DE69729134T2 - Pharmazeutische Tablette geeignet zur Wirkstofffreisetzung in aufeinanderfolgenden und vorherbestimmbaren Zeiträumen - Google Patents
Pharmazeutische Tablette geeignet zur Wirkstofffreisetzung in aufeinanderfolgenden und vorherbestimmbaren Zeiträumen Download PDFInfo
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- DE69729134T2 DE69729134T2 DE69729134T DE69729134T DE69729134T2 DE 69729134 T2 DE69729134 T2 DE 69729134T2 DE 69729134 T DE69729134 T DE 69729134T DE 69729134 T DE69729134 T DE 69729134T DE 69729134 T2 DE69729134 T2 DE 69729134T2
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- 229960005425 nitrendipine Drugs 0.000 description 1
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- NXFQHRVNIOXGAQ-YCRREMRBSA-N nitrofurantoin Chemical compound O1C([N+](=O)[O-])=CC=C1\C=N\N1C(=O)NC(=O)C1 NXFQHRVNIOXGAQ-YCRREMRBSA-N 0.000 description 1
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- 229940082615 organic nitrates used in cardiac disease Drugs 0.000 description 1
- ADIMAYPTOBDMTL-UHFFFAOYSA-N oxazepam Chemical compound C12=CC(Cl)=CC=C2NC(=O)C(O)N=C1C1=CC=CC=C1 ADIMAYPTOBDMTL-UHFFFAOYSA-N 0.000 description 1
- 229960004535 oxazepam Drugs 0.000 description 1
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- GDYUVHBMFVMBAF-LIRRHRJNSA-N oxyfedrine Chemical compound COC1=CC=CC(C(=O)CCN[C@@H](C)[C@H](O)C=2C=CC=CC=2)=C1 GDYUVHBMFVMBAF-LIRRHRJNSA-N 0.000 description 1
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- LSQZJLSUYDQPKJ-UHFFFAOYSA-N p-Hydroxyampicillin Natural products O=C1N2C(C(O)=O)C(C)(C)SC2C1NC(=O)C(N)C1=CC=C(O)C=C1 LSQZJLSUYDQPKJ-UHFFFAOYSA-N 0.000 description 1
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- PHUTUTUABXHXLW-UHFFFAOYSA-N pindolol Chemical compound CC(C)NCC(O)COC1=CC=CC2=NC=C[C]12 PHUTUTUABXHXLW-UHFFFAOYSA-N 0.000 description 1
- 229960002702 piroxicam Drugs 0.000 description 1
- QYSPLQLAKJAUJT-UHFFFAOYSA-N piroxicam Chemical compound OC=1C2=CC=CC=C2S(=O)(=O)N(C)C=1C(=O)NC1=CC=CC=N1 QYSPLQLAKJAUJT-UHFFFAOYSA-N 0.000 description 1
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- 239000011347 resin Substances 0.000 description 1
- 229920005989 resin Polymers 0.000 description 1
- 230000033764 rhythmic process Effects 0.000 description 1
- 229960000329 ribavirin Drugs 0.000 description 1
- HZCAHMRRMINHDJ-DBRKOABJSA-N ribavirin Natural products O[C@@H]1[C@H](O)[C@@H](CO)O[C@H]1N1N=CN=C1 HZCAHMRRMINHDJ-DBRKOABJSA-N 0.000 description 1
- 230000000630 rising effect Effects 0.000 description 1
- 229960003320 roxatidine Drugs 0.000 description 1
- 229960002052 salbutamol Drugs 0.000 description 1
- 239000004208 shellac Substances 0.000 description 1
- ZLGIYFNHBLSMPS-ATJNOEHPSA-N shellac Chemical compound OCCCCCC(O)C(O)CCCCCCCC(O)=O.C1C23[C@H](C(O)=O)CCC2[C@](C)(CO)[C@@H]1C(C(O)=O)=C[C@@H]3O ZLGIYFNHBLSMPS-ATJNOEHPSA-N 0.000 description 1
- 229940113147 shellac Drugs 0.000 description 1
- 235000013874 shellac Nutrition 0.000 description 1
- 239000011734 sodium Substances 0.000 description 1
