CN1147252A - 酰化的氨基苯磺酰脲,其制备方法以及其作为除草剂和植物生长调节剂的用途 - Google Patents
酰化的氨基苯磺酰脲,其制备方法以及其作为除草剂和植物生长调节剂的用途 Download PDFInfo
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- CN1147252A CN1147252A CN95192788A CN95192788A CN1147252A CN 1147252 A CN1147252 A CN 1147252A CN 95192788 A CN95192788 A CN 95192788A CN 95192788 A CN95192788 A CN 95192788A CN 1147252 A CN1147252 A CN 1147252A
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- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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Abstract
Description
No. | R1 | R2 | R3 | R4 | X | Y | Z | Mp.(℃) |
1 | H | H | COCH3 | H | OMe | OMe | CH | |
2 | H | H | CO-H | H | OMe | OMe | CH | |
3 | - | - | COOMe | - | - | - | - | |
4 | - | Me | COCH3 | - | - | - | - | |
5 | - | - | CO-H | - | - | - | - | |
6 | - | - | COOMe | - | - | - | - | |
7 | - | - | COCF3 | - | - | - | - | |
8 | Me | Me | CO-H | - | - | - | - | 126-127(分解) |
9 | - | - | - | - | - | Me | - | |
10 | - | - | - | - | - | Cl | - | |
11 | - | - | - | - | Me | Me | - | |
12 | - | - | - | - | Me | OMe | N | |
13 | - | - | - | - | OMe | OMe | N | |
14 | - | - | - | - | NMe2 | OCH2CF3 | N | |
15 | - | - | CO-CH3 | - | OMe | OMe | CH | 182-184(分解) |
16 | - | - | - | - | - | Cl | - | |
17 | - | - | - | - | - | Me | - | |
18 | - | - | - | - | Me | - | - |
No. | R1 | R2 | R3 | R4 | X | Y | Z | Mp.(℃) |
19 | Me | Me | CO-CH3 | H | OMe | OMe | N | |
20 | - | - | - | - | Me | OMe | - | |
21 | - | - | - | - | NMe2 | OCH2CF3 | - | |
22 | - | - | COCH2CH3 | - | OMe | OMe | CH | 135-140(分解) |
23 | - | - | - | - | OMe | Cl | - | |
24 | - | - | CO-CH2CH3 | - | OMe | Me | N | |
25 | Me | Me | CO-iPr | H | OMe | OMe | CH | 145-149(分解) |
26 | - | - | - | - | - | Cl | - | |
27 | - | - | - | - | - | Me | - | |
28 | - | - | - | - | Me | - | - | |
29 | - | - | - | - | OMe | - | N | |
30 | - | - | CO-tBu | - | - | OMe | CH | 202(分解) |
31 | - | - | CO-nPr | - | - | - | - | |
32 | - | - | CO-nBu | - | - | - | - | |
33 | - | - | CO-n-C5H11 | - | - | - | - | |
34 | - | - | CO-CH2Cl | - | - | - | - | |
35 | - | - | - | - | - | Cl | - | |
36 | - | - | CO-CHCl2 | - | - | OMe | - | |
37 | - | - | CO-CCl3 | - | - | - | - | |
38 | - | - | CO-CH2Br | - | - | - | - | |
39 | - | - | COCF3 | - | - | - | - | |
40 | Me | Me | COCF3 | H | OMe | Me | - | 203(分解) |
41 | - | - | - | - | - | Cl | - |
No. | R1 | R2 | R3 | R4 | X | Y | Z | Mp.(℃) |
62 | Me | Me | COOEt | H | Me | Me | CH | |
63 | - | - | - | - | OMe | Me | N | |
64 | Me | Me | COOiPr | H | OMe | OMe | CH | |
65 | - | - | COOCCH2CH2Cl | - | - | - | - | 154-155(分解) |
66 | - | - | - | - | OMe | Cl | - | |
67 | - | - | - | - | - | Me | - | |
68 | - | - | CO2CH2CH2Br | - | - | OMe | - | |
69 | - | - | CO2CH2CCl3 | - | - | - | - | |
70 | - | - | CO-NH2 | - | - | - | - | |
71 | - | - | CO-NHMe | - | - | - | - | |
