EA039373B1 - Производные пиперидино-пиримидина для лечения вирусных инфекций - Google Patents
Производные пиперидино-пиримидина для лечения вирусных инфекций Download PDFInfo
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- EA039373B1 EA039373B1 EA201992133A EA201992133A EA039373B1 EA 039373 B1 EA039373 B1 EA 039373B1 EA 201992133 A EA201992133 A EA 201992133A EA 201992133 A EA201992133 A EA 201992133A EA 039373 B1 EA039373 B1 EA 039373B1
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- Eurasian Patent Office
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12154474 | 2012-02-08 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA201992133A1 EA201992133A1 (ru) | 2020-02-05 |
| EA039373B1 true EA039373B1 (ru) | 2022-01-19 |
Family
ID=47678822
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA201992133A EA039373B1 (ru) | 2012-02-08 | 2013-02-07 | Производные пиперидино-пиримидина для лечения вирусных инфекций |
| EA201491486A EA033907B1 (ru) | 2012-02-08 | 2013-02-07 | Производные пиперидино-пиримидина, фармацевтическая композиция и их применение |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA201491486A EA033907B1 (ru) | 2012-02-08 | 2013-02-07 | Производные пиперидино-пиримидина, фармацевтическая композиция и их применение |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US9133192B2 (enExample) |
| EP (1) | EP2812331B1 (enExample) |
| JP (1) | JP6283320B2 (enExample) |
| KR (1) | KR102064807B1 (enExample) |
| CN (1) | CN104245695B (enExample) |
| AU (1) | AU2013218072B2 (enExample) |
| BR (1) | BR112014019699B1 (enExample) |
| CA (1) | CA2862823C (enExample) |
| CL (1) | CL2014002093A1 (enExample) |
| DK (1) | DK2812331T3 (enExample) |
| EA (2) | EA039373B1 (enExample) |
| ES (1) | ES2716811T3 (enExample) |
| IL (1) | IL233499B (enExample) |
| IN (1) | IN2014MN01736A (enExample) |
| MX (1) | MX357296B (enExample) |
| MY (1) | MY169159A (enExample) |
| NZ (1) | NZ627036A (enExample) |
| PH (1) | PH12014501738B1 (enExample) |
| SG (1) | SG11201404743TA (enExample) |
| UA (1) | UA112668C2 (enExample) |
| WO (1) | WO2013117615A1 (enExample) |
| ZA (1) | ZA201405820B (enExample) |
Families Citing this family (165)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI3590928T1 (sl) | 2011-04-08 | 2021-10-29 | Janssen Sciences Ireland Unlimited Co | Derivati pirimidina za zdravljenje virusnih okužb |
| BR112014011162A2 (pt) | 2011-11-09 | 2017-05-09 | Janssen R&D Ireland | derivados purínicos para o tratamento de infecções virais |
| DK2812331T3 (en) | 2012-02-08 | 2019-04-08 | Janssen Sciences Ireland Unlimited Co | PIPERIDINOPYRIMIDINE DERIVATIVES FOR TREATING VIRUS INFECTIONS |
| WO2014009509A1 (en) | 2012-07-13 | 2014-01-16 | Janssen R&D Ireland | Macrocyclic purines for the treatment of viral infections |
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