BR0009847A - Kit de partes, método de preparação de um kit de partes, formulação farmacêutica, método de tratamento de uma condição na qual inibição de trombina é requerida ou desejada, e, uso de um inibidor de trombina, ou de um derivado farmaceuticamente aceitável do mesmo - Google Patents
Kit de partes, método de preparação de um kit de partes, formulação farmacêutica, método de tratamento de uma condição na qual inibição de trombina é requerida ou desejada, e, uso de um inibidor de trombina, ou de um derivado farmaceuticamente aceitável do mesmoInfo
- Publication number
- BR0009847A BR0009847A BR0009847-7A BR0009847A BR0009847A BR 0009847 A BR0009847 A BR 0009847A BR 0009847 A BR0009847 A BR 0009847A BR 0009847 A BR0009847 A BR 0009847A
- Authority
- BR
- Brazil
- Prior art keywords
- kit
- parts
- pharmaceutically acceptable
- pharmaceutical formulation
- thrombin
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 4
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 4
- 101000712605 Theromyzon tessulatum Theromin Proteins 0.000 title abstract 3
- 229940122388 Thrombin inhibitor Drugs 0.000 title abstract 3
- 230000005764 inhibitory process Effects 0.000 title abstract 3
- 239000003868 thrombin inhibitor Substances 0.000 title abstract 3
- 108090000190 Thrombin Proteins 0.000 title abstract 2
- 229960004072 thrombin Drugs 0.000 title abstract 2
- 239000002671 adjuvant Substances 0.000 abstract 2
- 239000003085 diluting agent Substances 0.000 abstract 2
- 239000003937 drug carrier Substances 0.000 abstract 2
- 239000000651 prodrug Substances 0.000 abstract 2
- 229940002612 prodrug Drugs 0.000 abstract 2
- 239000000306 component Substances 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 229940127557 pharmaceutical product Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/55—Protease inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
"KIT DE PARTES, MéTODO DE PREPARAçãO DE UM KIT DE PARTES, FORMULAçãO FARMACêUTICA, MéTODO DE TRATAMENTO DE UMA CONDIçãO NA QUAL INIBIçãO DE TROMBINA é REQUERIDA OU DESEJADA, E, USO DE UM INIBIDOR DE TROMBINA, OU DE UM DERIVADO FARMACEUTICAMENTE ACEITáVEL DO MESMO". De acordo com a invenção é proporcionado um kit de partes compreendendo: (a) uma formulação farmacêutica incluindo um inibidor de trombina de baixo peso molecular, ou um seu derivado farmaceuticamente aceitável, misturado com um veiculo, adjuvante ou diluente farmaceuticamente aceitável; e (b) uma formulação farmacêutica incluindo uma pró-droga de um inibidor de trombina de baixo peso molecular, ou um derivado farmaceuticamente aceitável daquela pró-droga, misturado com um veículo, adjuvante ou diluente farmaceuticamente aceitável, cujos componentes (a) e (b) são, cada um, proporcionados em uma forma que é apropriada para administração conjunta de um com o outro, bem como o uso de um tal kit de partes no tratamento de uma condição na qual inibição de trombina é requerida ou desejada.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE9901442A SE523811C2 (sv) | 1999-04-21 | 1999-04-21 | Beredning innehållande en trombininhibitor med låg molekylvikt tillsammans med en prodrog av densamma |
SE9904419A SE9904419D0 (sv) | 1999-12-03 | 1999-12-03 | New use |
PCT/SE2000/000756 WO2000064470A1 (en) | 1999-04-21 | 2000-04-19 | A pharmaceutical formulation comprising a low molecular weight thrombin inhibitor and its prodrug |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0009847A true BR0009847A (pt) | 2002-01-08 |
Family
ID=26663557
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0009847-7A BR0009847A (pt) | 1999-04-21 | 2000-04-19 | Kit de partes, método de preparação de um kit de partes, formulação farmacêutica, método de tratamento de uma condição na qual inibição de trombina é requerida ou desejada, e, uso de um inibidor de trombina, ou de um derivado farmaceuticamente aceitável do mesmo |
