BG63542B1 - Методи и междинни съединения за получаване на заместени хроманолови производни - Google Patents

Методи и междинни съединения за получаване на заместени хроманолови производни Download PDF

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Publication number
BG63542B1
BG63542B1 BG103231A BG10323199A BG63542B1 BG 63542 B1 BG63542 B1 BG 63542B1 BG 103231 A BG103231 A BG 103231A BG 10323199 A BG10323199 A BG 10323199A BG 63542 B1 BG63542 B1 BG 63542B1
Authority
BG
Bulgaria
Prior art keywords
alkyl
compound
formula
phenyl
enantiomer
Prior art date
Application number
BG103231A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG103231A (en
Inventor
Joel HAWKINS
Anthony Piscopio
Stephane Caron
Sarah KELLY
Jefrey RAGGON
Michael CASTALDI
Robert DUGGER
Sally RUGGERI
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of BG103231A publication Critical patent/BG103231A/xx
Publication of BG63542B1 publication Critical patent/BG63542B1/bg

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/50Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
BG103231A 1996-09-16 1999-03-09 Методи и междинни съединения за получаване на заместени хроманолови производни BG63542B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16
PCT/IB1997/001024 WO1998011085A1 (en) 1996-09-16 1997-08-25 Processes and intermediates for preparing substituted chromanol derivatives

Publications (2)

Publication Number Publication Date
BG103231A BG103231A (en) 1999-12-30
BG63542B1 true BG63542B1 (bg) 2002-04-30

Family

ID=21831429

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103231A BG63542B1 (bg) 1996-09-16 1999-03-09 Методи и междинни съединения за получаване на заместени хроманолови производни

Country Status (39)

Country Link
US (4) US6096906A (es)
EP (1) EP0925292B1 (es)
JP (1) JP3117730B2 (es)
KR (1) KR100339164B1 (es)
CN (1) CN1108298C (es)
AP (1) AP726A (es)
AT (1) ATE249452T1 (es)
AU (1) AU713701B2 (es)
BG (1) BG63542B1 (es)
BR (1) BR9711482A (es)
CA (1) CA2265043C (es)
CO (1) CO4600635A1 (es)
DE (1) DE69724801T2 (es)
DK (1) DK0925292T3 (es)
DZ (1) DZ2308A1 (es)
EA (1) EA002204B1 (es)
ES (1) ES2206738T3 (es)
GT (3) GT199700104A (es)
HN (1) HN1997000127A (es)
HR (1) HRP970497B1 (es)
ID (1) ID19613A (es)
IL (1) IL128732A0 (es)
IS (1) IS4980A (es)
MA (1) MA24319A1 (es)
NO (1) NO991254L (es)
NZ (1) NZ334214A (es)
OA (1) OA10995A (es)
PA (1) PA8437901A1 (es)
PE (1) PE109798A1 (es)
PL (1) PL332351A1 (es)
PT (1) PT925292E (es)
SK (1) SK31399A3 (es)
TN (1) TNSN97155A1 (es)
TR (1) TR199900592T2 (es)
TW (1) TW449579B (es)
UA (1) UA58520C2 (es)
WO (1) WO1998011085A1 (es)
YU (1) YU13299A (es)
ZA (1) ZA978291B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
CA2433516A1 (en) * 2001-01-30 2002-08-08 Keith Michael Devries Processes for preparing chromanylbenzoic acids
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
ES2551916T3 (es) * 2007-07-23 2015-11-24 The Board Of Trustees Of The University Of Illinois Sistema para controlar la reactividad de los ácidos borónicos
US8338601B2 (en) * 2008-09-26 2012-12-25 Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
US8350099B2 (en) 2009-09-02 2013-01-08 E I Du Pont De Nemours And Company Fluorovinyl ether functionalized aromatic diesters, derivatives thereof, and process for the preparation thereof
US8378061B2 (en) * 2009-09-02 2013-02-19 E.I. Du Pont De Nemours And Company Polyester films with improved oil repellency
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
TW201113311A (en) * 2009-09-02 2011-04-16 Du Pont Polyaramid films comprising fluorovinylether functionalized aromatic moieties
AU2010289583A1 (en) * 2009-09-02 2012-03-15 E. I. Du Pont De Nemours And Company Polyesters comprising fluorovinylether functionalized aromatic moieties
WO2011028766A2 (en) * 2009-09-02 2011-03-10 E. I. Du Pont De Nemours And Company Fluorinated 4-oxo-chroman-carboxylates
WO2011103435A2 (en) 2010-02-18 2011-08-25 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
US10500178B2 (en) 2015-03-13 2019-12-10 The Board Of Trustees Of The Leland Stanford Junior University LTB4 inhibition to prevent and treat human lymphedema

