EE03180B1 - Bombesiini antagonistpeptiidid, farmatseutiline kompositsioon ja kasutamine - Google Patents
Bombesiini antagonistpeptiidid, farmatseutiline kompositsioon ja kasutamineInfo
- Publication number
- EE03180B1 EE03180B1 EE9400166A EE9400166A EE03180B1 EE 03180 B1 EE03180 B1 EE 03180B1 EE 9400166 A EE9400166 A EE 9400166A EE 9400166 A EE9400166 A EE 9400166A EE 03180 B1 EE03180 B1 EE 03180B1
- Authority
- EE
- Estonia
- Prior art keywords
- phenyl
- alkyl
- hydrogen
- moiety
- 10alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
- C07K7/086—Bombesin; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/02—Peptides of undefined number of amino acids; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- Genetics & Genomics (AREA)
- Animal Behavior & Ethology (AREA)
- Biophysics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Enzymes And Modification Thereof (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/031,325 US5369094A (en) | 1990-11-29 | 1993-03-15 | Polypeptide bombesin antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
EE03180B1 true EE03180B1 (et) | 1999-04-15 |
Family
ID=21858823
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EE9400166A EE03180B1 (et) | 1993-03-15 | 1994-11-23 | Bombesiini antagonistpeptiidid, farmatseutiline kompositsioon ja kasutamine |
Country Status (27)
Country | Link |
---|---|
US (1) | US5369094A (et) |
EP (1) | EP0646127B1 (et) |
JP (1) | JP3838656B2 (et) |
KR (1) | KR100306506B1 (et) |
AT (1) | ATE167874T1 (et) |
AU (1) | AU666270B2 (et) |
BR (1) | BR9404341A (et) |
CA (1) | CA2135787C (et) |
CZ (1) | CZ286750B6 (et) |
DE (1) | DE69411342T2 (et) |
DK (1) | DK0646127T3 (et) |
EE (1) | EE03180B1 (et) |
ES (1) | ES2120615T3 (et) |
FI (1) | FI945378A (et) |
HR (1) | HRP940164B1 (et) |
HU (1) | HU218288B (et) |
IL (2) | IL108851A (et) |
NO (1) | NO313418B1 (et) |
NZ (2) | NZ299913A (et) |
PL (1) | PL180372B1 (et) |
RU (1) | RU2114118C1 (et) |
SI (1) | SI9420001B (et) |
SK (1) | SK282267B6 (et) |
TW (1) | TW325478B (et) |
UA (1) | UA34456C2 (et) |
WO (1) | WO1994021674A1 (et) |
ZA (1) | ZA941767B (et) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5877277A (en) | 1987-09-24 | 1999-03-02 | Biomeasure, Inc. | Octapeptide bombesin analogs |
US5723578A (en) * | 1987-09-24 | 1998-03-03 | The Administrators Of Tulane Educational Fund | Peptide analogs of bombesin |
US5650395A (en) * | 1995-03-13 | 1997-07-22 | Hurel; Steven | Treatment of pulmonary hypertension |
US6989371B1 (en) | 1996-08-16 | 2006-01-24 | Dabur Research Foundation | Bombesin analogs for treatment of cancer |
DE69840647D1 (de) | 1997-04-22 | 2009-04-23 | Curator Of The University Of M | Konjugate aus peptiden, die liganden von gastrinrezeptoren sind |
KR20040062416A (ko) * | 2000-11-17 | 2004-07-07 | 워너-램버트 캄파니 엘엘씨 | 봄베신 길항제를 이용한 성기능 장애의 치료 |
ATE435035T1 (de) * | 2003-01-13 | 2009-07-15 | Bracco Imaging Spa | Verbesserte linker für radiopharmazeutische verbindungen |
US7922998B2 (en) * | 2003-01-13 | 2011-04-12 | Bracco Imaging S.P.A. | Gastrin releasing peptide compounds |
US7850947B2 (en) * | 2003-01-13 | 2010-12-14 | Bracco Imaging S.P.A. | Gastrin releasing peptide compounds |
US20060239923A1 (en) * | 2003-01-13 | 2006-10-26 | Bracco Imaging S.P.A. | Gastrin releasing peptide compounds |
