EP1090009A2 - Cell adhesion-inhibiting antinflammatory compounds - Google Patents
Cell adhesion-inhibiting antinflammatory compoundsInfo
- Publication number
- EP1090009A2 EP1090009A2 EP99926157A EP99926157A EP1090009A2 EP 1090009 A2 EP1090009 A2 EP 1090009A2 EP 99926157 A EP99926157 A EP 99926157A EP 99926157 A EP99926157 A EP 99926157A EP 1090009 A2 EP1090009 A2 EP 1090009A2
- Authority
- EP
- European Patent Office
- Prior art keywords
- thieno
- pyridine
- carboxamide
- chlorophenoxy
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US9070198A | 1998-06-04 | 1998-06-04 | |
US90701 | 1998-06-04 | ||
PCT/US1999/012419 WO1999062908A2 (en) | 1998-06-04 | 1999-06-03 | Cell adhesion-inhibiting antinflammatory compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
EP1090009A2 true EP1090009A2 (en) | 2001-04-11 |
Family
ID=22223903
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP99926157A Withdrawn EP1090009A2 (en) | 1998-06-04 | 1999-06-03 | Cell adhesion-inhibiting antinflammatory compounds |
Country Status (15)
Country | Link |
---|---|
EP (1) | EP1090009A2 (no) |
JP (1) | JP2002517396A (no) |
KR (1) | KR20010052570A (no) |
CN (1) | CN1332743A (no) |
AU (1) | AU4231299A (no) |
BG (1) | BG105109A (no) |
BR (1) | BR9910864A (no) |
CA (1) | CA2333770A1 (no) |
HU (1) | HUP0102366A2 (no) |
IL (1) | IL139811A0 (no) |
NO (1) | NO20006157L (no) |
PL (1) | PL345906A1 (no) |
SK (1) | SK18542000A3 (no) |
TR (1) | TR200100189T2 (no) |
WO (1) | WO1999062908A2 (no) |
Families Citing this family (129)
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ATE301651T1 (de) * | 1999-06-23 | 2005-08-15 | Aventis Pharma Gmbh | Substituierte benzimidazole |
US6689883B1 (en) | 1999-09-28 | 2004-02-10 | Bayer Pharmaceuticals Corporation | Substituted pyridines and pyridazines with angiogenesis inhibiting activity |
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US7977333B2 (en) | 2000-04-20 | 2011-07-12 | Bayer Healthcare Llc | Substituted pyridines and pyridazines with angiogenesis inhibiting activity |
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WO2003020729A1 (en) | 2001-08-30 | 2003-03-13 | Pharmacia & Upjohn Company | 4-THIOXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOXAMIDES AS ANT IVIRAL AGENTS |
AR038294A1 (es) | 2002-01-14 | 2005-01-12 | Upjohn Co | Oxotieno(3,2-b)piridincarboxamidas como agentes antivirales |
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KR20050006237A (ko) | 2002-05-06 | 2005-01-15 | 버텍스 파마슈티칼스 인코포레이티드 | 티아디아졸 또는 옥사디아졸 및 jak 단백질 키나제억제제로서의 이들의 용도 |
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IL154306A0 (en) * | 2003-02-05 | 2003-09-17 | Rimonyx Pharmaceuticals Ltd | Pharmaceutical compositions comprising thieno [2,3-c] pyridine derivatives and use thereof |
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1999
- 1999-06-03 IL IL13981199A patent/IL139811A0/xx unknown
- 1999-06-03 SK SK1854-2000A patent/SK18542000A3/sk unknown
- 1999-06-03 BR BR9910864-0A patent/BR9910864A/pt not_active Application Discontinuation
- 1999-06-03 PL PL99345906A patent/PL345906A1/xx not_active Application Discontinuation
- 1999-06-03 AU AU42312/99A patent/AU4231299A/en not_active Abandoned
- 1999-06-03 JP JP2000552119A patent/JP2002517396A/ja not_active Withdrawn
- 1999-06-03 TR TR2001/00189T patent/TR200100189T2/xx unknown
- 1999-06-03 HU HU0102366A patent/HUP0102366A2/hu unknown
- 1999-06-03 WO PCT/US1999/012419 patent/WO1999062908A2/en not_active Application Discontinuation
- 1999-06-03 CA CA002333770A patent/CA2333770A1/en not_active Abandoned
- 1999-06-03 CN CN99809253A patent/CN1332743A/zh active Pending
- 1999-06-03 EP EP99926157A patent/EP1090009A2/en not_active Withdrawn
- 1999-06-03 KR KR1020007013739A patent/KR20010052570A/ko not_active Application Discontinuation
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2000
- 2000-12-04 NO NO20006157A patent/NO20006157L/no not_active Application Discontinuation
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2001
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Non-Patent Citations (1)
Title |
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See references of WO9962908A2 * |
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WO1999062908A3 (en) | 2000-03-30 |
IL139811A0 (en) | 2002-02-10 |
CA2333770A1 (en) | 1999-12-09 |
WO1999062908A2 (en) | 1999-12-09 |
BR9910864A (pt) | 2002-02-05 |
PL345906A1 (en) | 2002-01-14 |
AU4231299A (en) | 1999-12-20 |
NO20006157D0 (no) | 2000-12-04 |
HUP0102366A2 (hu) | 2001-11-28 |
BG105109A (en) | 2001-11-30 |
SK18542000A3 (sk) | 2001-12-03 |
JP2002517396A (ja) | 2002-06-18 |
KR20010052570A (ko) | 2001-06-25 |
CN1332743A (zh) | 2002-01-23 |
TR200100189T2 (tr) | 2001-05-21 |
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