FR04C0013I1 - - Google Patents

Info

Publication number
FR04C0013I1
FR04C0013I1 FR04C0013C FR04C0013I1 FR 04C0013 I1 FR04C0013 I1 FR 04C0013I1 FR 04C0013 C FR04C0013 C FR 04C0013C FR 04C0013 I1 FR04C0013 I1 FR 04C0013I1
Authority
FR
France
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
Other languages
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21959336&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR04C0013(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of FR04C0013I1 publication Critical patent/FR04C0013I1/fr
Application granted granted Critical
Publication of FR04C0013I2 publication Critical patent/FR04C0013I2/fr
Active legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FR04C0013C 1997-06-11 2004-05-04 Active FR04C0013I2 (enrdf_load_stackoverflow)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4934897P 1997-06-11 1997-06-11
PCT/IB1998/000839 WO1998056802A1 (en) 1997-06-11 1998-05-29 4'-substituted-9-deoxo-9a-aza-9a-homoerythromycin a derivatives

Publications (2)

Publication Number Publication Date
FR04C0013I1 true FR04C0013I1 (enrdf_load_stackoverflow) 2004-06-11
FR04C0013I2 FR04C0013I2 (enrdf_load_stackoverflow) 2005-10-21

Family

ID=21959336

Family Applications (1)

Application Number Title Priority Date Filing Date
FR04C0013C Active FR04C0013I2 (enrdf_load_stackoverflow) 1997-06-11 2004-05-04

Country Status (49)

Country Link
US (4) US6420536B1 (enrdf_load_stackoverflow)
EP (1) EP0988310B9 (enrdf_load_stackoverflow)
JP (2) JP3315704B2 (enrdf_load_stackoverflow)
KR (1) KR100396168B1 (enrdf_load_stackoverflow)
CN (4) CN1172947C (enrdf_load_stackoverflow)
AP (1) AP1231A (enrdf_load_stackoverflow)
AR (1) AR013086A1 (enrdf_load_stackoverflow)
AT (1) ATE251173T1 (enrdf_load_stackoverflow)
AU (1) AU749816B2 (enrdf_load_stackoverflow)
BG (1) BG64391B1 (enrdf_load_stackoverflow)
BR (1) BRPI9810519B8 (enrdf_load_stackoverflow)
CA (1) CA2293823C (enrdf_load_stackoverflow)
CO (1) CO4950611A1 (enrdf_load_stackoverflow)
CZ (1) CZ298556B6 (enrdf_load_stackoverflow)
DE (2) DE69818665T2 (enrdf_load_stackoverflow)
DK (1) DK0988310T3 (enrdf_load_stackoverflow)
DZ (1) DZ2514A1 (enrdf_load_stackoverflow)
EA (1) EA002441B1 (enrdf_load_stackoverflow)
EG (1) EG24081A (enrdf_load_stackoverflow)
ES (1) ES2205487T3 (enrdf_load_stackoverflow)
FR (1) FR04C0013I2 (enrdf_load_stackoverflow)
GT (1) GT199800077A (enrdf_load_stackoverflow)
HN (1) HN1998000086A (enrdf_load_stackoverflow)
HR (1) HRP980314B1 (enrdf_load_stackoverflow)
HU (2) HU228005B1 (enrdf_load_stackoverflow)
ID (1) ID22992A (enrdf_load_stackoverflow)
IL (1) IL132809A0 (enrdf_load_stackoverflow)
IS (1) IS1998B (enrdf_load_stackoverflow)
LU (1) LU91076I9 (enrdf_load_stackoverflow)
MA (1) MA24564A1 (enrdf_load_stackoverflow)
ME (1) ME00876B (enrdf_load_stackoverflow)
MY (1) MY123354A (enrdf_load_stackoverflow)
NL (1) NL300150I2 (enrdf_load_stackoverflow)
NO (1) NO316911B1 (enrdf_load_stackoverflow)
NZ (2) NZ500660A (enrdf_load_stackoverflow)
OA (1) OA11224A (enrdf_load_stackoverflow)
PA (1) PA8452201A1 (enrdf_load_stackoverflow)
PE (1) PE79699A1 (enrdf_load_stackoverflow)
PL (1) PL191601B1 (enrdf_load_stackoverflow)
PT (1) PT988310E (enrdf_load_stackoverflow)
RS (1) RS49675B (enrdf_load_stackoverflow)
SI (1) SI0988310T1 (enrdf_load_stackoverflow)
SK (1) SK284171B6 (enrdf_load_stackoverflow)
TN (1) TNSN98082A1 (enrdf_load_stackoverflow)
TW (1) TW472060B (enrdf_load_stackoverflow)
UA (1) UA67744C2 (enrdf_load_stackoverflow)
UY (1) UY25040A1 (enrdf_load_stackoverflow)
WO (1) WO1998056802A1 (enrdf_load_stackoverflow)
ZA (1) ZA985017B (enrdf_load_stackoverflow)

