HK1032206A1 - Azabenzimidazole-based compounds for modulating serine/threonine protein kinase function. - Google Patents

Azabenzimidazole-based compounds for modulating serine/threonine protein kinase function.

Info

Publication number
HK1032206A1
HK1032206A1 HK01102854A HK01102854A HK1032206A1 HK 1032206 A1 HK1032206 A1 HK 1032206A1 HK 01102854 A HK01102854 A HK 01102854A HK 01102854 A HK01102854 A HK 01102854A HK 1032206 A1 HK1032206 A1 HK 1032206A1
Authority
HK
Hong Kong
Prior art keywords
threonine protein
azabenzimidazole
protein kinase
serine
based compounds
Prior art date
Application number
HK01102854A
Other languages
English (en)
Inventor
Gerald Mcmahon
Bernhard Kutscher
Heinz Weinberger
Harald App
Original Assignee
Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentaris Gmbh filed Critical Zentaris Gmbh
Publication of HK1032206A1 publication Critical patent/HK1032206A1/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HK01102854A 1997-09-26 2001-04-23 Azabenzimidazole-based compounds for modulating serine/threonine protein kinase function. HK1032206A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6014597P 1997-09-26 1997-09-26
PCT/US1998/019973 WO1999016438A1 (en) 1997-09-26 1998-09-23 Azabenzimidazole-based compounds for modulating serine/threonine protein kinase function

Publications (1)

Publication Number Publication Date
HK1032206A1 true HK1032206A1 (en) 2001-07-13

Family

ID=22027657

Family Applications (1)

Application Number Title Priority Date Filing Date
HK01102854A HK1032206A1 (en) 1997-09-26 2001-04-23 Azabenzimidazole-based compounds for modulating serine/threonine protein kinase function.

Country Status (28)

Country Link
US (2) US6093728A (bg)
EP (1) EP1017384B1 (bg)
JP (1) JP2001517699A (bg)
KR (1) KR100547929B1 (bg)
CN (1) CN1167420C (bg)
AR (1) AR017266A1 (bg)
AT (1) ATE281834T1 (bg)
AU (1) AU748849B2 (bg)
BG (1) BG64784B1 (bg)
BR (1) BR9812682A (bg)
CA (1) CA2305370C (bg)
DE (1) DE69827516T2 (bg)
DK (1) DK1017384T3 (bg)
ES (1) ES2230719T3 (bg)
HK (1) HK1032206A1 (bg)
HU (1) HUP0004024A3 (bg)
IL (4) IL135109A0 (bg)
NO (1) NO325663B1 (bg)
NZ (2) NZ503432A (bg)
PL (1) PL191618B1 (bg)
PT (1) PT1017384E (bg)
RU (1) RU2230553C2 (bg)
SK (1) SK285357B6 (bg)
TR (1) TR200001546T2 (bg)
TW (1) TW581815B (bg)
UA (1) UA72448C2 (bg)
WO (1) WO1999016438A1 (bg)
ZA (1) ZA988797B (bg)

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Also Published As

Publication number Publication date
KR100547929B1 (ko) 2006-02-02
CA2305370A1 (en) 1999-04-08
JP2001517699A (ja) 2001-10-09
US6093728A (en) 2000-07-25
CA2305370C (en) 2006-11-28
NZ503432A (en) 2002-11-26
PL339744A1 (en) 2001-01-02
ES2230719T3 (es) 2005-05-01
SK4152000A3 (en) 2002-02-05
ATE281834T1 (de) 2004-11-15
UA72448C2 (en) 2005-03-15
NO325663B1 (no) 2008-07-07
WO1999016438A1 (en) 1999-04-08
HUP0004024A2 (hu) 2001-04-28
DE69827516D1 (de) 2004-12-16
IL158649A0 (en) 2004-05-12
AU748849B2 (en) 2002-06-13
NZ517808A (en) 2003-07-25
IL135109A (en) 2007-07-04
ZA988797B (en) 1999-12-02
CN1278172A (zh) 2000-12-27
EP1017384B1 (en) 2004-11-10
SK285357B6 (sk) 2006-11-03
AU9578198A (en) 1999-04-23
NO20001555L (no) 2000-03-24
BR9812682A (pt) 2000-08-22
DE69827516T2 (de) 2005-12-01
KR20010015623A (ko) 2001-02-26
CN1167420C (zh) 2004-09-22
BG104356A (bg) 2000-12-29
BG64784B1 (bg) 2006-04-28
US6855723B2 (en) 2005-02-15
TW581815B (en) 2004-04-01
EP1017384A1 (en) 2000-07-12
AR017266A1 (es) 2001-09-05
DK1017384T3 (da) 2005-01-31
RU2230553C2 (ru) 2004-06-20
PT1017384E (pt) 2005-03-31
HUP0004024A3 (en) 2001-10-29
NO20001555D0 (no) 2000-03-24
PL191618B1 (pl) 2006-06-30
US20030181480A1 (en) 2003-09-25
IL135109A0 (en) 2001-05-20
IL158649A (en) 2006-12-10
TR200001546T2 (tr) 2000-10-23

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PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20080923