BR112014019699B1 - Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende - Google Patents

Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende Download PDF

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BR112014019699B1
BR112014019699B1 BR112014019699-0A BR112014019699A BR112014019699B1 BR 112014019699 B1 BR112014019699 B1 BR 112014019699B1 BR 112014019699 A BR112014019699 A BR 112014019699A BR 112014019699 B1 BR112014019699 B1 BR 112014019699B1
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formula
compound
alkyl
substituted
pharmaceutical composition
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BR112014019699-0A
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Portuguese (pt)
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BR112014019699A8 (pt
BR112014019699A2 (enExample
Inventor
Tim Hugo Maria Jonckers
David Craig Mc Gowan
Pierre Jean-Marie Bernard Raboisson
Mourad Daoubi Khamlichi
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Janssen Sciences Ireland Uc
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Publication of BR112014019699A8 publication Critical patent/BR112014019699A8/pt
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
BR112014019699-0A 2012-02-08 2013-02-07 Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende BR112014019699B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP12154474.6 2012-02-08
EP12154474 2012-02-08
PCT/EP2013/052372 WO2013117615A1 (en) 2012-02-08 2013-02-07 Piperidino-pyrimidine derivatives for the treatment of viral infections

Publications (3)

Publication Number Publication Date
BR112014019699A2 BR112014019699A2 (enExample) 2017-06-20
BR112014019699A8 BR112014019699A8 (pt) 2021-10-19
BR112014019699B1 true BR112014019699B1 (pt) 2021-12-07

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ID=47678822

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Application Number Title Priority Date Filing Date
BR112014019699-0A BR112014019699B1 (pt) 2012-02-08 2013-02-07 Derivados de piperidino-pirimidina, seu uso no tratamento de infecções virais e composição farmacêutica que os compreende

Country Status (22)

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US (2) US9133192B2 (enExample)
EP (1) EP2812331B1 (enExample)
JP (1) JP6283320B2 (enExample)
KR (1) KR102064807B1 (enExample)
CN (1) CN104245695B (enExample)
AU (1) AU2013218072B2 (enExample)
BR (1) BR112014019699B1 (enExample)
CA (1) CA2862823C (enExample)
CL (1) CL2014002093A1 (enExample)
DK (1) DK2812331T3 (enExample)
EA (2) EA033907B1 (enExample)
ES (1) ES2716811T3 (enExample)
IL (1) IL233499B (enExample)
IN (1) IN2014MN01736A (enExample)
MX (1) MX357296B (enExample)
MY (1) MY169159A (enExample)
NZ (1) NZ627036A (enExample)
PH (1) PH12014501738A1 (enExample)
SG (1) SG11201404743TA (enExample)
UA (1) UA112668C2 (enExample)
WO (1) WO2013117615A1 (enExample)
ZA (1) ZA201405820B (enExample)

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