Families Citing this family (54)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000086A (es) 1997-06-11 1999-03-08 Pfizer Prod Inc Derivados de 9 - desofo - 9 aza - 9a - homoeritromicina a - c - 4 sustituidos.
NZ502861A (en) * 1997-09-10 2001-03-30 Merck & Co Inc Method of treating livestock bacterial respiratory or enteric infections using 9a-azalides
EP1779853A3 (en) * 1997-09-10 2010-01-27 Merial Ltd. 9a-azalides as veterinary antimicrobial agents
US6339063B1 (en) 1997-09-10 2002-01-15 Merck & Co., Inc. 9a-azalides as veterinary antimicrobial agents
AP9801420A0 (en) * 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
EP1437360A3 (en) * 1998-08-19 2005-04-06 Pfizer Products Inc. C11 Carbamates of macrolide antibacterials
US6043227A (en) * 1998-08-19 2000-03-28 Pfizer Inc. C11 carbamates of macrolide antibacterials
US6100240A (en) * 1998-10-09 2000-08-08 Pfizer Inc Macrolide derivatives
CA2292359C (en) * 1999-01-28 2004-09-28 Pfizer Products Inc. Novel azalides and methods of making same
HUP0201341A3 (en) * 1999-05-18 2003-03-28 Pfizer Prod Inc Novel crystalline forms of a macrolide antibiotic, process for its preparation and pharmaceutical compositions containing it
CZ20013733A3 (cs) * 1999-05-24 2002-11-13 Pfizer Products Inc. Deriváty 13-methylerythromycinu
US6465437B1 (en) * 1999-06-30 2002-10-15 Pfizer Inc. Diphosphate salt of a 4″-substituted-9-deoxo-9A-AZA-9A- homoerythromycin derivative and its pharmaceutical composition
JP2003507487A (ja) * 1999-08-24 2003-02-25 アボット・ラボラトリーズ 抗菌活性を有する９ａ−アザライド類
US6764996B1 (en) 1999-08-24 2004-07-20 Abbott Laboratories 9a-azalides with antibacterial activity
US6608033B1 (en) * 1999-08-27 2003-08-19 Pfizer Inc. Treatment or prevention of coccidiosis
JP3893059B2 (ja) 2000-01-27 2007-03-14 ファイザー・プロダクツ・インク アザライド系抗生物質組成物
CA2407448A1 (en) * 2000-04-27 2001-11-01 Pfizer Products Inc. The use of azalide antibiotic compositions for treating or preventing a bacterial or protozoal infection in mammals
BR0209241A (pt) * 2001-04-27 2004-06-15 Pfizer Prod Inc Processo para preparação de derivados de9-deoxo-9a-aza-9a-homoeritromicina a 4-substituida
AU2002317415A1 (en) * 2001-08-01 2003-02-17 Pfizer Products Inc. Azalide antibiotic compositions
EP3738591A3 (en) 2003-03-10 2021-03-24 Merck Sharp & Dohme Corp. Novel antibacterial agents
WO2005030227A1 (en) 2003-09-23 2005-04-07 Enanta Pharmaceuticals, Inc. 9a, 11-3C-BICYCLIC 9a-AZALIDE DERIVATIVES
MXPA06005639A (es) * 2003-11-21 2006-08-17 Pfizer Prod Inc Adyuvante antimicrobiano.
EA011158B1 (ru) * 2004-03-16 2009-02-27 Бёрингер Ингельхайм Интернациональ Гмбх Замещённые глюкопиранозилом бензольные производные, содержащие эти соединения лекарственные средства, их применение и способ их получения
US20060116336A1 (en) * 2004-03-17 2006-06-01 American Pharmaceutical Partners, Inc. Lyophilized azithromycin formulation
US7468428B2 (en) * 2004-03-17 2008-12-23 App Pharmaceuticals, Llc Lyophilized azithromycin formulation
US7402568B2 (en) 2004-09-29 2008-07-22 Enanta Pharmaceuticals, Inc. Bicyclic 9a-azalide derivatives
US7767797B1 (en) * 2004-09-30 2010-08-03 Synovo Gmbh Macrocyclic compounds and methods of use thereof
US7271155B2 (en) 2005-01-07 2007-09-18 Enanta Pharmaceuticals, Inc. 9A, 11-2C-bicyclic 9a-azalide derivatives
