DE602006008942D1 - Formulierung eines thienopyridin-thrombozytenaggregationshemmers - Google Patents

Formulierung eines thienopyridin-thrombozytenaggregationshemmers

Info

Publication number
DE602006008942D1
DE602006008942D1 DE602006008942T DE602006008942T DE602006008942D1 DE 602006008942 D1 DE602006008942 D1 DE 602006008942D1 DE 602006008942 T DE602006008942 T DE 602006008942T DE 602006008942 T DE602006008942 T DE 602006008942T DE 602006008942 D1 DE602006008942 D1 DE 602006008942D1
Authority
DE
Germany
Prior art keywords
thrombozytenaggregationshemmers
thienopyridin
formulierung
eines
formulierung eines
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602006008942T
Other languages
English (en)
Inventor
David Brian Dziennik
Tamara Beth Edelman
Peter Lloyd Oren
Robert Louis Ternik
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37198935&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE602006008942(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of DE602006008942D1 publication Critical patent/DE602006008942D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)
DE602006008942T 2005-06-10 2006-06-06 Formulierung eines thienopyridin-thrombozytenaggregationshemmers Active DE602006008942D1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US68918305P 2005-06-10 2005-06-10
PCT/US2006/021860 WO2006135605A2 (en) 2005-06-10 2006-06-06 Formulation of a thienopyridine platelet aggregation inhibitor

Publications (1)

Publication Number Publication Date
DE602006008942D1 true DE602006008942D1 (en) 2009-10-15

Family

ID=37198935

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602006008942T Active DE602006008942D1 (en) 2005-06-10 2006-06-06 Formulierung eines thienopyridin-thrombozytenaggregationshemmers

Country Status (35)

Country Link
US (1) US20080176893A1 (de)
EP (1) EP1896019B1 (de)
JP (1) JP2008543755A (de)
KR (2) KR20100076050A (de)
CN (1) CN101193633B (de)
AR (1) AR054283A1 (de)
AT (1) ATE441413T1 (de)
AU (1) AU2006258102B2 (de)
BR (1) BRPI0611350B8 (de)
CA (1) CA2611668C (de)
CY (1) CY1109502T1 (de)
DE (1) DE602006008942D1 (de)
DK (1) DK1896019T3 (de)
DO (1) DOP2006000126A (de)
EA (1) EA011693B1 (de)
EC (1) ECSP077984A (de)
ES (1) ES2330373T3 (de)
HK (1) HK1116422A1 (de)
HR (1) HRP20090516T1 (de)
IL (1) IL187830A0 (de)
MA (1) MA29688B1 (de)
MX (1) MX2007015431A (de)
MY (1) MY151038A (de)
NO (1) NO20076317L (de)
NZ (1) NZ564003A (de)
PE (1) PE20070320A1 (de)
PL (1) PL1896019T3 (de)
PT (1) PT1896019E (de)
RS (1) RS51194B (de)
SI (1) SI1896019T1 (de)
TN (1) TNSN07466A1 (de)
TW (1) TWI318571B (de)
UA (1) UA91051C2 (de)
WO (1) WO2006135605A2 (de)
ZA (1) ZA200710697B (de)