Country Status (29)
Country | Link |
---|---|
US (3) | US6962905B1 (pt) |
EP (2) | EP1886691A3 (pt) |
JP (1) | JP2002542298A (pt) |
KR (1) | KR20010110788A (pt) |
CN (1) | CN100377742C (pt) |
AR (1) | AR023510A1 (pt) |
AT (1) | ATE383868T1 (pt) |
AU (1) | AU754405B2 (pt) |
BR (1) | BR0009847A (pt) |
CA (1) | CA2371008A1 (pt) |
CZ (1) | CZ20013757A3 (pt) |
DE (1) | DE60037816T2 (pt) |
DK (1) | DK1200118T3 (pt) |
EE (1) | EE200100543A (pt) |
ES (1) | ES2298141T3 (pt) |
HK (1) | HK1045465B (pt) |
HU (1) | HUP0200955A3 (pt) |
IL (1) | IL145840A0 (pt) |
IS (1) | IS6111A (pt) |
MY (1) | MY128061A (pt) |
NO (1) | NO20015107L (pt) |
NZ (1) | NZ514827A (pt) |
PL (1) | PL201793B1 (pt) |
PT (1) | PT1200118E (pt) |
RU (1) | RU2252783C2 (pt) |
SA (1) | SA00210092B1 (pt) |
SK (1) | SK14962001A3 (pt) |
TR (1) | TR200103017T2 (pt) |
WO (1) | WO2000064470A1 (pt) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE9900070D0 (sv) | 1999-01-13 | 1999-01-13 | Astra Ab | New use |
AR023510A1 (es) * | 1999-04-21 | 2002-09-04 | Astrazeneca Ab | Un equipo de partes, formulacion farmaceutica y uso de un inhibidor de trombina. |
US20020116222A1 (en) * | 2000-10-22 | 2002-08-22 | Standing Stone, Inc. | Method and system for administering anticoagulation therapy |
US6462021B1 (en) * | 2000-11-06 | 2002-10-08 | Astrazeneca Ab | Use of low molecular weight thrombin inhibitor |
DE10064797A1 (de) * | 2000-12-22 | 2002-06-27 | Knoll Ag | Orale und parenterale pharmazeutische Formulierung, umfassend eine niedermolekulare Thrombininhibitor-Pro-Pharmakon |
SE0101762D0 (sv) * | 2001-05-18 | 2001-05-18 | Astrazeneca Ab | New use |
SE0101932D0 (sv) * | 2001-05-31 | 2001-05-31 | Astrazeneca Ab | Pharmaceutical combinations |
SE0103590D0 (sv) | 2001-10-26 | 2001-10-26 | Astrazeneca Ab | New Combination |
US7838560B2 (en) | 2002-03-11 | 2010-11-23 | The Medicines Company (Leipzig) Gmbh | Urokinase inhibitors, production and use thereof |
SE0203349D0 (sv) * | 2002-11-12 | 2002-11-12 | Astrazeneca Ab | New use |
DE10301300B4 (de) | 2003-01-15 | 2009-07-16 | Curacyte Chemistry Gmbh | Verwendung von acylierten 4-Amidino- und 4-Guanidinobenzylaminen zur Inhibierung von Plasmakallikrein |
GB0306615D0 (en) * | 2003-03-22 | 2003-04-30 | Astrazeneca Ab | New use |
DE10342108A1 (de) * | 2003-09-11 | 2005-04-14 | Curacyte Chemistry Gmbh | Basisch-substituierte Benzylaminanaloga als Inhibitoren des Gerinnungsfaktors Xa, ihre Herstellung und Verwendung |
DE102005044319A1 (de) | 2005-09-16 | 2007-03-22 | Curacyte Chemistry Gmbh | 2-(Aminomethyl)-5-Chlor-Benzylamid-Derivate und ihre Verwendung als Hemmstoffe des Gerinnungsfaktors Xa |
DE102006050672A1 (de) | 2006-10-24 | 2008-04-30 | Curacyte Discovery Gmbh | Hemmstoffe des Plasmins und des Plasmakallikreins |
NZ700332A (en) * | 2010-03-30 | 2017-06-30 | Verseon Corp | Multisubstituted aromatic compounds as inhibitors of thrombin |
BR112015023214A8 (pt) | 2013-03-15 | 2019-12-24 | Verseon Corp | composto, composição farmacêutica, e, uso de um composto ou composição farmacêutica |
PL2968297T3 (pl) | 2013-03-15 | 2019-04-30 | Verseon Corp | Wielopodstawione związki aromatyczne jako inhibitory protezy serynowej |
RU2017112739A (ru) | 2014-09-17 | 2018-10-17 | Версеон Корпорейшн | Пиразолил-замещенные пиридоновые соединения как ингибиторы сериновых протеаз |
SG10201907699YA (en) | 2015-02-27 | 2019-09-27 | Verseon Corp | Substituted pyrazole compounds as serine protease inhibitors |
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DE19632772A1 (de) | 1996-08-14 | 1998-02-19 | Basf Ag | Neue Benzamidine |
DE19632773A1 (de) | 1996-08-14 | 1998-02-19 | Basf Ag | Neue Thrombininhibitoren |
PE121699A1 (es) | 1997-02-18 | 1999-12-08 | Boehringer Ingelheim Pharma | Heterociclos biciclicos disustituidos como inhibidores de la trombina |
