MX357296B - Derivados piperidinopirimidinicos para el tratamiento de infecciones viricas. - Google Patents

Derivados piperidinopirimidinicos para el tratamiento de infecciones viricas.

Info

Publication number
MX357296B
MX357296B MX2014009556A MX2014009556A MX357296B MX 357296 B MX357296 B MX 357296B MX 2014009556 A MX2014009556 A MX 2014009556A MX 2014009556 A MX2014009556 A MX 2014009556A MX 357296 B MX357296 B MX 357296B
Authority
MX
Mexico
Prior art keywords
piperidino
viral infections
treatment
pyrimidine derivatives
derivatives
Prior art date
Application number
MX2014009556A
Other languages
English (en)
Other versions
MX2014009556A (es
Inventor
Pierre Jean-Marie Bernard Raboisson
Gowan David Craig Mc
Tim Hugo Maria Jonckers
Khamlichi Mourad Daoubi
Original Assignee
Janssen Sciences Ireland Uc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47678822&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX357296(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc
Publication of MX2014009556A publication Critical patent/MX2014009556A/es
Publication of MX357296B publication Critical patent/MX357296B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Esta invención se refiere a derivados piperidinopirimidínicos, a procesos para su preparación, a composiciones farmacéuticas y a su uso en el tratamiento de infecciones víricas.
MX2014009556A 2012-02-08 2013-02-07 Derivados piperidinopirimidinicos para el tratamiento de infecciones viricas. MX357296B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12154474 2012-02-08
PCT/EP2013/052372 WO2013117615A1 (en) 2012-02-08 2013-02-07 Piperidino-pyrimidine derivatives for the treatment of viral infections

Publications (2)

Publication Number Publication Date
MX2014009556A MX2014009556A (es) 2014-11-10
MX357296B true MX357296B (es) 2018-07-03

Family

ID=47678822

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014009556A MX357296B (es) 2012-02-08 2013-02-07 Derivados piperidinopirimidinicos para el tratamiento de infecciones viricas.

Country Status (22)

Country Link
US (2) US9133192B2 (es)
EP (1) EP2812331B1 (es)
JP (1) JP6283320B2 (es)
KR (1) KR102064807B1 (es)
CN (1) CN104245695B (es)
AU (1) AU2013218072B2 (es)
CA (1) CA2862823C (es)
CL (1) CL2014002093A1 (es)
DK (1) DK2812331T3 (es)
EA (2) EA033907B1 (es)
ES (1) ES2716811T3 (es)
HK (1) HK1201254A1 (es)
IL (1) IL233499B (es)
IN (1) IN2014MN01736A (es)
MX (1) MX357296B (es)
MY (1) MY169159A (es)
NZ (1) NZ627036A (es)
PH (1) PH12014501738A1 (es)
SG (1) SG11201404743TA (es)
UA (1) UA112668C2 (es)
WO (1) WO2013117615A1 (es)
ZA (1) ZA201405820B (es)

Families Citing this family (132)

* Cited by examiner, † Cited by third party
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SI2694484T1 (sl) 2011-04-08 2018-10-30 Janssen Sciences Ireland Uc Derivati pirimidina za zdravljenje virusnih okužb
PL2776439T3 (pl) 2011-11-09 2018-12-31 Janssen Sciences Ireland Uc Pochodne puryny do leczenia zakażeń wirusowych
ES2716811T3 (es) * 2012-02-08 2019-06-17 Janssen Sciences Ireland Unlimited Co Derivados piperidinopirimidínicos para el tratamiento de infecciones víricas
EP2872515B1 (en) 2012-07-13 2016-06-08 Janssen Sciences Ireland UC Macrocyclic purines for the treatment of viral infections
HUE037064T2 (hu) 2012-10-10 2018-08-28 Janssen Sciences Ireland Uc Pirrolo[3,2-d]-pirimidin származékok vírusos fertõzések és egyéb betegségek kezelésére
EP2925729B1 (en) 2012-11-16 2017-10-18 Janssen Sciences Ireland UC Heterocyclic substituted 2-amino-quinazoline derivatives for the treatment of viral infections
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ES2657283T3 (es) 2013-05-24 2018-03-02 Janssen Sciences Ireland Uc Derivados de piridona para el tratamiento de infecciones virales y enfermedades adicionales
UA117590C2 (uk) 2013-06-27 2018-08-27 ЯНССЕН САЙЄНСЕЗ АЙРЛЕНД ЮСі ПОХІДНІ ПІРОЛО[3,2-d]ПІРИМІДИНУ ДЛЯ ЛІКУВАННЯ ВІРУСНИХ ІНФЕКЦІЙ ТА ІНШИХ ЗАХВОРЮВАНЬ
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