DK0978276T3 - Polymerovertrukken tablet omfattende amoxycillin og clavulanat - Google Patents

Polymerovertrukken tablet omfattende amoxycillin og clavulanat

Info

Publication number
DK0978276T3
DK0978276T3 DK99200891T DK99200891T DK0978276T3 DK 0978276 T3 DK0978276 T3 DK 0978276T3 DK 99200891 T DK99200891 T DK 99200891T DK 99200891 T DK99200891 T DK 99200891T DK 0978276 T3 DK0978276 T3 DK 0978276T3
Authority
DK
Denmark
Prior art keywords
amoxycillin
clavulanate
coated tablet
polymer coated
polymer
Prior art date
Application number
DK99200891T
Other languages
English (en)
Inventor
Creighton Pierce Smithk Conley
Nigel Philip M Smithk Davidson
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10754044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0978276(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Application granted granted Critical
Publication of DK0978276T3 publication Critical patent/DK0978276T3/da

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/2853Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893Tablet coating processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
DK99200891T 1994-04-23 1995-04-19 Polymerovertrukken tablet omfattende amoxycillin og clavulanat DK0978276T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9408117A GB9408117D0 (en) 1994-04-23 1994-04-23 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
DK0978276T3 true DK0978276T3 (da) 2003-01-20

Family

ID=10754044

Family Applications (4)

Application Number Title Priority Date Filing Date
DK00204182T DK1093813T3 (da) 1994-04-23 1995-04-19 Fremgangsmåde til at fremstille polymer-overtrukket tablet, der omfatter amoxycillin og clavunalat, belagt med et vandigt polymerfilmovertræk
DK95917937T DK0758235T3 (da) 1994-04-23 1995-04-19 Polymercoatet tablet omfattende amoxycillin og clavulanat
DK96202848T DK0761218T3 (da) 1994-04-23 1995-04-19 Fremgangsmåde til fremstilling af polymerovertrukne tabletter omfattende amoxycillin og clavulanat
DK99200891T DK0978276T3 (da) 1994-04-23 1995-04-19 Polymerovertrukken tablet omfattende amoxycillin og clavulanat

Family Applications Before (3)

Application Number Title Priority Date Filing Date
DK00204182T DK1093813T3 (da) 1994-04-23 1995-04-19 Fremgangsmåde til at fremstille polymer-overtrukket tablet, der omfatter amoxycillin og clavunalat, belagt med et vandigt polymerfilmovertræk
DK95917937T DK0758235T3 (da) 1994-04-23 1995-04-19 Polymercoatet tablet omfattende amoxycillin og clavulanat
DK96202848T DK0761218T3 (da) 1994-04-23 1995-04-19 Fremgangsmåde til fremstilling af polymerovertrukne tabletter omfattende amoxycillin og clavulanat

Country Status (35)

Country Link
US (1) US6051255A (da)
EP (5) EP0761218B1 (da)
JP (1) JP3622975B2 (da)
CN (1) CN1134258C (da)
AP (2) AP564A (da)
AT (6) ATE223706T1 (da)
AU (1) AU684949B2 (da)
BG (1) BG62842B1 (da)
BR (1) BR9507502A (da)
CA (1) CA2188496A1 (da)
CZ (2) CZ11376U1 (da)
DE (5) DE69519093T2 (da)
DK (4) DK1093813T3 (da)
DZ (1) DZ1876A1 (da)
ES (4) ES2152485T3 (da)
FI (1) FI964249A0 (da)
GB (1) GB9408117D0 (da)
GR (2) GR3035031T3 (da)
HK (5) HK1050992A1 (da)
HU (1) HU228399B1 (da)
IL (1) IL113433A (da)
MA (1) MA23528A1 (da)
MY (1) MY115351A (da)
NO (1) NO310703B1 (da)
NZ (1) NZ285080A (da)
OA (1) OA10377A (da)
PL (1) PL316966A1 (da)
PT (4) PT978276E (da)
RO (1) RO116997B1 (da)
RU (1) RU2152213C1 (da)
SA (1) SA95160343B1 (da)
SI (1) SI0758235T1 (da)
SK (1) SK282594B6 (da)
WO (1) WO1995028927A1 (da)
ZA (1) ZA953236B (da)

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US20030109503A1 (en) * 1995-06-06 2003-06-12 Smithkline Beecham P.L.C. Pharmaceutical formulations comprising clavulanic acid alone or in combination with other beta-lactam antibiotics
ATE208618T1 (de) * 1995-09-07 2001-11-15 Smithkline Beecham Corp Verwendung einer amoxicillin und clavulanat enthaltenden paediatrischen pharmazeutischen formulierung
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TWI225402B (en) 1996-03-13 2004-12-21 Biochemie Gmbh Auxiliary-free agglomerates
GB9613470D0 (en) 1996-06-27 1996-08-28 Ciba Geigy Ag Small solid oral dosage form
GB9616536D0 (en) 1996-08-06 1996-09-25 Quadrant Holdings Cambridge Co-amoxiclav dosage form
GB9617780D0 (en) * 1996-08-24 1996-10-02 Smithkline Beecham Plc Method of treatment
WO1998034598A2 (en) * 1997-02-07 1998-08-13 Gist-Brocades B.V. Homogeneous granulated formulations for dose sipping technology
US20030124187A1 (en) * 1997-02-14 2003-07-03 Smithkline Beecham Laboratoires Pharmaceutiques, Pharmaceutical formulations comprising amoxycillin and clavulanate
ATE243516T1 (de) * 1997-02-14 2003-07-15 Glaxosmithkline Lab Sas Amoxicillin und clavulanat enthaltende arzneizubereitungen
EP1023065A1 (en) * 1997-08-29 2000-08-02 Dsm N.V. Granules free of excipients
WO1999022769A1 (en) 1997-10-31 1999-05-14 Monsanto Company Gellan gum tablet coating
AU3817300A (en) 1999-04-01 2000-08-01 Dsm N.V. Agglomerates by crystallisation
CN100382782C (zh) * 1999-04-13 2008-04-23 比彻姆药品(Pte)有限公司 一种释放改良型药用制剂
US6878386B1 (en) 1999-04-13 2005-04-12 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising amoxycillin and potassium clavulanate
US7250176B1 (en) * 1999-04-13 2007-07-31 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection
US6294199B1 (en) 1999-04-13 2001-09-25 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising administering amoxycillin
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GB9930578D0 (en) * 1999-12-23 2000-02-16 Smithkline Beecham Plc Pharmaceutical formulations
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US6375982B1 (en) * 2000-07-05 2002-04-23 Capricorn Pharma, Inc. Rapid-melt semi-solid compositions, methods of making same and method of using same
US6756057B2 (en) 2000-10-12 2004-06-29 Beecham Pharmaceuticals (Pte) Limited Amoxicillin and potassium clavulanate dosage form
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US6541014B2 (en) * 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US20020068078A1 (en) * 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
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US20030070584A1 (en) * 2001-05-15 2003-04-17 Cynthia Gulian Dip coating compositions containing cellulose ethers
US8309118B2 (en) * 2001-09-28 2012-11-13 Mcneil-Ppc, Inc. Film forming compositions containing sucralose
WO2003066053A1 (en) * 2002-02-07 2003-08-14 Rutgers, The State University Antibiotic polymers
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US7405210B2 (en) 2003-05-21 2008-07-29 Osi Pharmaceuticals, Inc. Pyrrolopyridine-2-carboxylic acid amide inhibitors of glycogen phosphorylase
EP1648407A4 (en) 2003-07-21 2011-08-31 Middlebrook Pharmaceuticals Inc ANTIBIOTIC PRODUCT, CORRESPONDING USE AND FORMULATION
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CL2008003230A1 (es) * 2007-11-01 2009-11-27 Sanofi Aventis Healthcare Pty Ltd Composicion de recubrimiento de tableta que comprende polimero celulosico, plastificante, edulcorante y composicion de sabor en polvo la que comprende saborizante asociado con portador solido; fluido de recubrimiento de tableta que comprende dicha composicion; tableta farmaceutica; proceso de preparacion de dicha tableta.
EP2477611B1 (en) * 2009-09-18 2017-04-05 Sanofi (z)-2-cyano-3-hydroxy-but-2-enoic acid-(4'-trifluormethylphenyl)-amide tablet formulations with improved stability
TR200909787A2 (tr) 2009-12-25 2011-07-21 Bi̇lgi̇ç Mahmut Üçüncü kuşak bir sefalosporin ve klavulanik asit içeren farmasötik formülasyonlar.
TR201000687A1 (tr) 2010-01-29 2011-08-22 Bi̇lgi̇ç Mahmut Aktif madde olarak sefiksim ve klavulanik asit içeren efervesan formülasyonlar
TR201000686A1 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Bakteriyel enfeksiyonların tedavisinde suda çözünebilir sefdinir ve klavulanik asit formülasyonları.@
TR201000688A2 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Aktif madde olarak sefaklor ve klavulanik asit içeren efervesan formülasyonlar.
JP6041591B2 (ja) * 2011-09-13 2016-12-14 大日本住友製薬株式会社 イルベサルタンとアムロジピンまたはその塩を含有する安定化された医薬組成物
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GB1241844A (en) 1968-08-23 1971-08-04 Beecham Group Ltd Penicillins
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JO984B1 (en) 1977-10-11 1979-12-01 بيتشام غروب ليمتد A dry pharmaceutical compound with a suitable dosage unit for oral administration
NZ198241A (en) * 1980-09-27 1983-12-16 Beecham Group Ltd Tablet containing amoxycillin and potassium clavulanate
DE3266580D1 (en) * 1981-12-02 1985-10-31 Beecham Group Plc Pharmaceutical formulation comprising beta-lactam antibiotics
GB9408117D0 (en) * 1994-04-23 1994-06-15 Smithkline Beecham Corp Pharmaceutical formulations
CN100382782C (zh) * 1999-04-13 2008-04-23 比彻姆药品(Pte)有限公司 一种释放改良型药用制剂
EP1330236A2 (en) * 2000-10-12 2003-07-30 Beecham Pharmaceuticals (Pte) Limited Formulation containing amoxicillin