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
WO1993015066A1 (en) * 1992-01-23 1993-08-05 Pfizer Inc. Benzopyran and related ltb4 antagonists
BR9307277A (pt) * 1992-10-21 1999-05-11 Pfizer Derivados sulfonamida de compostos de anel cicloalquílico e heterocíclico substituído com hidróxi condensado com benzeno
JPH07507811A (ja) * 1992-10-21 1995-08-31 ファイザー・インク. 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸
CN1160399A (zh) * 1994-10-13 1997-09-24 美国辉瑞有限公司 苯并吡喃和苯并稠合化合物、其制备方法和它们作为白三烯b4(ltb4)拮抗剂的用途
JP3012339B2 (ja) * 1994-10-13 2000-02-21 ファイザー・インコーポレーテッド ベンゾピランおよびベンゾ縮合化合物、それらの製造、並びにロイコトリエンb▲下4▼(ltb▲下4▼)アンタゴニストとしてのそれらの用途
US5539128A (en) * 1994-11-30 1996-07-23 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
DZ2308A1 (fr) 2002-12-28
DE69724801T2 (de) 2004-06-17
DK0925292T3 (da) 2004-01-12
CO4600635A1 (es) 1998-05-08
US20020099227A1 (en) 2002-07-25
EA002204B1 (ru) 2002-02-28
JP3117730B2 (ja) 2000-12-18
ZA978291B (en) 1999-03-15
CA2265043C (en) 2003-01-14
NZ334214A (en) 2000-09-29
BR9711482A (pt) 1999-08-24
AU3781497A (en) 1998-04-02
JP2000502726A (ja) 2000-03-07
ES2206738T3 (es) 2004-05-16
TR199900592T2 (xx) 1999-06-21
TW449579B (en) 2001-08-11
NO991254D0 (no) 1999-03-15
TNSN97155A1 (fr) 2005-03-15
PT925292E (pt) 2004-01-30
EA199900204A1 (ru) 1999-08-26
YU13299A (sh) 2001-03-07
US6444826B1 (en) 2002-09-03
ATE249452T1 (de) 2003-09-15
GT199700104AA (es) 1999-03-28
DE69724801D1 (de) 2003-10-16
SK31399A3 (en) 2000-05-16
MA24319A1 (fr) 1998-04-01
US20020042526A1 (en) 2002-04-11
PE109798A1 (es) 1999-01-13
UA58520C2 (uk) 2003-08-15
GT199700104BA (es) 1999-03-28
CN1230954A (zh) 1999-10-06
EP0925292A1 (en) 1999-06-30
WO1998011085A1 (en) 1998-03-19
EP0925292B1 (en) 2003-09-10
IL128732A0 (en) 2000-01-31
CA2265043A1 (en) 1998-03-19
IS4980A (is) 1999-02-16
US6096906A (en) 2000-08-01
HRP970497A2 (en) 1998-08-31
AP726A (en) 1999-01-29
AP9701083A0 (en) 1997-10-31
GT199700104A (es) 1999-03-02
AU713701B2 (en) 1999-12-09
PL332351A1 (en) 1999-09-13
NO991254L (no) 1999-05-14
US6355825B1 (en) 2002-03-12
BG103231A (en) 1999-12-30
CN1108298C (zh) 2003-05-14
OA10995A (en) 2001-11-06
ID19613A (id) 1998-07-23
HRP970497B1 (en) 2002-06-30
US6288242B1 (en) 2001-09-11
KR20000036136A (ko) 2000-06-26
PA8437901A1 (es) 2000-05-24
KR100339164B1 (ko) 2002-06-01
HN1997000127A (es) 1997-12-20

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