- 229910052708 sodium Inorganic materials 0.000 description 1
- ZBMZVLHSJCTVON-UHFFFAOYSA-N sotalol Chemical compound CC(C)NCC(O)C1=CC=C(NS(C)(=O)=O)C=C1 ZBMZVLHSJCTVON-UHFFFAOYSA-N 0.000 description 1
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- 208000024891 symptom Diseases 0.000 description 1
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- 235000002906 tartaric acid Nutrition 0.000 description 1
- 230000002123 temporal effect Effects 0.000 description 1
- 229960000195 terbutaline Drugs 0.000 description 1
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- 229960000278 theophylline Drugs 0.000 description 1
- 229960002044 tolmetin sodium Drugs 0.000 description 1
- 235000010487 tragacanth Nutrition 0.000 description 1
- 239000000196 tragacanth Substances 0.000 description 1
- 229940116362 tragacanth Drugs 0.000 description 1
- 239000003204 tranquilizing agent Substances 0.000 description 1
- 230000002936 tranquilizing effect Effects 0.000 description 1
- VZCYOOQTPOCHFL-UHFFFAOYSA-N trans-butenedioic acid Natural products OC(=O)C=CC(O)=O VZCYOOQTPOCHFL-UHFFFAOYSA-N 0.000 description 1
- 238000012546 transfer Methods 0.000 description 1
- 229960000363 trapidil Drugs 0.000 description 1
- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
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- HEBKCHPVOIAQTA-SCDXWVJYSA-N xylitol Chemical compound OC[C@H](O)[C@@H](O)[C@H](O)CO HEBKCHPVOIAQTA-SCDXWVJYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT96MI000210A IT1282576B1 (it) | 1996-02-06 | 1996-02-06 | Compressa farmaceutica atta a cedere la sostanza attiva in tempi successivi e predeterminabili |
| ITMI960210 | 1996-02-06 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69729134D1 DE69729134D1 (de) | 2004-06-24 |
| DE69729134T2 true DE69729134T2 (de) | 2005-05-12 |
Family
ID=11373151
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69729134T Expired - Lifetime DE69729134T2 (de) | 1996-02-06 | 1997-02-04 | Pharmazeutische Tablette geeignet zur Wirkstofffreisetzung in aufeinanderfolgenden und vorherbestimmbaren Zeiträumen |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US6294200B1 (https=) |
| EP (1) | EP0788790B1 (https=) |
| JP (1) | JPH09221416A (https=) |
| AT (1) | ATE267007T1 (https=) |
| AU (1) | AU720914B2 (https=) |
| CA (1) | CA2196840C (https=) |
| DE (1) | DE69729134T2 (https=) |
| DK (1) | DK0788790T3 (https=) |
| ES (1) | ES2220999T3 (https=) |
| IT (1) | IT1282576B1 (https=) |
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| US10987313B2 (en) | 2013-10-07 | 2021-04-27 | Impax Laboratories, Llc | Muco-adhesive, controlled release formulations of levodopa and/or esters of levodopa and uses thereof |
| CN105658211A (zh) | 2013-10-07 | 2016-06-08 | 怡百克制药公司 | 左旋多巴和/或左旋多巴的酯的粘膜粘附性、控制释放调配物和其用途 |
| CN103948557A (zh) * | 2014-04-08 | 2014-07-30 | 闻晓光 | 一种新型控释片 |
| AU2016272089B2 (en) | 2015-06-03 | 2021-02-18 | Triastek, Inc. | Dosage forms and use thereof |
| AU2017261372B2 (en) * | 2016-05-05 | 2019-02-14 | Triastek, Inc. | Controlled release dosage form |