WO2006087642A2 (en) * 2005-01-14 2006-08-24 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. 9a-carbamoyl and thiocarbamoyl azalides with antimalarial activity
AU2008316830B2 (en) * 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
DK2358379T3 (en) 2008-10-24 2016-03-07 Cempra Pharmaceuticals Inc BIOFORSVAR USING TRIAZOLHOLDIGE macrolides
US9937194B1 (en) * 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
AU2010292010B2 (en) 2009-09-10 2016-01-07 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and MAC diseases
BR112012023950A2 (pt) 2010-03-22 2016-07-05 Cempra Pharmaceuticals Inc formas cristalinas de um macrolídeo, e usos dos mesmos
WO2011146829A1 (en) 2010-05-20 2011-11-24 Cempra Pharmaceuticals, Inc. Processes for preparing macrolides and ketolides and intermediates therefor
WO2012034058A1 (en) 2010-09-10 2012-03-15 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
EP2619214B1 (en) * 2010-09-20 2014-12-24 Novartis AG Novel process for the preparation of 9-deoxo-9a-aza-9a-homoerythromycin a modified in the c-4'' of the cladinose ring by an epoxide group
MX2013004013A (es) * 2010-10-10 2013-09-26 Synovo Gmbh Macrolidos antiinflamatorios.
CN102993250B (zh) * 2011-07-06 2016-02-10 洛阳惠中兽药有限公司 C-3取代的-9-脱氧-9a-氮杂-9a-高红霉素a衍生物
CN102260306B (zh) * 2011-07-22 2012-07-18 山东鲁抗舍里乐药业有限公司 一种制备泰拉霉素的方法
EP2736915A1 (en) 2011-07-27 2014-06-04 Farma GRS, d.o.o. New crystalline forms of tulathromycin
EP2830632A4 (en) 2012-03-27 2015-10-21 Cempra Pharmaceuticals Inc PARENTERAL FORMULATIONS FOR THE ADMINISTRATION OF MACROLIDE ANTIBIOTICS
CN102786569B (zh) * 2012-09-07 2016-12-07 安徽中升药业有限公司 泰拉霉素中间体及其制备方法与泰拉霉素的制备方法
CA2905975A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
MX356772B (es) 2013-03-15 2018-06-13 Cempra Pharmaceuticals Inc Procesos convergentes para la preparacion de agentes antibacterianos macrolidos.
EP3027634B1 (en) * 2013-07-31 2018-03-21 Farma GRS, d.o.o. Process for preparation of tulathromycin
CN103497227B (zh) * 2013-09-13 2015-09-30 青岛科技大学 一种泰拉菌素中间体的制备方法
CN104725446B (zh) * 2015-03-26 2017-10-27 宁夏泰瑞制药股份有限公司 一种从泰拉霉素粗品中分离泰拉霉素a和泰拉霉素b的方法
CN104861018A (zh) * 2015-06-17 2015-08-26 瑞普（天津）生物药业有限公司 一种泰拉菌素的制备方法
CN105646617A (zh) * 2016-01-21 2016-06-08 杭州海尔希畜牧科技有限公司 一种制备泰拉霉素的方法
FR3048612B1 (fr) 2016-03-14 2020-10-02 Septeos Tulathromycine potentialisee
CN106046077B (zh) * 2016-08-04 2019-07-26 湖北美天生物科技股份有限公司 一种泰拉霉素a的合成方法
CN108003207B (zh) * 2017-12-19 2019-05-10 海门慧聚药业有限公司 制备泰拉霉素的方法
CN111087433B (zh) * 2018-10-23 2023-03-21 湖北美天生物科技股份有限公司 一种泰拉霉素中间体的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
US4512982A (en) * 1984-04-13 1985-04-23 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method
CA2064634C (en) * 1991-04-04 1998-08-04 James V. Heck 9-deoxo-8a-aza-8a-homoerythromycin a derivatives modified at the 4"- and8a-positions
US5226958A (en) * 1991-04-11 1993-07-13 Pacemark, Inc. Sealant for pneumatic inner tubes and tubeless tires
EP0549040A1 (en) * 1991-12-20 1993-06-30 Merck & Co. Inc. Methods of making 4" derivatives of 9-deoxo-8a-aza-8a-alkyl-8a-homoerythromycin A
US5441939A (en) * 1994-03-04 1995-08-15 Pfizer Inc. 3"-desmethoxy derivatives of erythromycin and azithromycin
HN1998000086A (es) * 1997-06-11 1999-03-08 Pfizer Prod Inc Derivados de 9 - desofo - 9 aza - 9a - homoeritromicina a - c - 4 sustituidos.
UA70972C2 (uk) 1998-11-20 2004-11-15 Пфайзер Продактс Інк. 13-членні азаліди і їх застосування як антибіотиків

Also Published As

Publication number Publication date
HK1088014A1 (zh) 2006-10-27
IL132809A0 (en) 2001-03-19
US20040180842A1 (en) 2004-09-16
CZ442199A3 (cs) 2000-07-12
JP3315704B2 (ja) 2002-08-19
DE69818665D1 (de) 2003-11-06
PE79699A1 (es) 1999-08-25
CA2293823C (en) 2004-02-17
ATE251173T1 (de) 2003-10-15
LU91076I2 (fr) 2004-07-05
HK1028048A1 (en) 2001-02-02
HU228005B1 (en) 2012-08-28
YU58699A (enrdf_load_stackoverflow) 2002-08-12
NO996106D0 (no) 1999-12-10
SI0988310T1 (en) 2004-02-29
KR20010013632A (ko) 2001-02-26
HUS1200028I1 (hu) 2016-08-29
US6420536B1 (en) 2002-07-16
NO996106L (no) 2000-02-10
IS1998B (is) 2005-03-15
CN1566129A (zh) 2005-01-19
TNSN98082A1 (fr) 2005-03-15
CA2293823A1 (en) 1998-12-17
US20020061858A1 (en) 2002-05-23
CN1172947C (zh) 2004-10-27
EA002441B1 (ru) 2002-04-25
CZ298556B6 (cs) 2007-11-07
SK284171B6 (sk) 2004-10-05
EG24081A (en) 2008-05-11
AU749816B2 (en) 2002-07-04
AU7347598A (en) 1998-12-30
RS49675B (sr) 2007-11-15
SK168399A3 (en) 2000-11-07
BRPI9810519A (pt) 2000-09-19
DE122004000018I1 (de) 2004-09-30
PA8452201A1 (es) 2000-05-24
HK1068893A1 (en) 2005-07-29
NZ500660A (en) 2002-03-01
CN1793155A (zh) 2006-06-28
EP0988310B1 (en) 2003-10-01
LU91076I9 (en) 2018-07-02
US20040023896A1 (en) 2004-02-05
CO4950611A1 (es) 2000-09-01
AP9801255A0 (en) 1998-06-30
AR013086A1 (es) 2000-12-13
BRPI9810519B1 (pt) 2012-02-22
MA24564A1 (fr) 1998-12-31
EP0988310B9 (en) 2006-03-08
NL300150I1 (nl) 2004-08-02
CN1243766C (zh) 2006-03-01
ES2205487T3 (es) 2004-05-01
HN1998000086A (es) 1999-03-08
WO1998056802A1 (en) 1998-12-17
PL337505A1 (en) 2000-08-28
ZA985017B (en) 1999-12-17
DK0988310T3 (da) 2003-12-15
UY25040A1 (es) 2000-09-29
AP1231A (en) 2003-12-11
FR04C0013I2 (enrdf_load_stackoverflow) 2005-10-21
ID22992A (id) 1999-12-23
DE69818665T2 (de) 2004-04-29
HUP0002209A3 (en) 2003-05-28