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KR101442862B1 (ko) * 2006-12-07 2014-09-22 다이이찌 산쿄 가부시키가이샤 만니톨 또는 유당을 함유하는 고형 제제
BRPI0719529B8 (pt) * 2006-12-07 2021-05-25 Daiichi Sankyo Co Ltd método para produzir uma preparação sólida
CA2671975C (en) * 2006-12-07 2013-10-29 Daiichi Sankyo Company, Limited Film-coated preparation having improved stability
WO2008072532A1 (ja) * 2006-12-07 2008-06-19 Daiichi Sankyo Company, Limited 貯蔵安定性が改善された医薬組成物
CA2671979C (en) * 2006-12-07 2014-02-04 Daiichi Sankyo Company, Limited Pharmaceutical composition containing low-substituted hydroxypropyl cellulose
US20100179184A1 (en) * 2006-12-07 2010-07-15 Matthew John Moon Article of manufacture for prasugrel
EP2123656B1 (de) * 2007-03-02 2014-06-11 Daiichi Sankyo Company, Limited Verfahren zur herstellung von hochreinem prasugrelhydrochlorid
KR20150041173A (ko) 2007-04-27 2015-04-15 사이덱스 파마슈티칼스, 인크. 클로피도그렐 및 설포알킬 에테르 사이클로덱스트린을 함유하는 제형 및 사용 방법
GB2450117A (en) * 2007-06-13 2008-12-17 Reckitt Benckiser Healthcare A water- and oxygen-occlusive blister tablet pack
EP2257556A1 (de) 2008-02-06 2010-12-08 Helm AG Prasugrelsalze mit verbesserten eigenschaften
EP2107061A1 (de) * 2008-04-02 2009-10-07 Krka Tovarna Zdravil, D.D., Novo Mesto Herstellungsverfahren für optisch angereichertes Clopidogrel
PL2112155T3 (pl) 2008-04-25 2011-03-31 Sandoz Ag Wodorosiarczan (VI) 2-acetoksy-5-(α-cyklopropylokarbonylo-2-fluorobenzylo)-4,5,6,7-tetrahydrotieno[3,2-c]pirydyny i sposób jego otrzymywania
EP2398468B1 (de) 2009-02-17 2016-11-30 KRKA, D.D., Novo Mesto Pharmazeutische zusammensetzungen mit einer prasugrel-basis oder ihren pharmazeutisch annehmbaren säureadditionssalzen und herstellungsverfahren dafür
KR101743591B1 (ko) 2009-05-13 2017-06-20 사이덱스 파마슈티칼스, 인크. 프라수그렐 및 사이클로덱스트린 유도체를 포함하는 약학 조성물 및 그의 제조 및 사용 방법
DE102009036646A1 (de) 2009-08-07 2011-02-10 Ratiopharm Gmbh Prasugrel in nicht-kristalliner Form und pharmazeutische Zusammensetzung davon
JP2013032289A (ja) * 2009-10-28 2013-02-14 Daiichi Sankyo Co Ltd ワックス安定製剤
WO2011052499A1 (ja) * 2009-10-28 2011-05-05 第一三共株式会社 貯蔵安定性が改善された医薬組成物
WO2011092720A2 (en) * 2010-02-01 2011-08-04 Msn Laboratories Limited Pharmaceutical composition of prasugrel and its pharmaceutically acceptable salts
TR201007926A1 (tr) 2010-07-19 2012-02-21 Sanovel İlaç San.Ve Ti̇c.A.Ş. Prasugrel tablet formülasyonları.
TR201006802A1 (tr) * 2010-08-17 2012-03-21 Sanovel İlaç San. Ve Ti̇c. A.Ş. Prasugrelin oral yolla dağılan formülasyonları.
TR201005900A1 (tr) 2010-07-19 2012-02-21 Sanovel İlaç San. Ve Ti̇c. A.Ş. Geliştirilmiş stabiliteye sahip prasugrel granülleri.
EP2409685A3 (de) 2010-07-19 2012-02-01 Sanovel Ilac Sanayi ve Ticaret A.S. Sich im Mund auflösende Formulierungen aus Prasugrel
CZ2011872A3 (cs) 2011-12-22 2013-07-03 Zentiva, K.S. Farmaceutická formulace prasugrelu hydrobromidu
US8603537B2 (en) 2012-04-02 2013-12-10 Egis Pharmaceuticals Plc Prasugrel containing quickly released stable oral pharmaceutical compositions
EP2722036A1 (de) 2012-10-19 2014-04-23 Sanovel Ilac Sanayi ve Ticaret A.S. Feste orale Formulierungen aus Prasugrel
EP2722037A1 (de) 2012-10-19 2014-04-23 Sanovel Ilac Sanayi ve Ticaret A.S. Prasugrelformulierungen
CN102993210A (zh) * 2012-12-19 2013-03-27 苏春华 一种吡啶并噻吩的新化合物
EP2979693A1 (de) 2014-08-01 2016-02-03 Zaklady Farmaceutyczne Polpharma SA Pharmazeutische zusammensetzung mit prasugrel oder pharmazeutisch verträglichem salz davon und verfahren zu deren herstellung
WO2016122421A1 (en) 2015-01-29 2016-08-04 Pharmactive Ilaç Sanayi Ve Ticaret A.Ş. Stable pharmaceutical compositions containing prasugrel base
EP3158993A1 (de) 2015-10-22 2017-04-26 Zaklady Farmaceutyczne Polpharma SA Verfahren zur herstellung einer tablette mit prasugrel oder pharmazeutisch unbedenklichem salz davon
CN107304216A (zh) * 2016-04-20 2017-10-31 陕西合成药业股份有限公司 噻吩吡啶类衍生物及其制备方法和用途
HU231079B1 (hu) 2016-06-23 2020-06-29 Richter Gedeon Nyrt. Eljárás nagytisztaságú Prasugrel előállítására bromopentil szennyezés eltávolításával
GR1009230B (el) 2016-10-12 2018-02-22 Φαρματεν Αβεε Φαρμακευτικο σκευασμα που περιλαμβανει βεσυλικη πρασουγρελη

