FI964249A0 - Muovipäällysteinen, amoksisilliinia ja klavulanaattia käsittävä tabletti - Google Patents

Muovipäällysteinen, amoksisilliinia ja klavulanaattia käsittävä tabletti

Info

Publication number
FI964249A0
FI964249A0 FI964249A FI964249A FI964249A0 FI 964249 A0 FI964249 A0 FI 964249A0 FI 964249 A FI964249 A FI 964249A FI 964249 A FI964249 A FI 964249A FI 964249 A0 FI964249 A0 FI 964249A0
Authority
FI
Finland
Prior art keywords
clavulanate
amoxicillin
coated tablet
polymer coated
polymer
Prior art date
Application number
FI964249A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI964249A (fi
Inventor
Creighton Pierce Conley
Nigel Philip Mccreath Davidson
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10754044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI964249(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of FI964249A0 publication Critical patent/FI964249A0/fi
Publication of FI964249A publication Critical patent/FI964249A/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/2853Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893Tablet coating processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI964249A 1994-04-23 1996-10-22 Muovipäällysteinen, amoksisilliinia ja klavulanaattia käsittävä tabletti FI964249A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9408117A GB9408117D0 (en) 1994-04-23 1994-04-23 Pharmaceutical formulations
PCT/EP1995/001463 WO1995028927A1 (en) 1994-04-23 1995-04-19 Polymer coated tablet comprising amoxycillin and clavulanate

Publications (2)

Publication Number Publication Date
FI964249A0 true FI964249A0 (fi) 1996-10-22
FI964249A FI964249A (fi) 1996-10-22

Family

ID=10754044

Family Applications (1)

Application Number Title Priority Date Filing Date
FI964249A FI964249A (fi) 1994-04-23 1996-10-22 Muovipäällysteinen, amoksisilliinia ja klavulanaattia käsittävä tabletti

Country Status (35)

Country Link
US (1) US6051255A (xx)
EP (5) EP0758235B1 (xx)
JP (1) JP3622975B2 (xx)
CN (1) CN1134258C (xx)
AP (2) AP564A (xx)
AT (6) ATE203161T1 (xx)
AU (1) AU684949B2 (xx)
BG (1) BG62842B1 (xx)
BR (1) BR9507502A (xx)
CA (1) CA2188496A1 (xx)
CZ (2) CZ11376U1 (xx)
DE (5) DE69519093T2 (xx)
DK (4) DK0758235T3 (xx)
DZ (1) DZ1876A1 (xx)
ES (4) ES2180251T3 (xx)
FI (1) FI964249A (xx)
GB (1) GB9408117D0 (xx)
GR (2) GR3035031T3 (xx)
HK (5) HK1050992A1 (xx)
HU (1) HU228399B1 (xx)
IL (1) IL113433A (xx)
MA (1) MA23528A1 (xx)
MY (1) MY115351A (xx)
NO (1) NO310703B1 (xx)
NZ (1) NZ285080A (xx)
OA (1) OA10377A (xx)
PL (1) PL316966A1 (xx)
PT (4) PT761218E (xx)
RO (1) RO116997B1 (xx)
RU (1) RU2152213C1 (xx)
SA (1) SA95160343B1 (xx)
SI (1) SI0758235T1 (xx)
SK (1) SK282594B6 (xx)
WO (1) WO1995028927A1 (xx)
ZA (1) ZA953236B (xx)

