EA200200105A1 - СОЕДИНЕНИЯ, МОДУЛИРУЮЩИЕ АКТИВНОСТЬ PPARγ; - Google Patents

СОЕДИНЕНИЯ, МОДУЛИРУЮЩИЕ АКТИВНОСТЬ PPARγ;

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Publication number
EA200200105A1
EA200200105A1 EA200200105A EA200200105A EA200200105A1 EA 200200105 A1 EA200200105 A1 EA 200200105A1 EA 200200105 A EA200200105 A EA 200200105A EA 200200105 A EA200200105 A EA 200200105A EA 200200105 A1 EA200200105 A1 EA 200200105A1
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EA
Eurasian Patent Office
Prior art keywords
pparγ activity
compounds modulating
modulating pparγ
activity
compounds
Prior art date
Application number
EA200200105A
Other languages
English (en)
Other versions
EA004887B1 (ru
Inventor
Лоренс Р. МакДжи
Джонатан Б. Хауз
Стивен М. Рубенштейн
Ацуси Хагивара
Нобору Фурукава
Хисаси Синкаи
Original Assignee
Туларик Инк.
Джапэн Тобэкоу Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Туларик Инк., Джапэн Тобэкоу Инк. filed Critical Туларик Инк.
Publication of EA200200105A1 publication Critical patent/EA200200105A1/ru
Publication of EA004887B1 publication Critical patent/EA004887B1/ru

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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Abstract

Предложены модуляторы активности PPARγ, которые используются в фармацевтических композициях и способах лечения таких состояний, как диабет типа II и ожирение.Международная заявка была опубликована вместе с отчетом о международном поиске.
EA200200105A 1999-06-30 2000-06-28 СОЕДИНЕНИЯ, МОДУЛИРУЮЩИЕ АКТИВНОСТЬ PPARγ EA004887B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14167299P 1999-06-30 1999-06-30
PCT/US2000/018178 WO2001000579A1 (en) 1999-06-30 2000-06-28 COMPOUNDS FOR THE MODULATION OF PPARη ACTIVITY

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EA200200105A1 true EA200200105A1 (ru) 2002-06-27
EA004887B1 EA004887B1 (ru) 2004-08-26

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EP (1) EP1192137B1 (ru)
JP (1) JP4295458B2 (ru)
CN (1) CN1171872C (ru)
CA (1) CA2377309C (ru)
DK (1) DK1192137T3 (ru)
EA (1) EA004887B1 (ru)
ES (1) ES2437103T3 (ru)
HK (1) HK1043369B (ru)
IL (2) IL147308A0 (ru)
MX (2) MXPA01013199A (ru)
NZ (2) NZ516455A (ru)
SG (1) SG148834A1 (ru)
WO (1) WO2001000579A1 (ru)
ZA (1) ZA200200057B (ru)

Families Citing this family (52)

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Publication number Priority date Publication date Assignee Title
US6583157B2 (en) 1998-01-29 2003-06-24 Tularik Inc. Quinolinyl and benzothiazolyl modulators
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