UA112668C2 - Похідні піперидинопіримідину для лікування вірусних інфекцій - Google Patents

Похідні піперидинопіримідину для лікування вірусних інфекцій Download PDF

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UA112668C2
UA112668C2 UAA201407816A UAA201407816A UA112668C2 UA 112668 C2 UA112668 C2 UA 112668C2 UA A201407816 A UAA201407816 A UA A201407816A UA A201407816 A UAA201407816 A UA A201407816A UA 112668 C2 UA112668 C2 UA 112668C2
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formula
compound
pharmaceutically acceptable
nmr
mhz
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UAA201407816A
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Ukrainian (uk)
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Девід Крейг МакГован
П'єр Жан-Марі Бернар Рабуассон
Тім Хьюго Марія Йонкерс
Хамлічі Мурад Даубі
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Янссен Сайєнсиз Айрленд Юсі
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
UAA201407816A 2012-02-08 2013-07-02 Похідні піперидинопіримідину для лікування вірусних інфекцій UA112668C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12154474 2012-02-08
PCT/EP2013/052372 WO2013117615A1 (en) 2012-02-08 2013-02-07 Piperidino-pyrimidine derivatives for the treatment of viral infections

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UA112668C2 true UA112668C2 (uk) 2016-10-10

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UAA201407816A UA112668C2 (uk) 2012-02-08 2013-07-02 Похідні піперидинопіримідину для лікування вірусних інфекцій

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US (2) US9133192B2 (enExample)
EP (1) EP2812331B1 (enExample)
JP (1) JP6283320B2 (enExample)
KR (1) KR102064807B1 (enExample)
CN (1) CN104245695B (enExample)
AU (1) AU2013218072B2 (enExample)
BR (1) BR112014019699B1 (enExample)
CA (1) CA2862823C (enExample)
CL (1) CL2014002093A1 (enExample)
DK (1) DK2812331T3 (enExample)
EA (2) EA033907B1 (enExample)
ES (1) ES2716811T3 (enExample)
IL (1) IL233499B (enExample)
IN (1) IN2014MN01736A (enExample)
MX (1) MX357296B (enExample)
MY (1) MY169159A (enExample)
NZ (1) NZ627036A (enExample)
PH (1) PH12014501738B1 (enExample)
SG (1) SG11201404743TA (enExample)
UA (1) UA112668C2 (enExample)
WO (1) WO2013117615A1 (enExample)
ZA (1) ZA201405820B (enExample)

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