US7611692B2 (en) | 2003-01-13 | 2009-11-03 | Bracco Imaging S.P.A. | Gastrin releasing peptide compounds |
US7226577B2 (en) * | 2003-01-13 | 2007-06-05 | Bracco Imaging, S. P. A. | Gastrin releasing peptide compounds |
US8420050B2 (en) * | 2003-01-13 | 2013-04-16 | Bracco Imaging S.P.A. | Gastrin releasing peptide compounds |
US8709998B2 (en) | 2003-04-22 | 2014-04-29 | Ipsen Pharma S.A.S. | Peptide vectors |
US7795385B2 (en) * | 2004-12-17 | 2010-09-14 | Bexar Global, Inc. | Use of bombesin/gastrin-releasing peptide antagonists for the treatment of inflammatory conditions, acute lung injury and bipolar disorder |
FR2918566B1 (fr) * | 2007-07-11 | 2009-10-09 | Pierre Fabre Medicament Sa | Composition pharmaceutique stable d'un sel hydrosoluble de vinflunine. |
EP2100900A1 (en) * | 2008-03-07 | 2009-09-16 | Universitätsspital Basel | Bombesin analog peptide antagonist conjugates |
EP2198878A1 (en) * | 2008-12-18 | 2010-06-23 | University Of Miami | Polypeptide bombesin antagonists |
JP2013507364A (ja) | 2009-10-07 | 2013-03-04 | メルク・シャープ・エンド・ドーム・コーポレイション | 新規なtrpa1アンタゴニスト |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5084555A (en) * | 1989-08-21 | 1992-01-28 | The Administrators Of The Tulane Educational Fund | An octapeptide bombesin analog |
JP2795449B2 (ja) * | 1987-09-24 | 1998-09-10 | ジ・アドミニストレーターズ・オブ・ザ・ツーレイン・エデュケイショナル・ファンド | 治療用ペプチド |
US5162497A (en) * | 1987-09-24 | 1992-11-10 | The Administrators Of The Tulane Educational Fund | Bradykinin analogs with non-peptide bond |
AU618029B2 (en) * | 1987-11-02 | 1991-12-12 | Imperial Chemical Industries Plc | Polypeptide compounds |
GB8813356D0 (en) * | 1988-06-06 | 1988-07-13 | Ici Plc | Polypeptide compounds |
GR1000608B (el) * | 1988-07-21 | 1992-08-31 | Erba Carlo Spa | Μεθοδος για την παρασκευη ανταγωνιστων bombesin. |
HU208439B (en) * | 1988-10-14 | 1993-10-28 | Univ Tulane | Process for producing pharmaceutical peptides |
US5217955A (en) * | 1989-09-15 | 1993-06-08 | Biomeasure, Inc. | Treatment of cancer with peptide analog of bombesin, grp, litorin or neuromedin |
US5244883A (en) * | 1990-11-29 | 1993-09-14 | The Administrators Of The Tulane Educational Fund | Nonapeptide bombesin antagonists |
-
1993
- 1993-03-15 US US08/031,325 patent/US5369094A/en not_active Expired - Lifetime
-
1994
- 1994-02-23 TW TW083101048A patent/TW325478B/zh not_active IP Right Cessation
- 1994-03-03 IL IL10885194A patent/IL108851A/xx not_active IP Right Cessation
- 1994-03-07 NZ NZ299913A patent/NZ299913A/en not_active IP Right Cessation
- 1994-03-07 CZ CZ19942807A patent/CZ286750B6/cs not_active IP Right Cessation
- 1994-03-07 WO PCT/US1994/002511 patent/WO1994021674A1/en active IP Right Grant
- 1994-03-07 DE DE69411342T patent/DE69411342T2/de not_active Expired - Fee Related
- 1994-03-07 HU HU9403244A patent/HU218288B/hu not_active IP Right Cessation
- 1994-03-07 RU RU94046091A patent/RU2114118C1/ru not_active IP Right Cessation
- 1994-03-07 BR BR9404341-8A patent/BR9404341A/pt not_active Application Discontinuation
- 1994-03-07 SK SK1364-94A patent/SK282267B6/sk unknown
- 1994-03-07 JP JP52109194A patent/JP3838656B2/ja not_active Expired - Fee Related