Families Citing this family (67)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9407386D0 (en) 1994-04-14 1994-06-08 Smithkline Beecham Plc Pharmaceutical formulation
GB9408117D0 (en) * 1994-04-23 1994-06-15 Smithkline Beecham Corp Pharmaceutical formulations
DZ2028A1 (fr) * 1995-05-03 2002-10-23 Smithkline Beecham Plc Médicaments destinés au traitement d'infections bactériennes en pédiatrie.
US20030109503A1 (en) * 1995-06-06 2003-06-12 Smithkline Beecham P.L.C. Pharmaceutical formulations comprising clavulanic acid alone or in combination with other beta-lactam antibiotics
CN1289084C (zh) 1995-09-07 2006-12-13 史密丝克莱恩比彻姆有限公司 药物制剂
TWI225402B (en) 1996-03-13 2004-12-21 Biochemie Gmbh Auxiliary-free agglomerates
AT407701B (de) * 1996-08-12 2001-05-25 Biochemie Gmbh Zur direkttablettierung geeignete mischung, die als wesentliche komponenten amoxicillin-trihydrat und das kaliumsalz der clavulansäure enthält und verfahren zur herstellung dieser mischung
GB9613470D0 (en) 1996-06-27 1996-08-28 Ciba Geigy Ag Small solid oral dosage form
GB9616536D0 (en) 1996-08-06 1996-09-25 Quadrant Holdings Cambridge Co-amoxiclav dosage form
GB9617780D0 (en) * 1996-08-24 1996-10-02 Smithkline Beecham Plc Method of treatment
AU6496498A (en) * 1997-02-07 1998-08-26 Gist-Brocades B.V. Homogeneous granulated formulations for dose sipping technology
CN1194687C (zh) * 1997-02-14 2005-03-30 史密斯克莱恩比彻姆药物实验室 含有阿莫西林和克拉维酸盐的药物制剂
US20030124187A1 (en) * 1997-02-14 2003-07-03 Smithkline Beecham Laboratoires Pharmaceutiques, Pharmaceutical formulations comprising amoxycillin and clavulanate
AU9540898A (en) * 1997-08-29 1999-03-22 Dsm N.V. Granules free of excipients
US6395298B1 (en) 1997-10-31 2002-05-28 Pharmacia Corporation Gellan gum tablet coating
TR200102771T2 (tr) 1999-04-01 2002-04-22 Dsm N. V. Kristalleştirme ile elde edilen aglomeralar
US6878386B1 (en) 1999-04-13 2005-04-12 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising amoxycillin and potassium clavulanate
US7250176B1 (en) * 1999-04-13 2007-07-31 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection
DK200000133U3 (da) * 1999-04-13 2000-07-28 Beecham Pharm Pte Ltd Ny farmaceutisk formulering
US6294199B1 (en) 1999-04-13 2001-09-25 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising administering amoxycillin
US20040038948A1 (en) * 1999-12-07 2004-02-26 Uhrich Kathryn E. Therapeutic compositions and methods
GB9930578D0 (en) * 1999-12-23 2000-02-16 Smithkline Beecham Plc Pharmaceutical formulations
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US6565882B2 (en) * 2000-02-24 2003-05-20 Advancis Pharmaceutical Corp Antibiotic composition with inhibitor
WO2002002081A1 (en) * 2000-07-05 2002-01-10 Capricorn Pharma, Inc. Rapid-melt semi-solid compositions, methods of making same and methods of using same
US6375982B1 (en) * 2000-07-05 2002-04-23 Capricorn Pharma, Inc. Rapid-melt semi-solid compositions, methods of making same and method of using same
AU2001292185A1 (en) 2000-10-12 2002-04-22 Beecham Pharmaceuticals (Pte) Limited Formulation containing amoxicillin
US6756057B2 (en) 2000-10-12 2004-06-29 Beecham Pharmaceuticals (Pte) Limited Amoxicillin and potassium clavulanate dosage form
US20020068078A1 (en) * 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
US6541014B2 (en) * 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US20020197314A1 (en) * 2001-02-23 2002-12-26 Rudnic Edward M. Anti-fungal composition
AU4061702A (en) * 2001-05-15 2003-04-03 Mcneil-Ppc, Inc. Dip coating compositions containing starch or dextrin
US20030070584A1 (en) * 2001-05-15 2003-04-17 Cynthia Gulian Dip coating compositions containing cellulose ethers
US8309118B2 (en) * 2001-09-28 2012-11-13 Mcneil-Ppc, Inc. Film forming compositions containing sucralose
