HK74889A - Derivatives of cis,endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid,process for their preparation,medicines containing them and their use - Google Patents
Derivatives of cis,endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid,process for their preparation,medicines containing them and their useInfo
- Publication number
- HK74889A HK74889A HK748/89A HK74889A HK74889A HK 74889 A HK74889 A HK 74889A HK 748/89 A HK748/89 A HK 748/89A HK 74889 A HK74889 A HK 74889A HK 74889 A HK74889 A HK 74889A
- Authority
- HK
- Hong Kong
- Prior art keywords
- azabicyclo
- endo
- octane
- cis
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Heart & Thoracic Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE3143946 | 1981-11-05 | ||
DE19823226768 DE3226768A1 (de) | 1981-11-05 | 1982-07-17 | Derivate der cis, endo-2-azabicyclo-(3.3.0)-octan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung |
Publications (1)
Publication Number | Publication Date |
---|---|
HK74889A true HK74889A (en) | 1989-09-22 |
Family
ID=25797115
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK748/89A HK74889A (en) | 1981-11-05 | 1989-09-14 | Derivatives of cis,endo-2-azabicyclo-(3.3.0)-octane-3-carboxylic acid,process for their preparation,medicines containing them and their use |
Country Status (31)
Country | Link |
---|---|
US (4) | US4727160A (ru) |
EP (2) | EP0150263B1 (ru) |
JP (3) | JPH02104526A (ru) |
KR (1) | KR890000007B1 (ru) |
AR (1) | AR240675A1 (ru) |
AU (3) | AU565200B2 (ru) |
BG (1) | BG60532B2 (ru) |
CA (1) | CA1187087A (ru) |
CS (1) | CS247159B2 (ru) |
CZ (1) | CZ416291A3 (ru) |
DD (2) | DD203047A5 (ru) |
DE (3) | DE3226768A1 (ru) |
DK (2) | DK166624C (ru) |
DZ (1) | DZ473A1 (ru) |
ES (3) | ES8307746A1 (ru) |
FI (1) | FI81087C (ru) |
GR (1) | GR77381B (ru) |
HK (1) | HK74889A (ru) |
HU (2) | HU186594B (ru) |
IE (1) | IE56476B1 (ru) |
IL (1) | IL67172A (ru) |
JO (1) | JO1224B1 (ru) |
LU (1) | LU88260I2 (ru) |
MA (1) | MA19639A1 (ru) |
NL (1) | NL930039I2 (ru) |
NO (2) | NO156940C (ru) |
NZ (1) | NZ202378A (ru) |
PH (2) | PH22417A (ru) |
PT (1) | PT75792A (ru) |
SG (1) | SG1189G (ru) |
SU (1) | SU1277895A3 (ru) |
Families Citing this family (127)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
LU88621I2 (fr) * | 1980-10-23 | 1995-09-01 | Schering Corp | Sandopril |
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GR78413B (ru) * | 1981-12-29 | 1984-09-27 | Hoechst Ag | |
DE3246503A1 (de) * | 1982-12-16 | 1984-06-20 | Hoechst Ag, 6230 Frankfurt | Derivate der cis, endo-2-azabicyclo-(5.3.0)-decan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung |
DE3303112A1 (de) * | 1983-01-31 | 1984-08-09 | Hoechst Ag, 6230 Frankfurt | Verfahren zur racemattrennung optisch aktiver bicyclischer imino-(alpha)-carbonsaeuren |
US5175306A (en) * | 1983-01-31 | 1992-12-29 | Hoechst Aktiengesellschaft | Process for the resolution of racemates of optically active bicyclic imino-α-carboxylic esters |
DE3303344A1 (de) | 1983-02-02 | 1984-08-02 | Hoechst Ag, 6230 Frankfurt | Verfahren zur herstellung von n-alkylierten aminosaeuren und deren estern |
DE3324263A1 (de) * | 1983-07-06 | 1985-01-17 | Hoechst Ag, 6230 Frankfurt | Derivate der 2-azabicyclo(3.1.0)hexan-3-carbonsaeure, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung sowie 2-azabicyclo(3.1.0)hexan-derivate als zwischenprodukte und verfahren zu deren herstellung |
DE3333455A1 (de) * | 1983-09-16 | 1985-04-11 | Hoechst Ag, 6230 Frankfurt | Verfahren zur herstellung n-alkylierter dipeptide und deren estern |
DE3333454A1 (de) * | 1983-09-16 | 1985-04-11 | Hoechst Ag, 6230 Frankfurt | Verfahren zur herstellung von n-alkylierten dipeptiden und deren estern |
DE3410732A1 (de) * | 1984-03-23 | 1985-09-26 | Hoechst Ag, 6230 Frankfurt | Methode zur behandlung des glaukoms |
DE3413710A1 (de) * | 1984-04-12 | 1985-10-24 | Hoechst Ag, 6230 Frankfurt | Verfahren zur behandlung der herzinsuffizienz |
US5684016A (en) * | 1984-04-12 | 1997-11-04 | Hoechst Aktiengesellschaft | Method of treating cardiac insufficiency |
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DE3431541A1 (de) * | 1984-08-28 | 1986-03-06 | Hoechst Ag, 6230 Frankfurt | Cis,endo-2-azabicycloalkan-3-carbonsaeure-derivate, verfahren zu deren herstellung, deren verwendung sowie zwischenprodukte bei deren herstellung |
DE3660868D1 (en) * | 1985-02-04 | 1988-11-10 | Kanegafuchi Chemical Ind | Process for preparing ethyl-alpha-(1-carboxyethyl)-amino-gamma-oxo-gamma-phenylbutyrate |
US4925969A (en) * | 1985-02-04 | 1990-05-15 | Kanegafuchi Kagaku Kogyo Kabushiki Kaisha | Process for preparing ethyl-alpha-amino-gamma-oxo-gamma-phenybutyrate derivatives |
US4762821A (en) * | 1985-03-22 | 1988-08-09 | Syntex (U.S.A.) Inc. | N',N"-dialkylguanidino dipeptides |
DE3518514A1 (de) * | 1985-05-23 | 1986-11-27 | Hoechst Ag, 6230 Frankfurt | Neue derivate bicyclischer aminosaeuren, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung |
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1982
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- 1982-11-02 EP EP84111056A patent/EP0150263B1/de not_active Expired - Lifetime
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- 1982-11-02 EP EP82110070A patent/EP0079022B1/de not_active Expired
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- 1982-12-13 ES ES518133A patent/ES518133A0/es active Granted
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1983
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1984
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1987
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1988
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1989
- 1989-01-07 SG SG11/89A patent/SG1189G/en unknown
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- 1989-08-14 JP JP1207998A patent/JPH02104526A/ja active Granted
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1991
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1992
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1993
- 1993-05-19 NL NL930039C patent/NL930039I2/nl unknown
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1994
- 1994-02-23 BG BG98537A patent/BG60532B2/bg unknown
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1995
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