72 | - | - | CONHEt | - | - | - | - | 144(分解) |
73 | - | - | CONMe2 | - | - | - | - | |
74 | - | - | CONEt2 | - | - | - | - | |
75 | - | - | CO-N(Me)-OMe | - | - | - | - | |
76 | Me | Me | CS-NHMe | H | OMe | OMe | CH | |
77 | - | - | SO2CH3 | - | - | - | - | 190-191(分解) |
78 | - | - | - | - | - | Cl | - | |
79 | - | - | - | - | Me | Me | - | |
80 | - | - | - | - | Me | OMe | N | |
81 | - | - | SO2Et | - | - | - | - | |
82 | Me | Me | SO2Et | H | OMe | OMe | CH | |
83 | - | - | - | - | - | Cl | - | |
84 | - | - | - | - | Me | Me | - | |
85 | - | - | SO2CH2Cl | - | OMe | OMe | CH |
No. | R1 | R2 | R3 | R4 | X | Y | Z | Mp.(℃) |
86 | Me | Me | SO2CH2F | H | OMe | OMe | CH | |
87 | - | - | SO2NHMe | - | - | - | - | 128-129(分解) |
88 | - | - | SO2NMe2 | - | - | - | - | |
89 | Et | Et | CO-H | - | - | - | - | 64-67 |
90 | Et | Et | CO-CH3 | H | OMe | OMe | CH | 195-197(分解) |
91 | - | - | COOMe | - | - | - | - | |
92 | -(CH2)4- | CO-H | - | - | - | - | ||
93 | - | CO-CH3 | - | - | - | - | ||
94 | - | COOMe | - | - | - | - | ||
95 | -O-(CH2)3- | CO-H | - | - | - | - | ||
96 | - | CO-CH3 | - | - | - | - | ||
97 | - | COOCH3 | - | - | - | - | ||
98 | -O-(CH2)4- | CO-H | - | - | - | - | ||
99 | - | CO-CH3 | - | - | - | - | ||
100 | - | COOMe | - | - | - | - | ||
101 | -(CH2)2-O-(CH2)2- | CO-H | H | OMe | OMe | CH | ||
102 | - | CO-CH3 | - | - | - | - | ||
103 | - | CO-CH2CH3 | - | - | - | - | ||
104 | OMe | Me | CO-CH3 | - | - | - | - | |
105 | - | - | COOMe | - | - | - | - | |
106 | Me | Me | CO-H | Me | - | - | - | |
107 | Me | Me | CO-CH3 | Me | OMe | OMe | CH | |
108 | - | - | CO-CH2CH3 | - | - | - | - | |
109 | - | - | COOMe | - | - | - | - |
No. | R1 | R2 | R3 | R4 | X | Y | Z | Mp.(℃) |
110 | - | - | COCF3 | - | - | - | - | |
111 | H | Ph | COCH3 | H | OMe | OMe | CH | |
112 | - | - | COOCH3 | - | - | - | - | |
113 | Me | - | - | - | - | - | - | |
114 | Me | Me | CO-Et | - | Me | Me | CH | |
115 | - | - | CO-cPr | - | OMe | OMe | - | 196-197(分解) |
116 | Me | Et | CO-H | - | OMe | OMe | CH | 90(分解) |
117 | Me | nPr | CO-H | - | - | - | - | |
118 | Et | Me | CO-CH3 | - | - | - | - | 192-195 |
No. | R1 | R2 | R3 | R4 | M | X | Y | Z | Mp.(C) |
1 | Me | Me | CO-H | H | Na | OMe | OMe | CH | 205(分解) |
2 | - | - | - | - | K | OMe | OMe | CH | |
3 | - | - | - | - | NH4 | - | - | - | |
4 | - | - | - | - | HNEt3 | - | - | - | |
5 | - | - | - | - | Na | OMe | Cl | - | |
6 | - | - | - | - | - | OMe | Me | N |
No. | R1 | R2 | R3 | R4 | M | X | Y | Z | Mp.(℃) |
7 | - | - | CO-CH3 | - | - | - | OMe | CH | 196(分解)) |
8 | - | - | - | - | K | - | - | - | |
9 | - | - | - | - | Na | - | Cl | - | |
10 | - | - | - | - | - | Me | Me | - | |
11 | Me | Me | CO-CH3 | H | Na | OMe | Me | N | |
12 | - | - | COCH2CH3 | - | - | OMe | OMe | CH | 212(分解) |
13 | - | - | - | - | - | OMe | Cl | CH | |