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SE9704543D0 (sv) | 1997-12-05 | 1997-12-05 | Astra Ab | New compounds |
DE19754490A1 (de) | 1997-12-09 | 1999-06-10 | Boehringer Ingelheim Pharma | Durch einen Aminocarbonylrest substituierte Bicyclen, ihre Herstellung und ihre Verwendung als Arzneimittel |
HUP0100082A3 (en) | 1998-01-26 | 2001-12-28 | Abbott Gmbh & Co Kg | Thrombin inhibitor, peptide derivatives, pharmaceutical compositions comprising thereof and their use |
EP1049673A1 (de) | 1998-01-26 | 2000-11-08 | Basf Aktiengesellschaft | Heterocyclische amidine als kallikrein protease inhibitoren |
JP2002502844A (ja) | 1998-02-03 | 2002-01-29 | ベーリンガー インゲルハイム ファルマ コマンディトゲゼルシャフト | 5員複素環縮合ベンゾ誘導体、その調製及び医薬品としてのそれらの使用 |
DE19816983A1 (de) | 1998-04-17 | 1999-10-21 | Boehringer Ingelheim Pharma | Bicyclen, deren Herstellung und deren Verwendung als Arzneimittel |
TWI248435B (en) | 1998-07-04 | 2006-02-01 | Boehringer Ingelheim Pharma | Benzimidazoles, the preparation thereof and their use as pharmaceutical compositions |
DE19834751A1 (de) | 1998-08-01 | 2000-02-03 | Boehringer Ingelheim Pharma | Disubstituierte bicyclische Heterocyclen, ihre Herstellung und ihre Verwendung als Arzneimittel |
CA2320730A1 (en) * | 1998-12-23 | 2000-07-06 | Renhua Li | Thrombin or factor xa inhibitors |
AR023510A1 (es) * | 1999-04-21 | 2002-09-04 | Astrazeneca Ab | Un equipo de partes, formulacion farmaceutica y uso de un inhibidor de trombina. |
-
2000
- 2000-04-14 AR ARP000101756A patent/AR023510A1/es not_active Application Discontinuation
- 2000-04-19 NZ NZ514827A patent/NZ514827A/en unknown
- 2000-04-19 CZ CZ20013757A patent/CZ20013757A3/cs unknown
- 2000-04-19 JP JP2000613460A patent/JP2002542298A/ja active Pending
- 2000-04-19 EE EEP200100543A patent/EE200100543A/xx unknown
- 2000-04-19 AT AT00928047T patent/ATE383868T1/de not_active IP Right Cessation
- 2000-04-19 ES ES00928047T patent/ES2298141T3/es not_active Expired - Lifetime
- 2000-04-19 PL PL351917A patent/PL201793B1/pl unknown
- 2000-04-19 EP EP07120002A patent/EP1886691A3/en not_active Withdrawn
- 2000-04-19 TR TR2001/03017T patent/TR200103017T2/xx unknown
- 2000-04-19 DK DK00928047T patent/DK1200118T3/da active
- 2000-04-19 CA CA002371008A patent/CA2371008A1/en not_active Abandoned
- 2000-04-19 DE DE60037816T patent/DE60037816T2/de not_active Expired - Fee Related
- 2000-04-19 HU HU0200955A patent/HUP0200955A3/hu unknown
- 2000-04-19 BR BR0009847-7A patent/BR0009847A/pt not_active Application Discontinuation
- 2000-04-19 SK SK1496-2001A patent/SK14962001A3/sk unknown
- 2000-04-19 KR KR1020017013403A patent/KR20010110788A/ko active IP Right Grant
- 2000-04-19 EP EP00928047A patent/EP1200118B1/en not_active Expired - Lifetime
- 2000-04-19 US US09/582,863 patent/US6962905B1/en not_active Expired - Fee Related
- 2000-04-19 AU AU46336/00A patent/AU754405B2/en not_active Ceased
- 2000-04-19 MY MYPI20001656A patent/MY128061A/en unknown
- 2000-04-19 IL IL14584000A patent/IL145840A0/xx unknown
- 2000-04-19 PT PT00928047T patent/PT1200118E/pt unknown
- 2000-04-19 WO PCT/SE2000/000756 patent/WO2000064470A1/en active IP Right Grant
- 2000-04-19 RU RU2001128157/15A patent/RU2252783C2/ru active
- 2000-04-19 CN CNB008091447A patent/CN100377742C/zh not_active Expired - Fee Related
- 2000-05-15 SA SA00210092A patent/SA00210092B1/ar unknown
-
2001
- 2001-10-19 IS IS6111A patent/IS6111A/is unknown
- 2001-10-19 NO NO20015107A patent/NO20015107L/no not_active Application Discontinuation
-
2002
- 2002-09-27 HK HK02107166.1A patent/HK1045465B/zh not_active IP Right Cessation
-
2005
- 2005-08-18 US US11/206,006 patent/US20060009397A1/en not_active Abandoned
-
2007
- 2007-11-09 US US11/979,882 patent/US20080113960A1/en not_active Abandoned
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