AU2003210925A1 (en) * 2002-02-07 2003-09-02 Rutgers, The State University Antibiotic polymers
KR100967782B1 (ko) * 2002-02-14 2010-07-05 글락소 그룹 리미티드 N-((1-N-부틸-4-피페리디닐)메틸)-3,4-디하이드로-2H-(1,3)옥사지노(3,2-a)인돌-10-카복스아미드 또는 그의 염을포함하는 제약 조성물, 및 건식 과립화를 포함하는 그의제조 방법
GB0203528D0 (en) * 2002-02-14 2002-04-03 Glaxo Group Ltd Process and composition
US8637512B2 (en) 2002-07-29 2014-01-28 Glaxo Group Limited Formulations and method of treatment
KR100456833B1 (ko) * 2002-08-01 2004-11-10 주식회사 대웅 아목시실린 및 클라불라네이트를 함유하는 유핵정
US7429619B2 (en) * 2002-08-02 2008-09-30 Mcneil Consumer Healthcare Polyacrylic film forming compositions
CA2406592C (en) * 2002-10-04 2003-09-30 Duchesnay Inc. Method of preparing pharmaceutical dosage forms containing multiple active ingredients
US7405210B2 (en) 2003-05-21 2008-07-29 Osi Pharmaceuticals, Inc. Pyrrolopyridine-2-carboxylic acid amide inhibitors of glycogen phosphorylase
WO2005009365A2 (en) * 2003-07-21 2005-02-03 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
EP1648418A4 (en) * 2003-07-21 2011-11-16 Middlebrook Pharmaceuticals Inc ANTIBIOTIC PRODUCT, ITS USE AND FORMULATION
CA2533292C (en) 2003-07-21 2013-12-31 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
US8758820B2 (en) * 2003-08-11 2014-06-24 Shionogi Inc. Robust pellet
CA2535398C (en) * 2003-08-12 2013-11-12 Advancis Pharmaceuticals Corporation Antibiotic product, use and formulation thereof
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DE10341264A1 (de) * 2003-09-04 2005-03-24 Grünenthal GmbH Schmelzformulierte, multipartikuläre orale Darreichungsform
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ATE483708T1 (de) 2004-03-08 2010-10-15 Prosidion Ltd Pyrrolopyridin-2-carbonsäurehydrazide als inhibitoren von glykogenphosphorylase
EP1771158A4 (en) * 2004-07-02 2008-03-12 Advancis Pharmaceutical Corp TABLET FOR PULSED DELIVERY
KR100638315B1 (ko) * 2004-07-23 2006-10-25 주식회사 대웅제약 다중 필름 코팅된 코어층을 갖는 클라불라네이트 및아목시실린-함유 유핵정
TWI367755B (en) 2005-05-20 2012-07-11 Sankyo Co Film coated product
KR100780553B1 (ko) * 2005-08-18 2007-11-29 한올제약주식회사 메트포르민 서방정 및 그의 제조방법
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en) * 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
US8299052B2 (en) 2006-05-05 2012-10-30 Shionogi Inc. Pharmaceutical compositions and methods for improved bacterial eradication
CL2008003230A1 (es) * 2007-11-01 2009-11-27 Sanofi Aventis Healthcare Pty Ltd Composicion de recubrimiento de tableta que comprende polimero celulosico, plastificante, edulcorante y composicion de sabor en polvo la que comprende saborizante asociado con portador solido; fluido de recubrimiento de tableta que comprende dicha composicion; tableta farmaceutica; proceso de preparacion de dicha tableta.
NZ617025A (en) * 2009-09-18 2014-03-28 Sanofi Sa (z)-2-cyano-3-hydroxy-but-2-enoic acid-(4’-trifluormethylphenyl)-amide tablet formulations with improved stability
TR200909787A2 (tr) 2009-12-25 2011-07-21 Bi̇lgi̇ç Mahmut Üçüncü kuşak bir sefalosporin ve klavulanik asit içeren farmasötik formülasyonlar.
TR201000687A1 (tr) 2010-01-29 2011-08-22 Bi̇lgi̇ç Mahmut Aktif madde olarak sefiksim ve klavulanik asit içeren efervesan formülasyonlar
TR201000688A2 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Aktif madde olarak sefaklor ve klavulanik asit içeren efervesan formülasyonlar.
TR201000686A1 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Bakteriyel enfeksiyonların tedavisinde suda çözünebilir sefdinir ve klavulanik asit formülasyonları.@
JP6041591B2 (ja) * 2011-09-13 2016-12-14 大日本住友製薬株式会社 イルベサルタンとアムロジピンまたはその塩を含有する安定化された医薬組成物
US9387250B2 (en) 2013-03-15 2016-07-12 Rutgers, The State University Of New Jersey Therapeutic compositions for bone repair