- 1994-03-07 ES ES94912199T patent/ES2120615T3/es not_active Expired - Lifetime
- 1994-03-07 EP EP94912199A patent/EP0646127B1/en not_active Expired - Lifetime
- 1994-03-07 UA UA94119008A patent/UA34456C2/uk unknown
- 1994-03-07 CA CA002135787A patent/CA2135787C/en not_active Expired - Fee Related
- 1994-03-07 DK DK94912199T patent/DK0646127T3/da active
- 1994-03-07 AT AT94912199T patent/ATE167874T1/de not_active IP Right Cessation
- 1994-03-07 SI SI9420001A patent/SI9420001B/sl not_active IP Right Cessation
- 1994-03-07 KR KR1019940704104A patent/KR100306506B1/ko not_active IP Right Cessation
- 1994-03-07 AU AU64446/94A patent/AU666270B2/en not_active Ceased
- 1994-03-07 PL PL94306209A patent/PL180372B1/pl not_active IP Right Cessation
- 1994-03-07 NZ NZ263668A patent/NZ263668A/en unknown
- 1994-03-10 HR HR08/031,325A patent/HRP940164B1/xx not_active IP Right Cessation
- 1994-03-14 ZA ZA941767A patent/ZA941767B/xx unknown
- 1994-11-10 NO NO19944293A patent/NO313418B1/no unknown
- 1994-11-15 FI FI945378A patent/FI945378A/fi unknown
- 1994-11-23 EE EE9400166A patent/EE03180B1/et not_active IP Right Cessation
-
2003
- 2003-03-19 IL IL15499503A patent/IL154995A0/xx unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EE03180B1 (et) | Bombesiini antagonistpeptiidid, farmatseutiline kompositsioon ja kasutamine | |
CA2097192A1 (en) | Bombesin antagonists | |
AR034132A1 (es) | Analogos de somatostatina, un proceso para su produccion y composicion farmaceutica | |
TW343198B (en) | Cyclopeptides useful as adhesion inhibitors, process for the preparation thereof, and pharmaceutical composition containing them | |
HUP0003592A2 (hu) | LH-RH peptid analógok, alkalmazásuk, és ezeket tartalmazó gyógyászati készítmények | |
GB1533077A (en) | 4-substituted enkephalin derivatives | |
ES460618A1 (es) | Procedimiento para la preparacion de derivados de peptido | |
GB1357121A (en) | Peptide enzyme inhibitors | |
GB1224576A (en) | Novel tetrapeptide amides and the preparation thereof | |
SE9901773D0 (sv) | Förebyggande av karies i tänderna | |
GB1363801A (en) | Peptides and their preparation | |
ES416516A1 (es) | Un procedimiento para la preparacion de nonapeptidos. | |
GB1273873A (en) | Corticotropically highly active octadecapeptides | |
GB1269898A (en) | Amino acid derivatives | |
ES248724A1 (es) | Procedimiento para la obtenciën de nuevosdecapeptures ciclicos | |
TH17064B (th) | ตัวปฏิปักษ์ต่อโปลีเปปไทด์บอมเบซิน | |
TW340849B (en) | Novel cyclopeptides and pharmaceutical compositions as integrin inhibitors comprizing the same | |
FR4219M (et) | ||
TH35998A (th) | Lh-rh เป็ปไทด์ อะนาล็อก ประโยชน์ของสิ่งเหล่านั้นและองค์ประกอบทางเภสัชกรรมซึ่งประกอบด้วยสิ่งเหล่านั้น |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
KB4A | Valid patent at the end of a year |
Effective date: 20021231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20031231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20041231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20051231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20061231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20071231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20081231 |
|
MM4A | Lapsed by not paying the annual fees |
Effective date: 20081123 |