AU2011349331A1 - Glucagon analogs exhibiting GIP receptor activity - Google Patents
Glucagon analogs exhibiting GIP receptor activity Download PDFInfo
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- AU2011349331A1 AU2011349331A1 AU2011349331A AU2011349331A AU2011349331A1 AU 2011349331 A1 AU2011349331 A1 AU 2011349331A1 AU 2011349331 A AU2011349331 A AU 2011349331A AU 2011349331 A AU2011349331 A AU 2011349331A AU 2011349331 A1 AU2011349331 A1 AU 2011349331A1
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- amino acid
- peptide
- seq
- glucagon analog
- optionally
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Classifications
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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| US201061426285P | 2010-12-22 | 2010-12-22 | |
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| US201161514609P | 2011-08-03 | 2011-08-03 | |
| US61/514,609 | 2011-08-03 | ||
| PCT/US2011/066164 WO2012088116A2 (en) | 2010-12-22 | 2011-12-20 | Glucagon analogs exhibiting gip receptor activity |
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| AU2011349331A Abandoned AU2011349331A1 (en) | 2010-12-22 | 2011-12-20 | Glucagon analogs exhibiting GIP receptor activity |
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| PH (1) | PH12013501215A1 (OSRAM) |
| SG (1) | SG191194A1 (OSRAM) |
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| WO2012088116A2 (en) * | 2010-12-22 | 2012-06-28 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting gip receptor activity |
| US8975223B2 (en) * | 2010-12-22 | 2015-03-10 | Marcadia Biotech, Inc. | Methods for treating metabolic disorders and obesity with a peptide comprising the amino acid sequence of SEQ ID No. 146 |
| PH12013502671A1 (en) | 2011-06-22 | 2022-04-08 | Univ Indiana Res & Tech Corp | Glucagon/glp-1 receptor co-agonists |
| CN104093735B (zh) | 2011-09-23 | 2018-07-06 | 诺沃—诺迪斯克有限公司 | 新的胰高血糖素类似物 |
| US9340600B2 (en) * | 2012-06-21 | 2016-05-17 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting GIP receptor activity |
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| HUE033371T2 (en) | 2013-03-21 | 2017-11-28 | Sanofi Aventis Deutschland | Process for the preparation of peptide products containing a ring imide |
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| KR20130111923A (ko) | 2010-05-13 | 2013-10-11 | 인디애나 유니버시티 리서치 앤드 테크놀로지 코퍼레이션 | G-단백결합 수용체 활성을 나타내는 글루카곤 슈퍼패밀리 펩티드 |
| CA2796894A1 (en) | 2010-06-24 | 2011-12-29 | Indiana University Research And Technology Corporation | Amide based glucagon superfamily peptide prodrugs |
| WO2011163473A1 (en) | 2010-06-25 | 2011-12-29 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting enhanced solubility and stability in physiological ph buffers |
| WO2012088116A2 (en) * | 2010-12-22 | 2012-06-28 | Indiana University Research And Technology Corporation | Glucagon analogs exhibiting gip receptor activity |
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2011
- 2011-12-20 WO PCT/US2011/066164 patent/WO2012088116A2/en not_active Ceased
- 2011-12-20 AU AU2011349331A patent/AU2011349331A1/en not_active Abandoned
- 2011-12-20 ES ES11808086T patent/ES2713952T3/es active Active
- 2011-12-20 NZ NZ612297A patent/NZ612297A/en not_active IP Right Cessation
- 2011-12-20 MA MA36136A patent/MA34885B1/fr unknown
- 2011-12-20 CN CN201180068157.2A patent/CN103458920B/zh not_active Expired - Fee Related
- 2011-12-20 CA CA2821766A patent/CA2821766A1/en not_active Abandoned
- 2011-12-20 EP EP11808086.0A patent/EP2654773B1/en not_active Not-in-force
- 2011-12-20 PE PE2013001437A patent/PE20140186A1/es not_active Application Discontinuation
- 2011-12-20 JP JP2013546329A patent/JP6086067B2/ja not_active Expired - Fee Related
- 2011-12-20 PH PH1/2013/501215A patent/PH12013501215A1/en unknown
- 2011-12-20 BR BR112013015389A patent/BR112013015389A2/pt unknown
- 2011-12-20 US US13/331,816 patent/US8507428B2/en not_active Expired - Fee Related
- 2011-12-20 SG SG2013046412A patent/SG191194A1/en unknown
- 2011-12-20 EA EA201390941A patent/EA201390941A1/ru unknown
- 2011-12-20 KR KR1020137018994A patent/KR20130132931A/ko not_active Withdrawn
- 2011-12-20 MX MX2013006304A patent/MX2013006304A/es not_active Application Discontinuation
- 2011-12-21 AR ARP110104846A patent/AR084459A1/es not_active Application Discontinuation
-
2012
- 2012-12-27 US US13/728,110 patent/US9249206B2/en not_active Expired - Fee Related
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2013
- 2013-06-18 CO CO13145190A patent/CO6761302A2/es unknown
- 2013-06-18 CL CL2013001783A patent/CL2013001783A1/es unknown
- 2013-06-18 CR CR20130295A patent/CR20130295A/es not_active Application Discontinuation
- 2013-06-18 EC ECSP13012697 patent/ECSP13012697A/es unknown
-
2015
- 2015-03-23 US US14/665,508 patent/US20150259393A1/en not_active Abandoned
- 2015-12-28 US US14/981,187 patent/US9587005B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| JP2014507402A (ja) | 2014-03-27 |
| PE20140186A1 (es) | 2014-02-13 |
| US9249206B2 (en) | 2016-02-02 |
| WO2012088116A2 (en) | 2012-06-28 |
| US8507428B2 (en) | 2013-08-13 |
| CA2821766A1 (en) | 2012-06-28 |
| KR20130132931A (ko) | 2013-12-05 |
| MX2013006304A (es) | 2013-07-02 |
| US20160115215A1 (en) | 2016-04-28 |
| EP2654773B1 (en) | 2018-10-03 |
| NZ612297A (en) | 2015-10-30 |
| US20150259393A1 (en) | 2015-09-17 |
| WO2012088116A3 (en) | 2012-11-15 |
| ES2713952T3 (es) | 2019-05-24 |
| US9587005B2 (en) | 2017-03-07 |
| BR112013015389A2 (pt) | 2016-11-22 |
| US20120238493A1 (en) | 2012-09-20 |
| CN103458920B (zh) | 2016-07-06 |
| AR084459A1 (es) | 2013-05-15 |
| MA34885B1 (fr) | 2014-02-01 |
| JP6086067B2 (ja) | 2017-03-01 |
| ECSP13012697A (es) | 2013-10-31 |
| EP2654773A2 (en) | 2013-10-30 |
| CL2013001783A1 (es) | 2014-01-24 |
| US20130116173A1 (en) | 2013-05-09 |
| CR20130295A (es) | 2013-10-09 |
| SG191194A1 (en) | 2013-07-31 |
| PH12013501215A1 (en) | 2013-11-18 |
| CO6761302A2 (es) | 2013-09-30 |
| EA201390941A1 (ru) | 2013-12-30 |
| CN103458920A (zh) | 2013-12-18 |
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| Date | Code | Title | Description |
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| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |