HK1089444A1 - Dihydropteridinones, method for the production and use thereof in the form of drugs - Google Patents

Dihydropteridinones, method for the production and use thereof in the form of drugs

Info

Publication number
HK1089444A1
HK1089444A1 HK06109960.1A HK06109960A HK1089444A1 HK 1089444 A1 HK1089444 A1 HK 1089444A1 HK 06109960 A HK06109960 A HK 06109960A HK 1089444 A1 HK1089444 A1 HK 1089444A1
Authority
HK
Hong Kong
Prior art keywords
dihydropteridinones
drugs
production
isomers
rests
Prior art date
Application number
HK06109960.1A
Other languages
English (en)
Inventor
Matthias Hoffmann
Matthias Grauert
Trixi Brandl
Steffen Breitfelder
Christian Eickmeier
Martin Steegmaier
Gisela Schnapp
Anke Baum
Jens Juergen Quant
Flavio Solca
Florian Colbatzky
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of HK1089444A1 publication Critical patent/HK1089444A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Transplantation (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HK06109960.1A 2003-02-26 2006-09-07 Dihydropteridinones, method for the production and use thereof in the form of drugs HK1089444A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/EP2003/001935 WO2004076454A1 (de) 2003-02-26 2003-02-26 Dihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
HK1089444A1 true HK1089444A1 (en) 2006-12-01

Family

ID=32921552

Family Applications (1)

Application Number Title Priority Date Filing Date
HK06109960.1A HK1089444A1 (en) 2003-02-26 2006-09-07 Dihydropteridinones, method for the production and use thereof in the form of drugs

Country Status (27)

Country Link
EP (1) EP1599478B1 (pl)
JP (1) JP3876265B2 (pl)
KR (1) KR100983462B1 (pl)
CN (2) CN101200457A (pl)
AT (1) ATE361924T1 (pl)
AU (1) AU2003215591B2 (pl)
BR (1) BR0318145A (pl)
CA (1) CA2517020C (pl)
CY (1) CY1106752T1 (pl)
DE (1) DE50307267D1 (pl)
DK (1) DK1599478T3 (pl)
EA (1) EA008778B1 (pl)
ES (1) ES2287583T3 (pl)
HK (1) HK1089444A1 (pl)
HR (1) HRP20050735B1 (pl)
IL (1) IL170419A (pl)
ME (1) ME00376B (pl)
MX (1) MXPA05009068A (pl)
NO (1) NO332538B1 (pl)
NZ (1) NZ542498A (pl)
PL (1) PL226417B1 (pl)
PT (1) PT1599478E (pl)
RS (1) RS52386B (pl)
SI (1) SI1599478T1 (pl)
TW (1) TWI313600B (pl)
UA (1) UA80743C2 (pl)
WO (1) WO2004076454A1 (pl)

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CN110343109B (zh) * 2019-08-21 2021-11-23 郑州大学 一种二氢蝶啶酮-磺酰胺类衍生物及其药学上可接受的盐、其制备方法及其应用
WO2023196943A1 (en) 2022-04-08 2023-10-12 Inhibrx, Inc. Dr5 agonist and plk1 inhibitor or cdk inhibitor combination therapy

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IL170419A (en) 2013-11-28
EP1599478B1 (de) 2007-05-09
TWI313600B (en) 2009-08-21
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KR20050113198A (ko) 2005-12-01
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