EE200000706A - Bitsüklilised pürimidiinid ja bitsüklilised 3,4-dihüdropürimidiinid kui rakkude proliferatsiooni inhibiitorid - Google Patents

Bitsüklilised pürimidiinid ja bitsüklilised 3,4-dihüdropürimidiinid kui rakkude proliferatsiooni inhibiitorid

Info

Publication number
EE200000706A
EE200000706A EEP200000706A EEP200000706A EE200000706A EE 200000706 A EE200000706 A EE 200000706A EE P200000706 A EEP200000706 A EE P200000706A EE P200000706 A EEP200000706 A EE P200000706A EE 200000706 A EE200000706 A EE 200000706A
Authority
EE
Estonia
Prior art keywords
bicyclic
dihydropyrimidines
inhibitors
cell proliferation
pyrimidines
Prior art date
Application number
EEP200000706A
Other languages
English (en)
Inventor
Marino Hamby James
Daniel Hollis Showalter Howard
Laurence Toogood Peter
Myra Dobrusin Ellen
Bernard Kramer James
Conrad Schroeder Mel
A. Trumpp-Kallmeyer Susanne
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26775058&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EE200000706(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of EE200000706A publication Critical patent/EE200000706A/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
EEP200000706A 1998-05-26 1999-05-10 Bitsüklilised pürimidiinid ja bitsüklilised 3,4-dihüdropürimidiinid kui rakkude proliferatsiooni inhibiitorid EE200000706A (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8670898P 1998-05-26 1998-05-26
US12615899P 1999-03-25 1999-03-25
PCT/US1999/010187 WO1999061444A2 (en) 1998-05-26 1999-05-10 Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation

Publications (1)

Publication Number Publication Date
EE200000706A true EE200000706A (et) 2002-06-17

Family

ID=26775058

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200000706A EE200000706A (et) 1998-05-26 1999-05-10 Bitsüklilised pürimidiinid ja bitsüklilised 3,4-dihüdropürimidiinid kui rakkude proliferatsiooni inhibiitorid

Country Status (29)

Country Link
US (1) US7501425B1 (et)
EP (1) EP1080092B1 (et)
JP (1) JP2002516327A (et)
KR (1) KR20010043829A (et)
CN (1) CN1138778C (et)
AP (1) AP2000001964A0 (et)
AT (1) ATE402177T1 (et)
AU (1) AU763839B2 (et)
BG (1) BG104960A (et)
BR (1) BR9911590A (et)
CA (1) CA2329703C (et)
DE (1) DE69939168D1 (et)
EA (1) EA003640B1 (et)
EE (1) EE200000706A (et)
ES (1) ES2310039T3 (et)
GE (1) GEP20033093B (et)
HK (1) HK1039483A1 (et)
HR (1) HRP20000799A2 (et)
HU (1) HUP0102514A3 (et)
ID (1) ID27589A (et)
IL (1) IL139599A0 (et)
IS (1) IS5687A (et)
NO (1) NO20005928L (et)
NZ (1) NZ508268A (et)
PL (1) PL344248A1 (et)
SK (1) SK17532000A3 (et)
TR (1) TR200003429T2 (et)
WO (1) WO1999061444A2 (et)
YU (1) YU73300A (et)

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DE69939168D1 (de) 2008-09-04
EP1080092B1 (en) 2008-07-23
CA2329703A1 (en) 1999-12-02
NO20005928D0 (no) 2000-11-23
AP2000001964A0 (en) 2000-12-31
ATE402177T1 (de) 2008-08-15
ES2310039T3 (es) 2008-12-16
EA003640B1 (ru) 2003-08-28
CN1138778C (zh) 2004-02-18
US7501425B1 (en) 2009-03-10
AU4073499A (en) 1999-12-13
BG104960A (en) 2001-10-31
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NO20005928L (no) 2000-11-23
CN1302301A (zh) 2001-07-04
AU763839B2 (en) 2003-07-31
ID27589A (id) 2001-04-12
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EP1080092A2 (en) 2001-03-07
IS5687A (is) 2000-10-27
IL139599A0 (en) 2002-02-10
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BR9911590A (pt) 2001-02-13
HRP20000799A2 (en) 2001-06-30

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