14 | - | - | - | - | - | OMe | Me | N | |
15 | - | - | - | - | - | NMe2 | OCM2CF3 | N | |
16 | - | - | CO-iPr | - | - | OMe | OMe | CH | 208(分解) |
17 | - | - | COCF3 | - | - | - | - | - | 198-201(分解) |
18 | - | - | - | - | - | - | Cl | - | |
19 | Me | Me | COCF3 | H | Na | OMe | Me | N | |
20 | - | - | COOMe | - | - | - | - | - | 167-170(分解) |
21 | - | - | - | - | - | OMe | OMe | CH | 187-191(分解) |
22 | Me | Me | COOMe- | H | Na | OMe | Cl | CH | 267-270(分解) |
23 | - | - | - | - | - | - | Me | - | |
24 | - | - | - | - | - | Me | - | - | |
25 | - | - | - | - | K | OMe | OMe | - | |
26 | - | - | COOEt | - | Na | - | - | - | 194-198(分解) |
No. | R1 | R2 | R3 | R4 | M | X | Y | Z | Mp.(℃) |
27 | - | - | COOiPr | - | - | - | - | - | |
28 | - | - | CO2CH2CH2Cl | - | - | - | - | - | 159-165(分解) |
29 | - | - | SO2CH3 | - | - | - | - | - | 130-134(分解) |
30 | Me | Me | SO2NHMe | H | Na | OMe | OMe | CH | 187-189(分解) |
31 | - | - | SO2CH2Cl | - | - | - | - | - | |
32 | - | - | CO-oPr | - | - | - | - | - | 194(分解) |
33 | - | - | CO-NHEt | - | - | - | - | - | 195-198(分解) |
34 | - | - | CO-tBu | - | - | - | - | - | 201(分解) |
35 | - | Et | CO-H | - | - | - | - | - | |
36 | - | nPr | CO-H | - | - | - | - | - |
Claims (10)
Applications Claiming Priority (2)
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DEP4415049.0 | 1994-04-29 | ||
DE4415049A DE4415049A1 (de) | 1994-04-29 | 1994-04-29 | Acylierte Aminophenylsulfonylharnstoffe, Verfahren zu deren Herstellung und Verwendung als Herbizide und Wachstumsregulatoren |
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CNB001089552A Division CN1205192C (zh) | 1994-04-29 | 2000-05-24 | 酰化的氨基苯磺酰脲,其制备方法以及其作为除草剂和植物生长调节剂的用途 |
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CN95192788A Expired - Lifetime CN1066140C (zh) | 1994-04-29 | 1995-04-12 | 酰化的氨基苯磺酰脲,其制备方法以及其作为除草剂和植物生长调节剂的用途 |
CNB001089552A Expired - Lifetime CN1205192C (zh) | 1994-04-29 | 2000-05-24 | 酰化的氨基苯磺酰脲,其制备方法以及其作为除草剂和植物生长调节剂的用途 |
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CNB001089552A Expired - Lifetime CN1205192C (zh) | 1994-04-29 | 2000-05-24 | 酰化的氨基苯磺酰脲,其制备方法以及其作为除草剂和植物生长调节剂的用途 |
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US (2) | US5922646A (zh) |
EP (1) | EP0757679B1 (zh) |
JP (1) | JP3665339B2 (zh) |
KR (1) | KR100379594B1 (zh) |
CN (2) | CN1066140C (zh) |
AT (1) | ATE172456T1 (zh) |
AU (1) | AU2344195A (zh) |
BG (1) | BG62931B1 (zh) |
BR (1) | BR9507562A (zh) |
CA (1) | CA2189044C (zh) |
CZ (1) | CZ294362B6 (zh) |
DE (2) | DE4415049A1 (zh) |
DK (1) | DK0757679T3 (zh) |
ES (1) | ES2125012T3 (zh) |
HU (1) | HU222441B1 (zh) |
MX (1) | MX197808B (zh) |
PL (1) | PL183786B1 (zh) |
RO (1) | RO114894B1 (zh) |
RU (1) | RU2171253C2 (zh) |
TR (1) | TR28237A (zh) |
UA (1) | UA48134C2 (zh) |
WO (1) | WO1995029899A1 (zh) |
ZA (1) | ZA953436B (zh) |
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DE4440354A1 (de) * | 1994-11-11 | 1996-05-15 | Hoechst Schering Agrevo Gmbh | Kombinationen aus Phenylsulfonylharnstoff-Herbiziden und Safenern |
DE19540701A1 (de) | 1995-11-02 | 1997-05-07 | Hoechst Schering Agrevo Gmbh | Verfahren zur Herstellung von Aminophenylsulfonylharnstoffen und Zwischenprodukte zu den Verfahren |
DE19544743A1 (de) * | 1995-12-01 | 1997-06-05 | Hoechst Schering Agrevo Gmbh | 5-Acylamino-2-alkoxycarbonylphenylsulfonylharnstoffe als selektive Herbizide |
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TR200100458T2 (tr) | 1998-08-13 | 2001-07-23 | Aventis Cropscience Gmbh | Asilleştirilmiş aminofenilsulfonil üreli herbisit ilaçlar |
WO2000047566A1 (de) * | 1999-02-10 | 2000-08-17 | Aventis Cropscience Gmbh | Phenylsulfonylharnstoffe, verfahren zu ihrer herstellung und ihre verwendung als herbizide und pfanzenwachstumsregulatoren |
JP2002538151A (ja) | 1999-03-02 | 2002-11-12 | ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド | カテプシンの可逆的インヒビターとして有用な化合物 |
US6420364B1 (en) | 1999-09-13 | 2002-07-16 | Boehringer Ingelheim Pharmaceuticals, Inc. | Compound useful as reversible inhibitors of cysteine proteases |
ES2219404T3 (es) * | 1999-10-26 | 2004-12-01 | Bayer Cropscience Gmbh | Agentes herbicidas. |
DE19955056A1 (de) * | 1999-11-15 | 2001-05-17 | Aventis Cropscience Gmbh | Herbizid-Kombination mit acylierten Aminophenylsulfonylharnstoffen |
EP1242386B1 (en) * | 1999-12-09 | 2009-08-26 | Bayer CropScience AG | Nitro-sulfobenzamides |
EP1381277A2 (en) | 2001-04-27 | 2004-01-21 | Syngenta Participations AG | Herbicidal composition |
DE10135642A1 (de) * | 2001-07-21 | 2003-02-27 | Bayer Cropscience Gmbh | Herbizid-Kombinationen mit speziellen Sulfonylharnstoffen |
DE10160139A1 (de) | 2001-12-07 | 2003-06-18 | Bayer Cropscience Gmbh | Synergistische herbizide Mittel enthaltend bestimmte Herbizide aus der Gruppe der Benzoylcylohexandione |
DE10209430A1 (de) | 2002-03-05 | 2003-09-18 | Bayer Cropscience Gmbh | Herbizid-Kombination mit acylierten Aminophenylsulfonylharnstoffen |
DE10209478A1 (de) * | 2002-03-05 | 2003-09-18 | Bayer Cropscience Gmbh | Herbizid-Kombinationen mit speziellen Sulfonylharnstoffen |
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EP2052606A1 (de) | 2007-10-24 | 2009-04-29 | Bayer CropScience AG | Herbizid-Kombination |
DE102008037620A1 (de) | 2008-08-14 | 2010-02-18 | Bayer Crop Science Ag | Herbizid-Kombination mit Dimethoxytriazinyl-substituierten Difluormethansulfonylaniliden |
EA031196B1 (ru) | 2010-10-15 | 2018-11-30 | Байер Интеллектуэль Проперти Гмбх | Применение als ингибиторных гербицидов для контроля нежелательной вегетации в растениях beta vulgaris, толерантных к als ингибиторным гербицидам |
