GT199700104BA - Procedimientos e intermedios para preparar derivados de cromanol sustituidos - Google Patents
Procedimientos e intermedios para preparar derivados de cromanol sustituidosInfo
- Publication number
- GT199700104BA GT199700104BA GT199700104BL GT199700104L GT199700104BA GT 199700104B A GT199700104B A GT 199700104BA GT 199700104B L GT199700104B L GT 199700104BL GT 199700104 L GT199700104 L GT 199700104L GT 199700104B A GT199700104B A GT 199700104BA
- Authority
- GT
- Guatemala
- Prior art keywords
- intermediates
- procedures
- chromanol derivatives
- substituted chromanol
- prepare substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
- C07C33/40—Halogenated unsaturated alcohols
- C07C33/50—Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
- C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
- C07D311/22—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
Abstract
ESTA INVENCION SE REFIERE A LA PREPARACION DE DERIVADOS DE CROMANOL SUSTITUIDOS Y A INTERMEDIOS UTILES EN DICHA PREPARACION. LOS DERIVADOS DE CROMANOL SUSTITUIDOS QUE SE PREPARAN DE ACUERDO CON LA PRESENTE INVENCION, INHIBEN LA ACCION DE LTB4. ESTOS COMPUESTOS TIENEN LA ESTRUCTURA QUIMICA(XIII), EN LA QUE R3,R4,R7, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2637296P | 1996-09-16 | 1996-09-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
GT199700104BA true GT199700104BA (es) | 1999-03-28 |
Family
ID=21831429
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT199700104A GT199700104A (es) | 1996-09-16 | 1997-09-08 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos. |
GT199700104BL GT199700104BA (es) | 1996-09-16 | 1997-10-04 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos |
GT199700104AK GT199700104AA (es) | 1996-09-16 | 1997-10-04 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT199700104A GT199700104A (es) | 1996-09-16 | 1997-09-08 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos. |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT199700104AK GT199700104AA (es) | 1996-09-16 | 1997-10-04 | Procedimientos e intermedios para preparar derivados de cromanol sustituidos |
Country Status (39)
Country | Link |
---|---|
US (4) | US6096906A (es) |
EP (1) | EP0925292B1 (es) |
JP (1) | JP3117730B2 (es) |
KR (1) | KR100339164B1 (es) |
CN (1) | CN1108298C (es) |
AP (1) | AP726A (es) |
AT (1) | ATE249452T1 (es) |
AU (1) | AU713701B2 (es) |
BG (1) | BG63542B1 (es) |
BR (1) | BR9711482A (es) |
CA (1) | CA2265043C (es) |
CO (1) | CO4600635A1 (es) |
DE (1) | DE69724801T2 (es) |
DK (1) | DK0925292T3 (es) |
DZ (1) | DZ2308A1 (es) |
EA (1) | EA002204B1 (es) |
ES (1) | ES2206738T3 (es) |
GT (3) | GT199700104A (es) |
HN (1) | HN1997000127A (es) |
HR (1) | HRP970497B1 (es) |
ID (1) | ID19613A (es) |
IL (1) | IL128732A0 (es) |
IS (1) | IS4980A (es) |
MA (1) | MA24319A1 (es) |
NO (1) | NO991254L (es) |
NZ (1) | NZ334214A (es) |
OA (1) | OA10995A (es) |
PA (1) | PA8437901A1 (es) |
PE (1) | PE109798A1 (es) |
PL (1) | PL332351A1 (es) |
PT (1) | PT925292E (es) |
SK (1) | SK31399A3 (es) |
TN (1) | TNSN97155A1 (es) |