CN1793155B (zh) 2010-05-12
US6777393B2 (en) 2004-08-17
GT199800077A (es) 1999-12-02
CN1259136A (zh) 2000-07-05
NZ514871A (en) 2003-08-29
EA199901015A1 (ru) 2000-06-26
HRP980314A2 (en) 1999-04-30
JP2000514098A (ja) 2000-10-24
CN101691390A (zh) 2010-04-07
BRPI9810519B8 (pt) 2022-11-16
BG103945A (en) 2000-07-31
IS5252A (is) 1999-11-16
BG64391B1 (bg) 2004-12-30
DZ2514A1 (fr) 2003-02-01
US6936592B2 (en) 2005-08-30
ME00876B (me) 2012-06-20
EP0988310A1 (en) 2000-03-29
HRP980314B1 (en) 2004-04-30
PL191601B1 (pl) 2006-06-30
NL300150I2 (nl) 2004-09-01
NO316911B1 (no) 2004-06-21
DE122004000018I2 (de) 2011-01-13
KR100396168B1 (ko) 2003-08-27
PT988310E (pt) 2003-12-31
JP2002316933A (ja) 2002-10-31
MY123354A (en) 2006-05-31
UA67744C2 (uk) 2004-07-15
OA11224A (en) 2003-07-16
HUP0002209A2 (hu) 2000-12-28
TW472060B (en) 2002-01-11

Similar Documents

Publication Publication Date Title
BE2018C032I2 (enrdf_load_stackoverflow)
FR04C0013I1 (enrdf_load_stackoverflow)
CH0944937H2 (enrdf_load_stackoverflow)
BR9700653A (enrdf_load_stackoverflow)
BR9701757A (enrdf_load_stackoverflow)
CN3055519S (enrdf_load_stackoverflow)
CN3055123S (enrdf_load_stackoverflow)
BY4238C1 (enrdf_load_stackoverflow)
BY4349C1 (enrdf_load_stackoverflow)
CN3057614S (enrdf_load_stackoverflow)
CN3053170S (enrdf_load_stackoverflow)
CN3053500S (enrdf_load_stackoverflow)
CN3053524S (enrdf_load_stackoverflow)
CN3053525S (enrdf_load_stackoverflow)
CN3053852S (enrdf_load_stackoverflow)
CN3054099S (enrdf_load_stackoverflow)
CN3054162S (enrdf_load_stackoverflow)
CN3054602S (enrdf_load_stackoverflow)
CN3056209S (enrdf_load_stackoverflow)
CN3055113S (enrdf_load_stackoverflow)
CN3056076S (enrdf_load_stackoverflow)
CN3055179S (enrdf_load_stackoverflow)
CN3055389S (enrdf_load_stackoverflow)
CN3055471S (enrdf_load_stackoverflow)
CN3057436S (enrdf_load_stackoverflow)