HK1070285A1 - Pharmaceutical dosage form of amorphous nelfinavirmesylate - Google Patents

Pharmaceutical dosage form of amorphous nelfinavirmesylate

Info

Publication number
HK1070285A1
HK1070285A1 HK05103024A HK05103024A HK1070285A1 HK 1070285 A1 HK1070285 A1 HK 1070285A1 HK 05103024 A HK05103024 A HK 05103024A HK 05103024 A HK05103024 A HK 05103024A HK 1070285 A1 HK1070285 A1 HK 1070285A1
Authority
HK
Hong Kong
Prior art keywords
nelfinavirmesylate
amorphous
dosage form
pharmaceutical dosage
pharmaceutical
Prior art date
Application number
HK05103024A
Other languages
English (en)
Inventor
Martin Howard Infeld
Wantanee Phuapradit
Navnit Hargovindas Shah
Lin Zhang
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HK1070285A1 publication Critical patent/HK1070285A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2031Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK05103024A 2001-05-03 2005-04-11 Pharmaceutical dosage form of amorphous nelfinavirmesylate HK1070285A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28841001P 2001-05-03 2001-05-03
PCT/EP2002/004711 WO2002089835A2 (fr) 2001-05-03 2002-04-29 Forme dosifiee pharmaceutique de mesylate de nelfinavir amorphe

Publications (1)

Publication Number Publication Date
HK1070285A1 true HK1070285A1 (en) 2005-06-17

Family

ID=23106974

Family Applications (1)

Application Number Title Priority Date Filing Date
HK05103024A HK1070285A1 (en) 2001-05-03 2005-04-11 Pharmaceutical dosage form of amorphous nelfinavirmesylate

Country Status (37)

Country Link
US (1) US7014866B2 (fr)
EP (1) EP1390063B1 (fr)
JP (1) JP4101661B2 (fr)
KR (1) KR100554816B1 (fr)
CN (1) CN1255185C (fr)
AR (1) AR034320A1 (fr)
AT (1) ATE282428T1 (fr)
BG (1) BG108311A (fr)
BR (1) BR0209325A (fr)
CA (1) CA2444116C (fr)
CZ (1) CZ20033211A3 (fr)
DE (1) DE60201988T2 (fr)
EA (1) EA006627B1 (fr)
EC (1) ECSP034827A (fr)
ES (1) ES2231717T3 (fr)
GE (1) GEP20053466B (fr)
GT (1) GT200200079A (fr)
HK (1) HK1070285A1 (fr)
HR (1) HRP20030873B1 (fr)
HU (1) HU229938B1 (fr)
IL (2) IL158306A0 (fr)
IS (1) IS7010A (fr)
JO (1) JO2401B1 (fr)
MA (1) MA27018A1 (fr)
MX (1) MXPA03009971A (fr)
MY (1) MY128509A (fr)
NO (1) NO20034689D0 (fr)
NZ (1) NZ528689A (fr)
PA (1) PA8544501A1 (fr)
PE (1) PE20021159A1 (fr)
PL (1) PL366998A1 (fr)
PT (1) PT1390063E (fr)
RS (1) RS83503A (fr)
SK (1) SK14572003A3 (fr)
TW (1) TWI234461B (fr)
UA (1) UA76463C2 (fr)
WO (1) WO2002089835A2 (fr)

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Also Published As

Publication number Publication date
JO2401B1 (en) 2007-06-17
CZ20033211A3 (cs) 2004-09-15
CN1255185C (zh) 2006-05-10
MXPA03009971A (es) 2004-02-12
EA200301166A1 (ru) 2004-04-29
JP4101661B2 (ja) 2008-06-18
DE60201988D1 (de) 2004-12-23
ATE282428T1 (de) 2004-12-15
KR100554816B1 (ko) 2006-02-22
CN1547484A (zh) 2004-11-17
HUP0401238A3 (en) 2012-09-28
TWI234461B (en) 2005-06-21
BG108311A (bg) 2004-12-30
EA006627B1 (ru) 2006-02-24
KR20040007523A (ko) 2004-01-24
NO20034689L (no) 2003-10-20
PL366998A1 (en) 2005-02-07
CA2444116C (fr) 2009-01-20
HUP0401238A2 (hu) 2004-12-28
ES2231717T3 (es) 2005-05-16
PE20021159A1 (es) 2002-12-20
US20030021840A1 (en) 2003-01-30
UA76463C2 (en) 2006-08-15
GT200200079A (es) 2002-12-05
HU229938B1 (en) 2015-01-28
HRP20030873B1 (en) 2006-04-30
BR0209325A (pt) 2004-07-20
RS83503A (en) 2006-10-27
IL158306A0 (en) 2004-05-12
IL158306A (en) 2008-11-03
IS7010A (is) 2003-10-30
WO2002089835A3 (fr) 2003-05-01
NO20034689D0 (no) 2003-10-20
GEP20053466B (en) 2005-02-25
SK14572003A3 (sk) 2004-12-01
DE60201988T2 (de) 2005-12-15
JP2004527569A (ja) 2004-09-09
MA27018A1 (fr) 2004-12-20
PT1390063E (pt) 2005-03-31
NZ528689A (en) 2005-03-24
EP1390063B1 (fr) 2004-11-17
US7014866B2 (en) 2006-03-21
CA2444116A1 (fr) 2002-11-14
AR034320A1 (es) 2004-02-18
MY128509A (en) 2007-02-28
ECSP034827A (es) 2003-12-24
PA8544501A1 (es) 2002-11-18
EP1390063A2 (fr) 2004-02-25
WO2002089835A2 (fr) 2002-11-14
HRP20030873A2 (en) 2005-08-31

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