| EP3573602A4 (en) * | 2017-01-26 | 2020-09-16 | Triastek, Inc. | DOSAGE FORMS OF CONTROLLED RELEASE AT SPECIFIC GASTROINTESTINAL SITES |
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| EP3788884A1 (de) * | 2019-09-05 | 2021-03-10 | Delica AG | Kompostierbare kapsel sowie deren herstellung und verwendung |
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| CN114177155B (zh) * | 2020-09-08 | 2023-10-03 | 越洋医药开发(广州)有限公司 | 一种布洛芬控释片及其制备方法 |
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Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1022171A (en) | 1961-06-15 | 1966-03-09 | Wellcome Found | Prolonged release oral pharmaceutical tablets and their manufacture |
| FR2100858B1 (https=) | 1970-07-03 | 1975-06-06 | Daiichi Seiyaku Co | |
| US4077407A (en) | 1975-11-24 | 1978-03-07 | Alza Corporation | Osmotic devices having composite walls |
| US4898733A (en) * | 1985-11-04 | 1990-02-06 | International Minerals & Chemical Corp. | Layered, compression molded device for the sustained release of a beneficial agent |
| IT1201136B (it) * | 1987-01-13 | 1989-01-27 | Resa Farma | Compressa per uso farmaceutico atta al rilascio in tempi successivi di sostanze attive |
| DK469989D0 (da) * | 1989-09-22 | 1989-09-22 | Bukh Meditec | Farmaceutisk praeparat |
| IT1255522B (it) * | 1992-09-24 | 1995-11-09 | Ubaldo Conte | Compressa per impiego terapeutico atta a cedere una o piu' sostanze attive con differenti velocita' |
| IT1264517B1 (it) * | 1993-05-31 | 1996-09-24 | Ekita Investments Nv | Compressa farmaceutica atta al rilascio in tempi successivi dei principi attivi in essa veicolati |
| JP3725542B2 (ja) * | 1993-10-19 | 2005-12-14 | 大正製薬株式会社 | ピコサルフェート剤形 |
-
1996
- 1996-02-06 IT IT96MI000210A patent/IT1282576B1/it active IP Right Grant
-
1997
- 1997-02-04 US US08/795,382 patent/US6294200B1/en not_active Expired - Lifetime
- 1997-02-04 ES ES97101689T patent/ES2220999T3/es not_active Expired - Lifetime
- 1997-02-04 DE DE69729134T patent/DE69729134T2/de not_active Expired - Lifetime
- 1997-02-04 AT AT97101689T patent/ATE267007T1/de active
- 1997-02-04 EP EP97101689A patent/EP0788790B1/en not_active Expired - Lifetime
- 1997-02-04 AU AU12526/97A patent/AU720914B2/en not_active Expired
- 1997-02-04 DK DK97101689T patent/DK0788790T3/da active
- 1997-02-05 CA CA002196840A patent/CA2196840C/en not_active Expired - Lifetime
- 1997-02-05 JP JP9022465A patent/JPH09221416A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| IT1282576B1 (it) | 1998-03-31 |
| AU720914B2 (en) | 2000-06-15 |
| EP0788790A2 (en) | 1997-08-13 |
| EP0788790A3 (en) | 1998-11-04 |
| ATE267007T1 (de) | 2004-06-15 |
| AU1252697A (en) | 1997-08-28 |
| DE69729134D1 (de) | 2004-06-24 |
| CA2196840C (en) | 2001-12-04 |
| CA2196840A1 (en) | 1997-08-07 |
| US6294200B1 (en) | 2001-09-25 |
| EP0788790B1 (en) | 2004-05-19 |
| JPH09221416A (ja) | 1997-08-26 |
| DK0788790T3 (da) | 2004-09-20 |
| ITMI960210A0 (https=) | 1996-02-06 |
| ITMI960210A1 (it) | 1997-08-06 |
| ES2220999T3 (es) | 2004-12-16 |
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