EA034781B1 - Арильные, гетероарильные и гетероциклические соединения для лечения расстройства, опосредованного фактором d комплемента - Google Patents

Арильные, гетероарильные и гетероциклические соединения для лечения расстройства, опосредованного фактором d комплемента Download PDF

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Publication number
EA034781B1
EA034781B1 EA201890594A EA201890594A EA034781B1 EA 034781 B1 EA034781 B1 EA 034781B1 EA 201890594 A EA201890594 A EA 201890594A EA 201890594 A EA201890594 A EA 201890594A EA 034781 B1 EA034781 B1 EA 034781B1
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Eurasian Patent Office
Prior art keywords
alkyl
compound
disorder
pharmaceutically acceptable
independently selected
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EA201890594A
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English (en)
Russian (ru)
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EA201890594A1 (ru
Inventor
Джейсон Аллан Вайлс
Авинаш С. Фадке
Милинд Дешпанде
Атул Агарвал
Давей Чэнь
Венкат Рао Гадхачанда
Акихиро Хашимото
Годвин Пэйс
Цюпин Ван
Сянчжу Ван
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Ачиллион Фармасьютикалс, Инк.
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Publication of EA201890594A1 publication Critical patent/EA201890594A1/ru
Publication of EA034781B1 publication Critical patent/EA034781B1/ru

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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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EA201890594A 2015-08-26 2016-08-25 Арильные, гетероарильные и гетероциклические соединения для лечения расстройства, опосредованного фактором d комплемента EA034781B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201562209972P 2015-08-26 2015-08-26
PCT/US2016/048696 WO2017035353A1 (en) 2015-08-26 2016-08-25 Aryl, heteroaryl, and heterocyclic compounds for treatment of medical disorders

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EA201890594A1 EA201890594A1 (ru) 2018-08-31
EA034781B1 true EA034781B1 (ru) 2020-03-19

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EA201890594A EA034781B1 (ru) 2015-08-26 2016-08-25 Арильные, гетероарильные и гетероциклические соединения для лечения расстройства, опосредованного фактором d комплемента
EA201992884A EA201992884A3 (ru) 2015-08-26 2016-08-25 Арильные, гетероарильные и гетероциклические соединения для лечения заболеваний

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US20190211033A1 (en) 2019-07-11
US12139497B2 (en) 2024-11-12
JP7532561B2 (ja) 2024-08-13
KR102668548B1 (ko) 2024-05-22
AU2021202728A1 (en) 2021-05-27
CN114044800A (zh) 2022-02-15
EA201992884A3 (ru) 2020-08-31
US20210269458A1 (en) 2021-09-02
CN108024992A (zh) 2018-05-11
AU2016311425B2 (en) 2021-02-04
US10287301B2 (en) 2019-05-14
JP2021119169A (ja) 2021-08-12
IL295844B1 (en) 2024-10-01
IL295844A (en) 2022-10-01
JP7210637B2 (ja) 2023-01-23
HUE061088T2 (hu) 2023-05-28
EP3340981B1 (en) 2022-10-12

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