DK1599478T3 - Dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel - Google Patents

Dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel

Info

Publication number
DK1599478T3
DK1599478T3 DK03816028T DK03816028T DK1599478T3 DK 1599478 T3 DK1599478 T3 DK 1599478T3 DK 03816028 T DK03816028 T DK 03816028T DK 03816028 T DK03816028 T DK 03816028T DK 1599478 T3 DK1599478 T3 DK 1599478T3
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DK
Denmark
Prior art keywords
dihydropteridinones
drug
preparation
isomers
rests
Prior art date
Application number
DK03816028T
Other languages
English (en)
Inventor
Steffen Breitfelder
Christian Eickmeier
Martin Steegmaier
Gisela Schnapp
Anke Baum
Jens Juergen Quant
Flavio Solca
Florian Colbatzky
Matthias Hoffmann
Matthias Grauert
Trixi Brandl
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Application granted granted Critical
Publication of DK1599478T3 publication Critical patent/DK1599478T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D475/00—Heterocyclic compounds containing pteridine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK03816028T 2003-02-26 2003-02-26 Dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel DK1599478T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/EP2003/001935 WO2004076454A1 (de) 2003-02-26 2003-02-26 Dihydropteridinone, verfahren zu deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
DK1599478T3 true DK1599478T3 (da) 2007-09-17

Family

ID=32921552

Family Applications (1)

Application Number Title Priority Date Filing Date
DK03816028T DK1599478T3 (da) 2003-02-26 2003-02-26 Dihydropteridinoner, fremgangsmåde til fremstilling af disse og anvendelse af disse som lægemiddel

Country Status (27)

Country Link
EP (1) EP1599478B1 (da)
JP (1) JP3876265B2 (da)
KR (1) KR100983462B1 (da)
CN (2) CN100537570C (da)
AT (1) ATE361924T1 (da)
AU (1) AU2003215591B2 (da)
BR (1) BR0318145A (da)
CA (1) CA2517020C (da)
CY (1) CY1106752T1 (da)
DE (1) DE50307267D1 (da)
DK (1) DK1599478T3 (da)
EA (1) EA008778B1 (da)
ES (1) ES2287583T3 (da)
HK (1) HK1089444A1 (da)
HR (1) HRP20050735B1 (da)
IL (1) IL170419A (da)
ME (1) ME00376B (da)
MX (1) MXPA05009068A (da)
NO (1) NO332538B1 (da)
NZ (1) NZ542498A (da)
PL (1) PL226417B1 (da)
PT (1) PT1599478E (da)
RS (1) RS52386B (da)
SI (1) SI1599478T1 (da)
TW (1) TWI313600B (da)
UA (1) UA80743C2 (da)
WO (1) WO2004076454A1 (da)

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WO2002076985A1 (en) * 2001-03-23 2002-10-03 Smithkline Beecham Corporation Compounds useful as kinase inhibitors for the treatment of hyperproliferative diseases
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