CN1805958A - 稠合的n-杂环化合物和它们作为crf受体拮抗剂的用途 - Google Patents

稠合的n-杂环化合物和它们作为crf受体拮抗剂的用途 Download PDF

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Publication number
CN1805958A
CN1805958A CNA2004800161898A CN200480016189A CN1805958A CN 1805958 A CN1805958 A CN 1805958A CN A2004800161898 A CNA2004800161898 A CN A2004800161898A CN 200480016189 A CN200480016189 A CN 200480016189A CN 1805958 A CN1805958 A CN 1805958A
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Prior art keywords
methyl
compound
phenyl
dihydro
pyrrolo
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Pending
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CNA2004800161898A
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Chinese (zh)
Inventor
丹尼尔·安德烈奥蒂
乔瓦尼·伯纳斯科尼
埃米莉亚诺·卡斯蒂格利奥尼
斯蒂法尼亚·康蒂尼
罗马诺·迪法比奥
伊莱特拉·法佐拉里
阿尔多·弗里亚尼
加布里拉·金蒂尔
马里奥·马蒂奥利
安娜·明加迪
法比奥·萨巴蒂尼
伊维斯·圣丹尼斯
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Neurocrine Biosciences Inc
SB Pharmco Puerto Rico Inc
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Neurocrine Biosciences Inc
SB Pharmco Puerto Rico Inc
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Publication of CN1805958A publication Critical patent/CN1805958A/zh
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CNA2004800161898A 2003-04-09 2004-04-07 稠合的n-杂环化合物和它们作为crf受体拮抗剂的用途 Pending CN1805958A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0308208.8 2003-04-09
GBGB0308208.8A GB0308208D0 (en) 2003-04-09 2003-04-09 Chemical compounds
US48532203P 2003-07-07 2003-07-07
US60/485,322 2003-07-07

Related Child Applications (1)

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CNA2008101656972A Division CN101434604A (zh) 2003-04-09 2004-04-07 稠合的n-杂环化合物和它们作为crf受体拮抗剂的用途

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CN1805958A true CN1805958A (zh) 2006-07-19

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CNA2004800161898A Pending CN1805958A (zh) 2003-04-09 2004-04-07 稠合的n-杂环化合物和它们作为crf受体拮抗剂的用途

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US (2) US7427630B2 (https=)
EP (3) EP2186813A1 (https=)
JP (2) JP4866722B2 (https=)
KR (1) KR20060021826A (https=)
CN (1) CN1805958A (https=)
AR (1) AR044005A1 (https=)
AT (2) ATE473226T1 (https=)
AU (1) AU2004232551C1 (https=)
BR (1) BRPI0409117A (https=)
CA (1) CA2521929C (https=)
DE (2) DE602004027998D1 (https=)
GB (1) GB0308208D0 (https=)
IS (1) IS8119A (https=)
MA (1) MA27796A1 (https=)
MX (1) MXPA05010874A (https=)
NO (1) NO20055238L (https=)
NZ (1) NZ542780A (https=)
PL (1) PL378755A1 (https=)
RU (1) RU2382785C2 (https=)
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CA2550948A1 (en) * 2003-12-22 2005-07-14 Sb Pharmco Puerto Rico Inc. Crf receptor antagonists and methods relating thereto
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DE602005014375D1 (de) * 2004-10-19 2009-06-18 Neurocrine Biosciences Inc Crf-rezeptor-antagonisten und zugehörige verfahren
GB0519957D0 (en) * 2005-09-30 2005-11-09 Sb Pharmco Inc Chemical compound
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US7598255B2 (en) 2005-08-04 2009-10-06 Janssen Pharmaceutica Nv Pyrimidine compounds as serotonin receptor modulators
US8088779B2 (en) * 2005-09-30 2012-01-03 Smithkline Beecham (Cork) Limited Pyrazolo [1,5-alpha] pyrimidinyl derivatives useful as corticotropin-releasing factor (CRF) receptor antagonists
US8329701B2 (en) 2006-07-06 2012-12-11 Array Biopharma Inc. Dihydrofuro pyrimidines as AKT protein kinase inhibitors
EP2049500B1 (en) * 2006-07-06 2011-09-07 Array Biopharma, Inc. Cyclopenta [d] pyrimidines as akt protein kinase inhibitors
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