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1241844A (en) 1968-08-23 1971-08-04 Beecham Group Ltd Penicillins
GB1508977A (en) 1974-04-20 1978-04-26 Beecham Group Ltd Beta-lactam antibiotic from streptomyces clavuligerus
US4098897A (en) * 1975-04-14 1978-07-04 Beecham Group Limited Anti bacterial agents
JO984B1 (en) 1977-10-11 1979-12-01 بيتشام غروب ليمتد A dry pharmaceutical compound with a suitable dosage unit for oral administration
NZ198241A (en) * 1980-09-27 1983-12-16 Beecham Group Ltd Tablet containing amoxycillin and potassium clavulanate
DE3266580D1 (en) * 1981-12-02 1985-10-31 Beecham Group Plc Pharmaceutical formulation comprising beta-lactam antibiotics
GB9408117D0 (en) * 1994-04-23 1994-06-15 Smithkline Beecham Corp Pharmaceutical formulations
DK200000133U3 (da) * 1999-04-13 2000-07-28 Beecham Pharm Pte Ltd Ny farmaceutisk formulering
AU2001292185A1 (en) * 2000-10-12 2002-04-22 Beecham Pharmaceuticals (Pte) Limited Formulation containing amoxicillin

Also Published As

Publication number Publication date
JPH09512027A (ja) 1997-12-02
HU228399B1 (en) 2013-03-28
DE69521799T2 (de) 2002-06-13
AU684949B2 (en) 1998-01-08
ES2161288T3 (es) 2001-12-01
DE69528608T2 (de) 2003-06-26
AP564A (en) 1996-11-21
NO964488D0 (no) 1996-10-22
DK1093813T3 (da) 2003-02-17
ATE226074T1 (de) 2002-11-15
DE69521799D1 (de) 2001-08-23
WO1995028927A1 (en) 1995-11-02
DE69528608D1 (de) 2002-11-21
CN1134258C (zh) 2004-01-14
ATE196845T1 (de) 2000-10-15
HK1009936A1 (en) 1999-06-11
DK0761218T3 (da) 2000-12-18
EP0761218A1 (en) 1997-03-12
ATE223706T1 (de) 2002-09-15
US6051255A (en) 2000-04-18
DK0758235T3 (da) 2001-10-29
HK1027024A1 (en) 2001-01-05
DE69519093D1 (de) 2000-11-16
OA10377A (en) 2001-11-21
RO116997B1 (ro) 2001-09-28
AP9600868A0 (en) 1996-10-31
GR3036844T3 (en) 2002-01-31
MY115351A (en) 2003-05-31
ES2152485T3 (es) 2001-02-01
CZ11376U1 (cs) 2001-07-12
CZ294168B6 (cs) 2004-10-13
NZ285080A (en) 1998-05-27
PT758235E (pt) 2001-10-31
NO310703B1 (no) 2001-08-20
HU9602922D0 (en) 1996-12-30
GR3035031T3 (en) 2001-03-30
CN1149829A (zh) 1997-05-14
PL316966A1 (en) 1997-03-03
AP9500733A0 (en) 1995-04-30
EP1243267A3 (en) 2002-10-30
BR9507502A (pt) 1997-09-02
DE69519093T2 (de) 2001-07-19
SA95160343B1 (ar) 2005-05-04
EP0978276A2 (en) 2000-02-09
IL113433A (en) 2003-06-24
EP1093813A3 (en) 2001-05-30
JP3622975B2 (ja) 2005-02-23
IL113433A0 (en) 1995-07-31
DK0978276T3 (da) 2003-01-20
SK135496A3 (en) 1997-05-07
DE29522153U1 (de) 2000-04-06
ES2180251T3 (es) 2003-02-01
BG62842B1 (bg) 2000-09-29
HUT76335A (en) 1997-08-28
CZ309096A3 (en) 1997-04-16
PT761218E (pt) 2001-03-30
ATE203161T1 (de) 2001-08-15
MA23528A1 (fr) 1995-12-31
DE69528204D1 (de) 2002-10-17
ZA953236B (en) 1995-12-27
DE69528204T2 (de) 2003-08-07
CA2188496A1 (en) 1995-11-02
ES2182754T3 (es) 2003-03-16
DZ1876A1 (fr) 2002-02-17
AT5350U1 (de) 2002-06-25
EP0761218B1 (en) 2000-10-11
GB9408117D0 (en) 1994-06-15
SK282594B6 (sk) 2002-10-08
AT5349U1 (de) 2002-06-25
FI964249A (fi) 1996-10-22
NO964488L (no) 1996-12-17
EP1093813A2 (en) 2001-04-25
HK1036404A1 (en) 2002-01-04
EP0758235A1 (en) 1997-02-19
BG100933A (en) 1997-07-31
RU2152213C1 (ru) 2000-07-10
PT1093813E (pt) 2003-02-28
PT978276E (pt) 2003-01-31
AU2406895A (en) 1995-11-16
HK1021860A1 (en) 2000-07-07
EP0978276A3 (en) 2000-04-12
EP1093813B1 (en) 2002-10-16
EP0978276B1 (en) 2002-09-11
SI0758235T1 (en) 2001-10-31
HK1050992A1 (zh) 2003-07-18
EP1243267A2 (en) 2002-09-25
EP0758235B1 (en) 2001-07-18

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