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AU2012251597B2 (en) | 2011-05-04 | 2015-11-05 | Bayer Intellectual Property Gmbh | Use of ALS inhibitor herbicides for control of unwanted vegetation in ALS inhibitor herbicide tolerant Brassica, such as B. napus, plants |
BR112014005654A2 (pt) | 2011-09-12 | 2017-03-28 | Bayer Cropscience Lp | métodos para melhorar a saúde e promover o crescimento de uma planta e/ou de melhorar o amadurecimento da fruta |
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CN108712862B (zh) * | 2016-04-11 | 2021-12-07 | 花王株式会社 | 植物的培育方法 |
JP6962696B2 (ja) | 2016-04-11 | 2021-11-05 | 花王株式会社 | 土壌改良剤 |
CA3203568A1 (en) | 2020-12-01 | 2022-06-09 | Bayer Aktiengesellschaft | Compositions comprising mesosulfuron-methyl and tehp |
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-
1994
- 1994-04-29 DE DE4415049A patent/DE4415049A1/de not_active Withdrawn
-
1995
- 1995-04-12 JP JP52795395A patent/JP3665339B2/ja not_active Expired - Lifetime
- 1995-04-12 KR KR1019960706094A patent/KR100379594B1/ko not_active IP Right Cessation
- 1995-04-12 EP EP95917311A patent/EP0757679B1/de not_active Expired - Lifetime
- 1995-04-12 CN CN95192788A patent/CN1066140C/zh not_active Expired - Lifetime
- 1995-04-12 DK DK95917311T patent/DK0757679T3/da active
- 1995-04-12 CA CA002189044A patent/CA2189044C/en not_active Expired - Lifetime
- 1995-04-12 RO RO96-01949A patent/RO114894B1/ro unknown
- 1995-04-12 ES ES95917311T patent/ES2125012T3/es not_active Expired - Lifetime
- 1995-04-12 WO PCT/EP1995/001344 patent/WO1995029899A1/de active IP Right Grant
- 1995-04-12 BR BR9507562A patent/BR9507562A/pt not_active IP Right Cessation
- 1995-04-12 MX MX9605256A patent/MX197808B/es unknown
- 1995-04-12 CZ CZ19963130A patent/CZ294362B6/cs not_active IP Right Cessation
- 1995-04-12 AT AT95917311T patent/ATE172456T1/de active
- 1995-04-12 HU HU9602966A patent/HU222441B1/hu active Protection Beyond IP Right Term
- 1995-04-12 DE DE59503993T patent/DE59503993D1/de not_active Expired - Lifetime
- 1995-04-12 RU RU96121627/04A patent/RU2171253C2/ru active
- 1995-04-12 PL PL95317128A patent/PL183786B1/pl unknown
- 1995-04-12 AU AU23441/95A patent/AU2344195A/en not_active Abandoned
- 1995-04-27 TR TR00484/95A patent/TR28237A/xx unknown
- 1995-04-28 ZA ZA953436A patent/ZA953436B/xx unknown
- 1995-12-04 UA UA96104325A patent/UA48134C2/uk unknown
-
1996
- 1996-10-16 BG BG100913A patent/BG62931B1/bg unknown
-
1997
- 1997-08-04 US US08/906,238 patent/US5922646A/en not_active Expired - Lifetime
-
1999
- 1999-02-25 US US09/257,669 patent/US6498253B1/en not_active Expired - Lifetime
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2000
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CN106889099A (zh) * | 2017-04-14 | 2017-06-27 | 江苏莱科化学有限公司 | 一种含甲酰氨基嘧磺隆与唑嘧磺草胺的除草组合物 |
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