TR (1) | TR199900592T2 (es) |
TW (1) | TW449579B (es) |
UA (1) | UA58520C2 (es) |
WO (1) | WO1998011085A1 (es) |
YU (1) | YU13299A (es) |
ZA (1) | ZA978291B (es) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6436987B1 (en) * | 2000-06-08 | 2002-08-20 | Pfizer Inc. | Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid |
BR0206771A (pt) * | 2001-01-30 | 2004-02-25 | Pfizer Prod Inc | Processos para a preparação de cidos cromanilbenzóicos |
AU4239302A (en) * | 2001-06-28 | 2003-01-02 | Pfizer Products Inc. | Benzoic acid substituted benzopyrans for the treatment of atherosclerosis |
ES2551916T3 (es) | 2007-07-23 | 2015-11-24 | The Board Of Trustees Of The University Of Illinois | Sistema para controlar la reactividad de los ácidos borónicos |
WO2010036921A2 (en) | 2008-09-26 | 2010-04-01 | The Board Of Trustees Of The University Of Illinois | Slow release of organoboronic acids in cross-coupling reactions |
US8304513B2 (en) * | 2009-09-02 | 2012-11-06 | E I Du Pont De Nemours And Company | Polyesters comprising fluorovinylether functionalized aromatic moieties |
US8378061B2 (en) * | 2009-09-02 | 2013-02-19 | E.I. Du Pont De Nemours And Company | Polyester films with improved oil repellency |
TW201127822A (en) * | 2009-09-02 | 2011-08-16 | Du Pont | Fluorinated 4-oxo-chroman-carboxylates |
CN102612509A (zh) | 2009-09-02 | 2012-07-25 | 纳幕尔杜邦公司 | 氟醚官能化的芳族二酯及其衍生物 |
CA2773142A1 (en) * | 2009-09-02 | 2011-03-10 | Neville Everton Drysdale | Polyaramid comprising fluorovinylether functionalized aromatic moieties |
US20110218319A1 (en) * | 2009-09-02 | 2011-09-08 | E. I. Du Pont De Nemours And Company | Polyaramid films comprising fluorovinylether functionalized aromatic moieties |
US8557980B2 (en) | 2010-02-18 | 2013-10-15 | The Board Of Trustees Of The University Of Illinois | Methods for forming protected organoboronic acids |
US10500178B2 (en) | 2015-03-13 | 2019-12-10 | The Board Of Trustees Of The Leland Stanford Junior University | LTB4 inhibition to prevent and treat human lymphedema |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9119920D0 (en) * | 1991-09-18 | 1991-10-30 | Glaxo Group Ltd | Chemical compounds |
ES2098547T3 (es) * | 1992-01-23 | 1997-05-01 | Pfizer | Benzopirano y otros antagonistas de ltb4 relacionados. |
MX9300312A (es) * | 1992-01-23 | 1993-07-31 | Pfizer | Antagonistas benzopiranicos y relacionado de ltb. |
JPH07507811A (ja) * | 1992-10-21 | 1995-08-31 | ファイザー・インク. | 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸 |
KR950704309A (ko) * | 1992-10-21 | 1995-11-17 | 알렌 제이. 스피겔 | 벤젠융합된 하이드록시 치환-사이클로알킬 및 헤테로사이클릭 고리 화합물의 설폰아미드 유도체(sulfonamide derivatives of benzenefused hydroxy substituted cycloalkyl and heterocyclic ring compounds) |
MX9702734A (es) * | 1994-10-13 | 1997-06-28 | Pfizer | Benzopirano y compuestos benzocondensados, su preparacion y su uso como antagonistas de leucotrieno b4 (ltb4). |
KR100232341B1 (ko) * | 1994-10-13 | 2000-07-01 | 디. 제이. 우드 | 류코트리엔 b4(ltb4) 길항물질로서의 벤조피란 및 벤조-축합된 화합물 |
US5539128A (en) * | 1994-11-30 | 1996-07-23 | Pfizer Inc. | Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline |
