CA2398226A1 - Comprime de nelfinavir a dose elevee et methode de production connexe - Google Patents

Comprime de nelfinavir a dose elevee et methode de production connexe Download PDF

Info

Publication number
CA2398226A1
CA2398226A1 CA002398226A CA2398226A CA2398226A1 CA 2398226 A1 CA2398226 A1 CA 2398226A1 CA 002398226 A CA002398226 A CA 002398226A CA 2398226 A CA2398226 A CA 2398226A CA 2398226 A1 CA2398226 A1 CA 2398226A1
Authority
CA
Canada
Prior art keywords
nelfinavir
tablet
mixture
binder
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002398226A
Other languages
English (en)
Inventor
Grace Chen
James L. Gallagher
Yosyong Surakitbanharn
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of CA2398226A1 publication Critical patent/CA2398226A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Inorganic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Glanulating (AREA)
CA002398226A 2002-01-28 2002-08-15 Comprime de nelfinavir a dose elevee et methode de production connexe Abandoned CA2398226A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35142002P 2002-01-28 2002-01-28
US60/351,420 2002-01-28

Publications (1)

Publication Number Publication Date
CA2398226A1 true CA2398226A1 (fr) 2003-07-28

Family

ID=27663002

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002398226A Abandoned CA2398226A1 (fr) 2002-01-28 2002-08-15 Comprime de nelfinavir a dose elevee et methode de production connexe

Country Status (23)

Country Link
EP (1) EP1469836A1 (fr)
JP (1) JP2005521661A (fr)
KR (1) KR20040079952A (fr)
CN (1) CN1713895A (fr)
AR (1) AR038236A1 (fr)
BR (1) BR0307190A (fr)
CA (1) CA2398226A1 (fr)
GT (1) GT200300016A (fr)
HN (1) HN2003000048A (fr)
HU (1) HUP0500512A2 (fr)
IL (1) IL162724A0 (fr)
MX (1) MXPA04007237A (fr)
NI (1) NI200300001A (fr)
NO (1) NO20043238L (fr)
NZ (1) NZ533283A (fr)
PA (1) PA8564301A1 (fr)
PE (1) PE20030730A1 (fr)
PL (1) PL373882A1 (fr)
RU (1) RU2004123206A (fr)
SV (1) SV2004001467A (fr)
TW (1) TW200302111A (fr)
WO (1) WO2003063837A1 (fr)
ZA (1) ZA200404367B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008053276A1 (fr) * 2006-10-30 2008-05-08 Collette Nv Pièce de transition pour le transfert de poudre ou de matière granulaire depuis une ouverture de déversement vers une chaîne de convoyage et procédé de transfert de poudre ou de matière granulaire
MX2010002438A (es) * 2007-09-03 2010-03-30 Lucent Technologies Inc Metodo y sistema para verificar automaticamente el estado de conectividad de un enlace de protocolo de internet en una red de protocolo de internet.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6499984B1 (en) * 2000-05-22 2002-12-31 Warner-Lambert Company Continuous production of pharmaceutical granulation
MXPA03009971A (es) * 2001-05-03 2004-02-12 Hoffmann La Roche FORMA DE DOSIFICACIoN FARMACEUTICA DE MESILATO DE NELFINAVIR AMORFO.

Also Published As

Publication number Publication date
NI200300001A (es) 2004-12-21
RU2004123206A (ru) 2005-04-20
PE20030730A1 (es) 2003-08-28
CN1713895A (zh) 2005-12-28
PA8564301A1 (es) 2003-09-05
SV2004001467A (es) 2004-05-07
HUP0500512A2 (hu) 2005-09-28
EP1469836A1 (fr) 2004-10-27
IL162724A0 (en) 2005-11-20
NO20043238L (no) 2004-08-02
BR0307190A (pt) 2004-11-03
ZA200404367B (en) 2006-05-31
NZ533283A (en) 2006-12-22
MXPA04007237A (es) 2004-10-29
KR20040079952A (ko) 2004-09-16
AR038236A1 (es) 2005-01-05
TW200302111A (en) 2003-08-01
WO2003063837A1 (fr) 2003-08-07
PL373882A1 (en) 2005-09-19
JP2005521661A (ja) 2005-07-21
GT200300016A (es) 2003-09-11
HN2003000048A (es) 2003-10-28

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued