FI945378A0 - Bombesiinin polypeptidiantagonistit - Google Patents

Bombesiinin polypeptidiantagonistit

Info

Publication number
FI945378A0
FI945378A0 FI945378A FI945378A FI945378A0 FI 945378 A0 FI945378 A0 FI 945378A0 FI 945378 A FI945378 A FI 945378A FI 945378 A FI945378 A FI 945378A FI 945378 A0 FI945378 A0 FI 945378A0
Authority
FI
Finland
Prior art keywords
phenyl
alkyl
hydrogen
moiety
10alkyl
Prior art date
Application number
FI945378A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI945378A (fi
Inventor
Andrew Victor Schally
Ren Zhi Cai
Original Assignee
Univ Tulane
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Tulane filed Critical Univ Tulane
Publication of FI945378A0 publication Critical patent/FI945378A0/fi
Publication of FI945378A publication Critical patent/FI945378A/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • C07K7/086—Bombesin; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/02—Peptides of undefined number of amino acids; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
FI945378A 1993-03-15 1994-11-15 Bombesiinin polypeptidiantagonistit FI945378A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/031,325 US5369094A (en) 1990-11-29 1993-03-15 Polypeptide bombesin antagonists
PCT/US1994/002511 WO1994021674A1 (en) 1993-03-15 1994-03-07 Polypeptide bombesin antagonists

Publications (2)

Publication Number Publication Date
FI945378A0 true FI945378A0 (fi) 1994-11-15
FI945378A FI945378A (fi) 1994-11-15

Family

ID=21858823

Family Applications (1)

Application Number Title Priority Date Filing Date
FI945378A FI945378A (fi) 1993-03-15 1994-11-15 Bombesiinin polypeptidiantagonistit

Country Status (27)

Country Link
US (1) US5369094A (sl)
EP (1) EP0646127B1 (sl)
JP (1) JP3838656B2 (sl)
KR (1) KR100306506B1 (sl)
AT (1) ATE167874T1 (sl)
AU (1) AU666270B2 (sl)
BR (1) BR9404341A (sl)
CA (1) CA2135787C (sl)
CZ (1) CZ286750B6 (sl)
DE (1) DE69411342T2 (sl)
DK (1) DK0646127T3 (sl)
EE (1) EE03180B1 (sl)
ES (1) ES2120615T3 (sl)
FI (1) FI945378A (sl)
HR (1) HRP940164B1 (sl)
HU (1) HU218288B (sl)
IL (2) IL108851A (sl)
NO (1) NO313418B1 (sl)
NZ (2) NZ299913A (sl)
PL (1) PL180372B1 (sl)
RU (1) RU2114118C1 (sl)
SI (1) SI9420001B (sl)
SK (1) SK282267B6 (sl)
TW (1) TW325478B (sl)
UA (1) UA34456C2 (sl)
WO (1) WO1994021674A1 (sl)
ZA (1) ZA941767B (sl)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5877277A (en) 1987-09-24 1999-03-02 Biomeasure, Inc. Octapeptide bombesin analogs
US5723578A (en) * 1987-09-24 1998-03-03 The Administrators Of Tulane Educational Fund Peptide analogs of bombesin
US5650395A (en) * 1995-03-13 1997-07-22 Hurel; Steven Treatment of pulmonary hypertension
US6989371B1 (en) 1996-08-16 2006-01-24 Dabur Research Foundation Bombesin analogs for treatment of cancer
US6200546B1 (en) 1997-04-22 2001-03-13 The Curators Of The University Of Missouri Gastrin receptor-avid peptide conjugates
JP2004525864A (ja) * 2000-11-17 2004-08-26 ワーナー−ランバート カンパニー リミティド ライアビリティー カンパニー ボンベシンアンタゴニストを用いた性機能障害の治療
US7850947B2 (en) * 2003-01-13 2010-12-14 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
EP1583564B1 (en) * 2003-01-13 2009-07-01 Bracco Imaging S.p.A Improved linkers for radiopharmaceutical compounds
US8420050B2 (en) * 2003-01-13 2013-04-16 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
US7611692B2 (en) * 2003-01-13 2009-11-03 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
US7922998B2 (en) * 2003-01-13 2011-04-12 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
US20060239923A1 (en) * 2003-01-13 2006-10-26 Bracco Imaging S.P.A. Gastrin releasing peptide compounds
US7226577B2 (en) * 2003-01-13 2007-06-05 Bracco Imaging, S. P. A. Gastrin releasing peptide compounds
AU2004232314B2 (en) 2003-04-22 2007-11-22 Ipsen Pharma S.A.S. Peptide vectors
US7795385B2 (en) * 2004-12-17 2010-09-14 Bexar Global, Inc. Use of bombesin/gastrin-releasing peptide antagonists for the treatment of inflammatory conditions, acute lung injury and bipolar disorder
FR2918566B1 (fr) * 2007-07-11 2009-10-09 Pierre Fabre Medicament Sa Composition pharmaceutique stable d'un sel hydrosoluble de vinflunine.
EP2100900A1 (en) * 2008-03-07 2009-09-16 Universitätsspital Basel Bombesin analog peptide antagonist conjugates
EP2198878A1 (en) * 2008-12-18 2010-06-23 University Of Miami Polypeptide bombesin antagonists
WO2011043954A1 (en) 2009-10-07 2011-04-14 Merck Sharp & Dohme Corp. Novel trpa1 antagonists

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5162497A (en) * 1987-09-24 1992-11-10 The Administrators Of The Tulane Educational Fund Bradykinin analogs with non-peptide bond
WO1989002897A1 (en) * 1987-09-24 1989-04-06 The Administrators Of The Tulane Educational Fund Therapeutic peptides
US5084555A (en) * 1989-08-21 1992-01-28 The Administrators Of The Tulane Educational Fund An octapeptide bombesin analog
AU618029B2 (en) * 1987-11-02 1991-12-12 Imperial Chemical Industries Plc Polypeptide compounds
GB8813356D0 (en) * 1988-06-06 1988-07-13 Ici Plc Polypeptide compounds
GR1000608B (el) * 1988-07-21 1992-08-31 Erba Carlo Spa Μεθοδος για την παρασκευη ανταγωνιστων bombesin.
JP2919889B2 (ja) * 1988-10-14 1999-07-19 アドミニストレイターズ オブ ザ テューレイン エデュケイショナル ファンド 治療用ペプチド
US5217955A (en) * 1989-09-15 1993-06-08 Biomeasure, Inc. Treatment of cancer with peptide analog of bombesin, grp, litorin or neuromedin
US5244883A (en) * 1990-11-29 1993-09-14 The Administrators Of The Tulane Educational Fund Nonapeptide bombesin antagonists

Also Published As

Publication number Publication date
HRP940164A2 (en) 1996-08-31
ZA941767B (en) 1994-10-06
PL180372B1 (pl) 2001-01-31
IL108851A0 (en) 1994-06-24
ATE167874T1 (de) 1998-07-15
SK136494A3 (en) 1995-08-09
CZ280794A3 (en) 1995-07-12
KR100306506B1 (ko) 2001-12-01
NO313418B1 (no) 2002-09-30
AU666270B2 (en) 1996-02-01
ES2120615T3 (es) 1998-11-01
UA34456C2 (uk) 2001-03-15
JP3838656B2 (ja) 2006-10-25
DE69411342D1 (de) 1998-08-06
SI9420001A (en) 1995-08-31
HRP940164B1 (en) 2000-02-29
KR950701646A (ko) 1995-04-28
DK0646127T3 (da) 1999-04-12
EP0646127A1 (en) 1995-04-05
IL108851A (en) 2003-05-29
NO944293D0 (no) 1994-11-10
PL306209A1 (en) 1995-03-06
RU2114118C1 (ru) 1998-06-27
HU218288B (en) 2000-07-28
JPH07507330A (ja) 1995-08-10
CZ286750B6 (en) 2000-06-14
US5369094A (en) 1994-11-29
IL154995A0 (en) 2003-10-31
RU94046091A (ru) 1996-09-27
WO1994021674A1 (en) 1994-09-29
HUT69727A (en) 1995-09-28
NO944293L (no) 1995-01-02
EP0646127B1 (en) 1998-07-01
CA2135787C (en) 2008-08-12
DE69411342T2 (de) 1998-11-19
CA2135787A1 (en) 1994-09-29
TW325478B (en) 1998-01-21
BR9404341A (pt) 1999-08-31
FI945378A (fi) 1994-11-15
SK282267B6 (sk) 2001-12-03
AU6444694A (en) 1994-10-11
NZ299913A (en) 2000-07-28
EE03180B1 (et) 1999-04-15
NZ263668A (en) 1997-06-24
SI9420001B (sl) 1999-08-31

Similar Documents

Publication Publication Date Title
FI945378A0 (fi) Bombesiinin polypeptidiantagonistit
SE9604341D0 (sv) Hepta-peptide oxytocin analogue
CA2097192A1 (en) Bombesin antagonists
AR034132A1 (es) Analogos de somatostatina, un proceso para su produccion y composicion farmaceutica
HUP0003592A2 (hu) LH-RH peptid analógok, alkalmazásuk, és ezeket tartalmazó gyógyászati készítmények
IT1244501B (it) Derivati amminoacilici e oligopeptidici dell'allopurinolo dotati di attivita' immunostimolante e composizioni farmaceutiche che li contengono
GB1533077A (en) 4-substituted enkephalin derivatives
ES460618A1 (es) Procedimiento para la preparacion de derivados de peptido
GB1224576A (en) Novel tetrapeptide amides and the preparation thereof
GB1363801A (en) Peptides and their preparation
GB1357121A (en) Peptide enzyme inhibitors
ES416516A1 (es) Un procedimiento para la preparacion de nonapeptidos.
GB1273873A (en) Corticotropically highly active octadecapeptides
GB1269898A (en) Amino acid derivatives
ES248724A1 (es) Procedimiento para la obtenciën de nuevosdecapeptures ciclicos
TW340849B (en) Novel cyclopeptides and pharmaceutical compositions as integrin inhibitors comprizing the same
TH17064B (th) ตัวปฏิปักษ์ต่อโปลีเปปไทด์บอมเบซิน
GB1039536A (en) Manufacture of highly active isomers of hypertensin ó and of its analogues