-
1997
- 1997-08-25 ES ES97934679T patent/ES2206738T3/es not_active Expired - Lifetime
- 1997-08-25 BR BR9711482A patent/BR9711482A/pt not_active Application Discontinuation
- 1997-08-25 IL IL12873297A patent/IL128732A0/xx unknown
- 1997-08-25 NZ NZ334214A patent/NZ334214A/xx unknown
- 1997-08-25 US US09/367,235 patent/US6096906A/en not_active Expired - Fee Related
- 1997-08-25 JP JP10513430A patent/JP3117730B2/ja not_active Expired - Fee Related
- 1997-08-25 DK DK97934679T patent/DK0925292T3/da active
- 1997-08-25 DE DE69724801T patent/DE69724801T2/de not_active Expired - Fee Related
- 1997-08-25 EA EA199900204A patent/EA002204B1/ru not_active IP Right Cessation
- 1997-08-25 WO PCT/IB1997/001024 patent/WO1998011085A1/en not_active Application Discontinuation
- 1997-08-25 KR KR1019997002175A patent/KR100339164B1/ko not_active IP Right Cessation
- 1997-08-25 PL PL97332351A patent/PL332351A1/xx unknown
- 1997-08-25 UA UA99031394A patent/UA58520C2/uk unknown
- 1997-08-25 SK SK313-99A patent/SK31399A3/sk unknown
- 1997-08-25 CA CA002265043A patent/CA2265043C/en not_active Expired - Fee Related
- 1997-08-25 AU AU37814/97A patent/AU713701B2/en not_active Ceased
- 1997-08-25 EP EP97934679A patent/EP0925292B1/en not_active Expired - Lifetime
- 1997-08-25 PT PT97934679T patent/PT925292E/pt unknown
- 1997-08-25 CN CN97197985A patent/CN1108298C/zh not_active Expired - Fee Related
- 1997-08-25 AT AT97934679T patent/ATE249452T1/de not_active IP Right Cessation
- 1997-08-25 YU YU13299A patent/YU13299A/sh unknown
- 1997-08-25 TR TR1999/00592T patent/TR199900592T2/xx unknown
- 1997-08-29 HN HN1997000127A patent/HN1997000127A/es unknown
- 1997-09-04 CO CO97051475A patent/CO4600635A1/es unknown
- 1997-09-05 PA PA19978437901A patent/PA8437901A1/es unknown
- 1997-09-08 GT GT199700104A patent/GT199700104A/es unknown
- 1997-09-11 AP APAP/P/1997/001083A patent/AP726A/en active
- 1997-09-12 PE PE1997000813A patent/PE109798A1/es not_active Application Discontinuation
- 1997-09-12 TW TW086113297A patent/TW449579B/zh active
- 1997-09-15 MA MA24797A patent/MA24319A1/fr unknown
- 1997-09-15 TN TNTNSN97155A patent/TNSN97155A1/fr unknown
- 1997-09-15 DZ DZ970158A patent/DZ2308A1/xx active
- 1997-09-15 ID IDP973183A patent/ID19613A/id unknown
- 1997-09-15 ZA ZA978291A patent/ZA978291B/xx unknown
- 1997-09-16 HR HR970497A patent/HRP970497B1/xx not_active IP Right Cessation
- 1997-10-04 GT GT199700104BL patent/GT199700104BA/es unknown
- 1997-10-04 GT GT199700104AK patent/GT199700104AA/es unknown
-
1999
- 1999-02-16 IS IS4980A patent/IS4980A/is unknown
- 1999-03-09 BG BG103231A patent/BG63542B1/bg unknown
- 1999-03-12 OA OA9900056A patent/OA10995A/en unknown
- 1999-03-15 NO NO991254A patent/NO991254L/no not_active Application Discontinuation
-
2000
- 2000-02-23 US US09/511,475 patent/US6288242B1/en not_active Expired - Fee Related
-
2001
- 2001-03-21 US US09/813,546 patent/US6355825B1/en not_active Expired - Fee Related
- 2001-10-31 US US09/999,240 patent/US6444826B1/en not_active Expired - Fee Related
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