ES2713952T3 - Análogos de glucagón que muestran actividad de receptor de GIP - Google Patents
Análogos de glucagón que muestran actividad de receptor de GIP Download PDFInfo
- Publication number
- ES2713952T3 ES2713952T3 ES11808086T ES11808086T ES2713952T3 ES 2713952 T3 ES2713952 T3 ES 2713952T3 ES 11808086 T ES11808086 T ES 11808086T ES 11808086 T ES11808086 T ES 11808086T ES 2713952 T3 ES2713952 T3 ES 2713952T3
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- Prior art keywords
- amino acid
- peptide
- seq
- alkyl
- glucagon
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Classifications
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Diabetes (AREA)
- Toxicology (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Nutrition Science (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Child & Adolescent Psychology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Surgical Instruments (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201061426285P | 2010-12-22 | 2010-12-22 | |
| US201161514609P | 2011-08-03 | 2011-08-03 | |
| PCT/US2011/066164 WO2012088116A2 (en) | 2010-12-22 | 2011-12-20 | Glucagon analogs exhibiting gip receptor activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2713952T3 true ES2713952T3 (es) | 2019-05-24 |
Family
ID=45476658
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES11808086T Active ES2713952T3 (es) | 2010-12-22 | 2011-12-20 | Análogos de glucagón que muestran actividad de receptor de GIP |
Country Status (22)
| Country | Link |
|---|---|
| US (4) | US8507428B2 (OSRAM) |
| EP (1) | EP2654773B1 (OSRAM) |
| JP (1) | JP6086067B2 (OSRAM) |
| KR (1) | KR20130132931A (OSRAM) |
| CN (1) | CN103458920B (OSRAM) |
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| AU (1) | AU2011349331A1 (OSRAM) |
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-
2011
- 2011-12-20 WO PCT/US2011/066164 patent/WO2012088116A2/en not_active Ceased
- 2011-12-20 AU AU2011349331A patent/AU2011349331A1/en not_active Abandoned
- 2011-12-20 ES ES11808086T patent/ES2713952T3/es active Active
- 2011-12-20 NZ NZ612297A patent/NZ612297A/en not_active IP Right Cessation
- 2011-12-20 MA MA36136A patent/MA34885B1/fr unknown
- 2011-12-20 CN CN201180068157.2A patent/CN103458920B/zh not_active Expired - Fee Related
- 2011-12-20 CA CA2821766A patent/CA2821766A1/en not_active Abandoned
- 2011-12-20 EP EP11808086.0A patent/EP2654773B1/en not_active Not-in-force
- 2011-12-20 PE PE2013001437A patent/PE20140186A1/es not_active Application Discontinuation
- 2011-12-20 JP JP2013546329A patent/JP6086067B2/ja not_active Expired - Fee Related
- 2011-12-20 PH PH1/2013/501215A patent/PH12013501215A1/en unknown
- 2011-12-20 BR BR112013015389A patent/BR112013015389A2/pt unknown
- 2011-12-20 US US13/331,816 patent/US8507428B2/en not_active Expired - Fee Related
- 2011-12-20 SG SG2013046412A patent/SG191194A1/en unknown
- 2011-12-20 EA EA201390941A patent/EA201390941A1/ru unknown
- 2011-12-20 KR KR1020137018994A patent/KR20130132931A/ko not_active Withdrawn
- 2011-12-20 MX MX2013006304A patent/MX2013006304A/es not_active Application Discontinuation
- 2011-12-21 AR ARP110104846A patent/AR084459A1/es not_active Application Discontinuation
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2012
- 2012-12-27 US US13/728,110 patent/US9249206B2/en not_active Expired - Fee Related
-
2013
- 2013-06-18 CO CO13145190A patent/CO6761302A2/es unknown
- 2013-06-18 CL CL2013001783A patent/CL2013001783A1/es unknown
- 2013-06-18 CR CR20130295A patent/CR20130295A/es not_active Application Discontinuation
- 2013-06-18 EC ECSP13012697 patent/ECSP13012697A/es unknown
-
2015
- 2015-03-23 US US14/665,508 patent/US20150259393A1/en not_active Abandoned
- 2015-12-28 US US14/981,187 patent/US9587005B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| JP2014507402A (ja) | 2014-03-27 |
| PE20140186A1 (es) | 2014-02-13 |
| US9249206B2 (en) | 2016-02-02 |
| WO2012088116A2 (en) | 2012-06-28 |
| US8507428B2 (en) | 2013-08-13 |
| CA2821766A1 (en) | 2012-06-28 |
| AU2011349331A1 (en) | 2013-07-11 |
| KR20130132931A (ko) | 2013-12-05 |
| MX2013006304A (es) | 2013-07-02 |
| US20160115215A1 (en) | 2016-04-28 |
| EP2654773B1 (en) | 2018-10-03 |
| NZ612297A (en) | 2015-10-30 |
| US20150259393A1 (en) | 2015-09-17 |
| WO2012088116A3 (en) | 2012-11-15 |
| US9587005B2 (en) | 2017-03-07 |
| BR112013015389A2 (pt) | 2016-11-22 |
| US20120238493A1 (en) | 2012-09-20 |
| CN103458920B (zh) | 2016-07-06 |
| AR084459A1 (es) | 2013-05-15 |
| MA34885B1 (fr) | 2014-02-01 |
| JP6086067B2 (ja) | 2017-03-01 |
| ECSP13012697A (es) | 2013-10-31 |
| EP2654773A2 (en) | 2013-10-30 |
| CL2013001783A1 (es) | 2014-01-24 |
| US20130116173A1 (en) | 2013-05-09 |
| CR20130295A (es) | 2013-10-09 |
| SG191194A1 (en) | 2013-07-31 |
| PH12013501215A1 (en) | 2013-11-18 |
| CO6761302A2 (es) | 2013-09-30 |
| EA201390941A1 (ru) | 2013-12-30 |
| CN103458920A (zh) | 2013-12-18 |
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