zh
Application granted granted Critical
Publication of CN1278735C publication Critical patent/CN1278735C/zh
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K11/00Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15Depsipeptides; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
CNB028044843A 2001-02-01 2002-01-21 具有改进活性的环缩酚肽的晶型 Expired - Lifetime CN1278735C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10104362A DE10104362A1 (de) 2001-02-01 2001-02-01 Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
DE10104362.7 2001-02-01

Publications (2)

Publication Number Publication Date
CN1592631A CN1592631A (zh) 2005-03-09
CN1278735C true CN1278735C (zh) 2006-10-11

Family

ID=7672376

Family Applications (1)

Application Number Title Priority Date Filing Date
CNB028044843A Expired - Lifetime CN1278735C (zh) 2001-02-01 2002-01-21 具有改进活性的环缩酚肽的晶型

Country Status (27)

Country Link
US (1) US20040115483A1 (enExample)
EP (1) EP1357932B1 (enExample)
JP (1) JP2004525111A (enExample)
KR (2) KR20030081378A (enExample)
CN (1) CN1278735C (enExample)
AT (1) ATE284703T1 (enExample)
AU (1) AU2002226415B2 (enExample)
BR (1) BRPI0206841B8 (enExample)
CA (1) CA2436832C (enExample)
CR (1) CR7039A (enExample)
CZ (1) CZ299564B6 (enExample)
DE (2) DE10104362A1 (enExample)
EE (1) EE05490B1 (enExample)
ES (1) ES2233805T3 (enExample)
HR (1) HRP20030635A2 (enExample)
HU (1) HU229229B1 (enExample)
IL (2) IL157026A0 (enExample)
MX (1) MXPA03006866A (enExample)
NO (1) NO331289B1 (enExample)
NZ (1) NZ527230A (enExample)
PL (1) PL213106B1 (enExample)
PT (1) PT1357932E (enExample)
RU (1) RU2300390C2 (enExample)
SK (1) SK286280B6 (enExample)
UA (1) UA74623C2 (enExample)
WO (1) WO2002066048A1 (enExample)
ZA (1) ZA200305864B (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080003546A1 (en) * 2006-06-29 2008-01-03 Dunbar Kimberly L Animated digital charted yarncraft instruction
US10081656B2 (en) 2015-05-20 2018-09-25 Merial, Inc. Anthelmintic depsipeptide compounds
HUE065907T2 (hu) 2015-12-28 2024-06-28 Boehringer Ingelheim Vetmedica Gmbh Anthelmintikus hatású depszipeptid vegyületek
EP3541789A1 (en) 2016-11-16 2019-09-25 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
CN114195732A (zh) * 2022-01-04 2022-03-18 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型iii及其制备方法
CN114262303A (zh) * 2022-01-04 2022-04-01 丽珠集团福州福兴医药有限公司 一种艾默德斯的单晶型ii及其制备方法
CN115010680A (zh) * 2022-07-13 2022-09-06 丽珠集团福州福兴医药有限公司 单晶型i的艾默德斯及其制备方法
CN114989110A (zh) * 2022-07-13 2022-09-02 丽珠集团福州福兴医药有限公司 单晶型ⅳ的艾默德斯及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2096907A (en) * 1981-04-22 1982-10-27 Exxon Research Engineering Co Distillation column with steam stripping
ES2166359T3 (es) * 1992-03-17 2002-04-16 Fujisawa Pharmaceutical Co Derivado de depsipeptido, su produccion y uso.
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE4400464A1 (de) * 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
JP3985050B2 (ja) * 1995-06-30 2007-10-03 アステラス製薬株式会社 デプシペプチド誘導体その製造法およびその新規中間体
CA2232668C (en) * 1995-09-22 2011-10-18 Meiji Seika Kaisha, Ltd. Novel derivatives of cyclodepsipeptide pf1022 substance
DE69806800T2 (de) * 1997-11-10 2002-12-05 Fujisawa Pharmaceutical Co., Ltd. Kristall eines depsipeptid-derivates und verfahren zu seiner herstellung
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere

Also Published As

Publication number Publication date
CN1592631A (zh) 2005-03-09
BR0206841A (pt) 2004-02-25
NO331289B1 (no) 2011-11-21
WO2002066048A1 (de) 2002-08-29
EP1357932B1 (de) 2004-12-15
HU229229B1 (en) 2013-09-30
DE10104362A1 (de) 2002-08-08
BRPI0206841B1 (pt) 2018-02-14
CA2436832C (en) 2013-06-11
HK1075013A1 (en) 2005-12-02
ZA200305864B (en) 2004-08-27
CR7039A (es) 2004-06-08
WO2002066048A8 (de) 2003-11-20
NZ527230A (en) 2005-04-29
PL362389A1 (en) 2004-11-02
ATE284703T1 (de) 2005-01-15
KR20030081378A (ko) 2003-10-17
EE05490B1 (et) 2011-12-15
IL157026A0 (en) 2004-02-08
DE50201777D1 (de) 2005-01-20
HUP0302880A2 (hu) 2003-12-29
JP2004525111A (ja) 2004-08-19
HUP0302880A3 (en) 2005-05-30
EE200300365A (et) 2003-10-15
CZ20032063A3 (cs) 2003-11-12
HRP20030635A2 (en) 2005-10-31
BRPI0206841B8 (pt) 2021-05-25
CA2436832A1 (en) 2002-08-29
PL213106B1 (pl) 2013-01-31
NO20033413D0 (no) 2003-07-30
EP1357932A1 (de) 2003-11-05
UA74623C2 (en) 2006-01-16
RU2003126589A (ru) 2005-02-27
SK286280B6 (sk) 2008-06-06
MXPA03006866A (es) 2004-05-31
PT1357932E (pt) 2005-04-29
RU2300390C2 (ru) 2007-06-10
CZ299564B6 (cs) 2008-09-03
US20040115483A1 (en) 2004-06-17
ES2233805T3 (es) 2005-06-16
IL157026A (en) 2010-11-30
NO20033413L (no) 2003-09-26
SK9882003A3 (en) 2003-12-02
KR20090041451A (ko) 2009-04-28
AU2002226415B2 (en) 2007-03-22

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