FI115629B - Menetelmä entsyymi-inhibiittorien valmistamiseksi - Google Patents
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- FI115629B FI115629B FI962315A FI962315A FI115629B FI 115629 B FI115629 B FI 115629B FI 962315 A FI962315 A FI 962315A FI 962315 A FI962315 A FI 962315A FI 115629 B FI115629 B FI 115629B
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Classifications
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- C—CHEMISTRY; METALLURGY
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- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
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- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
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- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
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Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
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| GB9324803 | 1993-12-03 | ||
| GB939324803A GB9324803D0 (en) | 1993-12-03 | 1993-12-03 | Enzyme inhibitors |
| GB9324981 | 1993-12-06 | ||
| GB939324981A GB9324981D0 (en) | 1993-12-06 | 1993-12-06 | Enzyme inhibitors |
| GB9402615 | 1994-11-30 | ||
| PCT/GB1994/002615 WO1995015309A1 (en) | 1993-12-03 | 1994-11-30 | Dp-iv-serine protease inhibitors |
Publications (3)
| Publication Number | Publication Date |
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| FI962315A0 FI962315A0 (fi) | 1996-06-03 |
| FI962315A FI962315A (fi) | 1996-08-05 |
| FI115629B true FI115629B (fi) | 2005-06-15 |
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| Application Number | Title | Priority Date | Filing Date |
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| FI962315A FI115629B (fi) | 1993-12-03 | 1996-06-03 | Menetelmä entsyymi-inhibiittorien valmistamiseksi |
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| US (2) | US5939560A (ko) |
| EP (1) | EP0731789A1 (ko) |
| JP (1) | JP3970317B2 (ko) |
| KR (1) | KR100347828B1 (ko) |
| CN (1) | CN1079792C (ko) |
| AU (1) | AU1113395A (ko) |
| CA (1) | CA2178066A1 (ko) |
| CZ (1) | CZ289931B6 (ko) |
| FI (1) | FI115629B (ko) |
| HU (1) | HUT76274A (ko) |
| IL (1) | IL111785A0 (ko) |
| NO (1) | NO306458B1 (ko) |
| PL (1) | PL182723B1 (ko) |
| WO (1) | WO1995015309A1 (ko) |
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| US3639382A (en) * | 1967-12-22 | 1972-02-01 | Merck & Co Inc | O-ethyl threonine derivatives |
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| DE69124371T2 (de) * | 1990-04-14 | 1997-06-12 | New England Medical Center Inc | Typ-iv-dipeptidyl-aminopeptidase-inhibitoren |
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| CA2121369C (en) * | 1991-10-22 | 2003-04-29 | William W. Bachovchin | Inhibitors of dipeptidyl-aminopeptidase type iv |
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1994
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- 1994-11-30 PL PL94314838A patent/PL182723B1/pl not_active IP Right Cessation
- 1994-11-30 CA CA002178066A patent/CA2178066A1/en not_active Abandoned
- 1994-11-30 CZ CZ19961595A patent/CZ289931B6/cs not_active IP Right Cessation
- 1994-11-30 EP EP95902193A patent/EP0731789A1/en not_active Withdrawn
- 1994-11-30 US US08/647,887 patent/US5939560A/en not_active Expired - Fee Related
- 1994-11-30 HU HU9601508A patent/HUT76274A/hu unknown
- 1994-11-30 AU AU11133/95A patent/AU1113395A/en not_active Abandoned
- 1994-11-30 JP JP51547795A patent/JP3970317B2/ja not_active Expired - Fee Related
- 1994-11-30 KR KR1019960702901A patent/KR100347828B1/ko not_active IP Right Cessation
- 1994-11-30 CN CN94194782A patent/CN1079792C/zh not_active Expired - Fee Related
- 1994-11-30 WO PCT/GB1994/002615 patent/WO1995015309A1/en active IP Right Grant
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1996
- 1996-05-31 NO NO962269A patent/NO306458B1/no unknown
- 1996-06-03 FI FI962315A patent/FI115629B/fi not_active IP Right Cessation
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1999
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Also Published As
| Publication number | Publication date |
|---|---|
| US5939560A (en) | 1999-08-17 |
| HUT76274A (en) | 1997-07-28 |
| CN1141033A (zh) | 1997-01-22 |
| PL182723B1 (pl) | 2002-02-28 |
| NO962269L (no) | 1996-07-30 |
| JPH09509921A (ja) | 1997-10-07 |
| FI962315A (fi) | 1996-08-05 |
| JP3970317B2 (ja) | 2007-09-05 |
| PL314838A1 (en) | 1996-09-30 |
| NO962269D0 (no) | 1996-05-31 |
| US6201132B1 (en) | 2001-03-13 |
| CZ289931B6 (cs) | 2002-04-17 |
| WO1995015309A1 (en) | 1995-06-08 |
| FI962315A0 (fi) | 1996-06-03 |
| AU1113395A (en) | 1995-06-19 |
| IL111785A0 (en) | 1995-01-24 |
| CN1079792C (zh) | 2002-02-27 |
| HU9601508D0 (en) | 1996-07-29 |
| KR100347828B1 (ko) | 2003-01-06 |
| CZ159596A3 (en) | 1997-01-15 |
| EP0731789A1 (en) | 1996-09-18 |
| NO306458B1 (no) | 1999-11-08 |
| CA2178066A1 (en) | 1995-06-08 |
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