Also Published As

Publication number Publication date
DK0761218T3 (da) 2000-12-18
EP0761218A1 (en) 1997-03-12
PT1093813E (pt) 2003-02-28
CA2188496A1 (en) 1995-11-02
DE69528608T2 (de) 2003-06-26
HK1027024A1 (en) 2001-01-05
DK1093813T3 (da) 2003-02-17
HUT76335A (en) 1997-08-28
ATE223706T1 (de) 2002-09-15
SK282594B6 (sk) 2002-10-08
US6051255A (en) 2000-04-18
MY115351A (en) 2003-05-31
CZ11376U1 (cs) 2001-07-12
GR3036844T3 (en) 2002-01-31
FI964249A (fi) 1996-10-22
NO964488D0 (no) 1996-10-22
PT978276E (pt) 2003-01-31
GB9408117D0 (en) 1994-06-15
EP1093813A2 (en) 2001-04-25
HK1009936A1 (en) 1999-06-11
CZ309096A3 (en) 1997-04-16
PT761218E (pt) 2001-03-30
EP1093813B1 (en) 2002-10-16
NZ285080A (en) 1998-05-27
NO964488L (no) 1996-12-17
HU228399B1 (en) 2013-03-28
IL113433A (en) 2003-06-24
AP564A (en) 1996-11-21
CN1134258C (zh) 2004-01-14
HK1050992A1 (zh) 2003-07-18
ES2161288T3 (es) 2001-12-01
DE69519093T2 (de) 2001-07-19
SI0758235T1 (en) 2001-10-31
ZA953236B (en) 1995-12-27
DK0758235T3 (da) 2001-10-29
EP0761218B1 (en) 2000-10-11
PL316966A1 (en) 1997-03-03
EP0978276A2 (en) 2000-02-09
GR3035031T3 (en) 2001-03-30
HK1036404A1 (en) 2002-01-04
PT758235E (pt) 2001-10-31
DE69528204D1 (de) 2002-10-17
EP1093813A3 (en) 2001-05-30
DE69528204T2 (de) 2003-08-07
RO116997B1 (ro) 2001-09-28
DE69528608D1 (de) 2002-11-21
HU9602922D0 (en) 1996-12-30
HK1021860A1 (en) 2000-07-07
AP9600868A0 (en) 1996-10-31
MA23528A1 (fr) 1995-12-31
AT5349U1 (de) 2002-06-25
AU684949B2 (en) 1998-01-08
SA95160343B1 (ar) 2005-05-04
OA10377A (en) 2001-11-21
DE29522153U1 (de) 2000-04-06
EP1243267A3 (en) 2002-10-30
EP0978276B1 (en) 2002-09-11
FI964249A0 (fi) 1996-10-22
JP3622975B2 (ja) 2005-02-23
ATE226074T1 (de) 2002-11-15
ES2180251T3 (es) 2003-02-01
EP0758235A1 (en) 1997-02-19
EP0978276A3 (en) 2000-04-12
AU2406895A (en) 1995-11-16
BG100933A (en) 1997-07-31
SK135496A3 (en) 1997-05-07
BR9507502A (pt) 1997-09-02
IL113433A0 (en) 1995-07-31
EP1243267A2 (en) 2002-09-25
AT5350U1 (de) 2002-06-25
DE69519093D1 (de) 2000-11-16
ES2152485T3 (es) 2001-02-01
AP9500733A0 (en) 1995-04-30
ATE203161T1 (de) 2001-08-15
CZ294168B6 (cs) 2004-10-13
ATE196845T1 (de) 2000-10-15
ES2182754T3 (es) 2003-03-16
NO310703B1 (no) 2001-08-20
DZ1876A1 (fr) 2002-02-17
JPH09512027A (ja) 1997-12-02
EP0758235B1 (en) 2001-07-18
BG62842B1 (bg) 2000-09-29
RU2152213C1 (ru) 2000-07-10
DE69521799D1 (de) 2001-08-23
WO1995028927A1 (en) 1995-11-02
CN1149829A (zh) 1997-05-14
DE69521799T2 (de) 2002-06-13

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