PT1017384E - Compostos com base no azabenzimidazole para modulacao da funcao de uma cinase de proteina serina/treonina - Google Patents

Compostos com base no azabenzimidazole para modulacao da funcao de uma cinase de proteina serina/treonina

Info

Publication number
PT1017384E
PT1017384E PT98949464T PT98949464T PT1017384E PT 1017384 E PT1017384 E PT 1017384E PT 98949464 T PT98949464 T PT 98949464T PT 98949464 T PT98949464 T PT 98949464T PT 1017384 E PT1017384 E PT 1017384E
Authority
PT
Portugal
Prior art keywords
serine
azabenzimidazole
protein kinase
function
treonine
Prior art date
Application number
PT98949464T
Other languages
English (en)
Inventor
Gerald Mcmahon
Harald App
Bernhard Kutscher
Weinberger Heinz
Original Assignee
Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zentaris Gmbh filed Critical Zentaris Gmbh
Publication of PT1017384E publication Critical patent/PT1017384E/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT98949464T 1997-09-26 1998-09-23 Compostos com base no azabenzimidazole para modulacao da funcao de uma cinase de proteina serina/treonina PT1017384E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6014597P 1997-09-26 1997-09-26

Publications (1)

Publication Number Publication Date
PT1017384E true PT1017384E (pt) 2005-03-31

Family

ID=22027657

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98949464T PT1017384E (pt) 1997-09-26 1998-09-23 Compostos com base no azabenzimidazole para modulacao da funcao de uma cinase de proteina serina/treonina

Country Status (28)

Country Link
US (2) US6093728A (pt)
EP (1) EP1017384B1 (pt)
JP (1) JP2001517699A (pt)
KR (1) KR100547929B1 (pt)
CN (1) CN1167420C (pt)
AR (1) AR017266A1 (pt)
AT (1) ATE281834T1 (pt)
AU (1) AU748849B2 (pt)
BG (1) BG64784B1 (pt)
BR (1) BR9812682A (pt)
CA (1) CA2305370C (pt)
DE (1) DE69827516T2 (pt)
DK (1) DK1017384T3 (pt)
ES (1) ES2230719T3 (pt)
HK (1) HK1032206A1 (pt)
HU (1) HUP0004024A3 (pt)
IL (4) IL158649A0 (pt)
NO (1) NO325663B1 (pt)
NZ (2) NZ503432A (pt)
PL (1) PL191618B1 (pt)
PT (1) PT1017384E (pt)
RU (1) RU2230553C2 (pt)
SK (1) SK285357B6 (pt)
TR (1) TR200001546T2 (pt)
TW (1) TW581815B (pt)
UA (1) UA72448C2 (pt)
WO (1) WO1999016438A1 (pt)
ZA (1) ZA988797B (pt)

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Also Published As

Publication number Publication date
HUP0004024A3 (en) 2001-10-29
IL158649A (en) 2006-12-10
HK1032206A1 (en) 2001-07-13
CN1278172A (zh) 2000-12-27
NO20001555L (no) 2000-03-24
CN1167420C (zh) 2004-09-22
UA72448C2 (en) 2005-03-15
DE69827516T2 (de) 2005-12-01
TR200001546T2 (tr) 2000-10-23
ATE281834T1 (de) 2004-11-15
BR9812682A (pt) 2000-08-22
SK4152000A3 (en) 2002-02-05
US20030181480A1 (en) 2003-09-25
AU748849B2 (en) 2002-06-13
US6093728A (en) 2000-07-25
DK1017384T3 (da) 2005-01-31
DE69827516D1 (de) 2004-12-16
IL135109A0 (en) 2001-05-20
EP1017384B1 (en) 2004-11-10
JP2001517699A (ja) 2001-10-09
US6855723B2 (en) 2005-02-15
WO1999016438A1 (en) 1999-04-08
NO20001555D0 (no) 2000-03-24
PL339744A1 (en) 2001-01-02
SK285357B6 (sk) 2006-11-03
RU2230553C2 (ru) 2004-06-20
IL135109A (en) 2007-07-04
AR017266A1 (es) 2001-09-05
BG104356A (en) 2000-12-29
IL158649A0 (en) 2004-05-12
HUP0004024A2 (hu) 2001-04-28
BG64784B1 (bg) 2006-04-28
CA2305370A1 (en) 1999-04-08
NZ517808A (en) 2003-07-25
KR20010015623A (ko) 2001-02-26
ES2230719T3 (es) 2005-05-01
AU9578198A (en) 1999-04-23
EP1017384A1 (en) 2000-07-12
CA2305370C (en) 2006-11-28
KR100547929B1 (ko) 2006-02-02
NZ503432A (en) 2002-11-26
PL191618B1 (pl) 2006-06-30
ZA988797B (en) 1999-12-02
TW581815B (en) 2004-04-01
NO325663B1 (no) 2008-07-07

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