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Publication number Priority date Publication date Assignee Title
FI101150B (fi) * 1991-09-09 1998-04-30 Sankyo Co Menetelmä lääkeaineina käyttökelpoisten tetrahydrotienopyridiinin johd annaisten valmistamiseksi
ES2308633T3 (es) * 2000-07-06 2008-12-01 Daiichi Sankyo Company, Limited Sal de adicion de maleato de derivados de la hidropiridina.
JP4001199B2 (ja) * 2000-07-06 2007-10-31 第一三共株式会社 ヒドロピリジン誘導体酸付加塩
EP1243524A3 (de) * 2001-03-16 2004-04-07 Pfizer Products Inc. Pharmazeutisches Kit fÜr sauerstoffempfindliche Medikamente
JP4394873B2 (ja) * 2001-12-19 2010-01-06 武田薬品工業株式会社 酸素に不安定な化合物を含有する固形組成物およびその安定化方法
SI21302A (sl) * 2002-10-11 2004-04-30 LEK farmacevtska dru�ba d.d. Stabiliziran farmacevtski izdelek z amorfno aktivno učinkovino
US20050020554A1 (en) * 2003-06-06 2005-01-27 Ahmed Salah U. Stability of hormone formulations
PT1653930E (pt) * 2003-08-05 2008-03-12 Zentiva As Métodos para a estabilização da atorvastatina

Also Published As

Publication number Publication date
MA29688B1 (fr) 2008-08-01
MX2007015431A (es) 2008-02-21
NZ564003A (en) 2011-07-29
CA2611668A1 (en) 2006-12-21
RS51194B (sr) 2010-10-31
DOP2006000126A (es) 2006-12-15
JP2008543755A (ja) 2008-12-04
WO2006135605A3 (en) 2007-04-12
KR20100076050A (ko) 2010-07-05
HK1116422A1 (en) 2008-12-24
BRPI0611350B1 (pt) 2020-09-15
CN101193633A (zh) 2008-06-04
ES2330373T3 (es) 2009-12-09
EP1896019A2 (de) 2008-03-12
ATE441413T1 (de) 2009-09-15
ZA200710697B (en) 2009-08-26
AR054283A1 (es) 2007-06-13
BRPI0611350B8 (pt) 2021-05-25
UA91051C2 (ru) 2010-06-25
EA200702670A1 (ru) 2008-04-28
CA2611668C (en) 2013-10-15
DK1896019T3 (da) 2009-10-26
SI1896019T1 (sl) 2010-01-29
AU2006258102A1 (en) 2006-12-21
IL187830A0 (en) 2008-04-13
HRP20090516T1 (en) 2009-10-31
TNSN07466A1 (en) 2009-03-17
MY151038A (en) 2014-03-31
NO20076317L (no) 2008-02-29
CN101193633B (zh) 2011-12-14
CY1109502T1 (el) 2014-08-13
AU2006258102B2 (en) 2011-09-15
US20080176893A1 (en) 2008-07-24
PL1896019T3 (pl) 2010-01-29
BRPI0611350A2 (pt) 2010-12-07
PE20070320A1 (es) 2007-05-12
TW200718420A (en) 2007-05-16
WO2006135605A2 (en) 2006-12-21
ECSP077984A (es) 2008-01-23
EA011693B1 (ru) 2009-04-28
PT1896019E (pt) 2009-11-19
EP1896019B1 (de) 2009-09-02
TWI318571B (en) 2009-12-21
KR20080008413A (ko) 2008-01-23

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Legal Events

Date Code Title Description
8363 Opposition against the patent
8328 Change in the person/name/address of the agent

Representative=s name: DR. SCHOEN & PARTNER, 80336 MUENCHEN