GT199700104BA - Procedimientos e intermedios para preparar derivados de cromanol sustituidos - Google Patents

Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Info

Publication number
GT199700104BA
GT199700104BA GT199700104BL GT199700104L GT199700104BA GT 199700104B A GT199700104B A GT 199700104BA GT 199700104B L GT199700104B L GT 199700104BL GT 199700104 L GT199700104 L GT 199700104L GT 199700104B A GT199700104B A GT 199700104BA
Authority
GT
Guatemala
Prior art keywords
intermediates
procedures
chromanol derivatives
substituted chromanol
prepare substituted
Prior art date
Application number
GT199700104BL
Other languages
English (en)
Inventor
Anthony Piscopio
Joel M Hawkins
Stephane Caron
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT199700104BA publication Critical patent/GT199700104BA/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/50Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds

Abstract

ESTA INVENCION SE REFIERE A LA PREPARACION DE DERIVADOS DE CROMANOL SUSTITUIDOS Y A INTERMEDIOS UTILES EN DICHA PREPARACION. LOS DERIVADOS DE CROMANOL SUSTITUIDOS QUE SE PREPARAN DE ACUERDO CON LA PRESENTE INVENCION, INHIBEN LA ACCION DE LTB4. ESTOS COMPUESTOS TIENEN LA ESTRUCTURA QUIMICA(XIII), EN LA QUE R3,R4,R7, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE.
GT199700104BL 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos GT199700104BA (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16

Publications (1)

Publication Number Publication Date
GT199700104BA true GT199700104BA (es) 1999-03-28

Family

ID=21831429

Family Applications (3)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.
GT199700104BL GT199700104BA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos
GT199700104AK GT199700104AA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Family Applications Before (1)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.

Family Applications After (1)

Application Number Title Priority Date Filing Date
GT199700104AK GT199700104AA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Country Status (39)

Country Link
US (4) US6096906A (es)
EP (1) EP0925292B1 (es)
JP (1) JP3117730B2 (es)
KR (1) KR100339164B1 (es)
CN (1) CN1108298C (es)
AP (1) AP726A (es)
AT (1) ATE249452T1 (es)
AU (1) AU713701B2 (es)
BG (1) BG63542B1 (es)
BR (1) BR9711482A (es)
CA (1) CA2265043C (es)
CO (1) CO4600635A1 (es)
DE (1) DE69724801T2 (es)
DK (1) DK0925292T3 (es)
DZ (1) DZ2308A1 (es)
EA (1) EA002204B1 (es)
ES (1) ES2206738T3 (es)
GT (3) GT199700104A (es)
HN (1) HN1997000127A (es)
HR (1) HRP970497B1 (es)
ID (1) ID19613A (es)
IL (1) IL128732A0 (es)
IS (1) IS4980A (es)
MA (1) MA24319A1 (es)
NO (1) NO991254L (es)
NZ (1) NZ334214A (es)
OA (1) OA10995A (es)
PA (1) PA8437901A1 (es)
PE (1) PE109798A1 (es)
PL (1) PL332351A1 (es)
PT (1) PT925292E (es)
SK (1) SK31399A3 (es)
TN (1) TNSN97155A1 (es)
TR (1) TR199900592T2 (es)
TW (1) TW449579B (es)
UA (1) UA58520C2 (es)
WO (1) WO1998011085A1 (es)
YU (1) YU13299A (es)
ZA (1) ZA978291B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
BR0206771A (pt) * 2001-01-30 2004-02-25 Pfizer Prod Inc Processos para a preparação de cidos cromanilbenzóicos
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
ES2551916T3 (es) 2007-07-23 2015-11-24 The Board Of Trustees Of The University Of Illinois Sistema para controlar la reactividad de los ácidos borónicos
WO2010036921A2 (en) 2008-09-26 2010-04-01 The Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
US8304513B2 (en) * 2009-09-02 2012-11-06 E I Du Pont De Nemours And Company Polyesters comprising fluorovinylether functionalized aromatic moieties
US8378061B2 (en) * 2009-09-02 2013-02-19 E.I. Du Pont De Nemours And Company Polyester films with improved oil repellency
TW201127822A (en) * 2009-09-02 2011-08-16 Du Pont Fluorinated 4-oxo-chroman-carboxylates
CN102612509A (zh) 2009-09-02 2012-07-25 纳幕尔杜邦公司 氟醚官能化的芳族二酯及其衍生物
CA2773142A1 (en) * 2009-09-02 2011-03-10 Neville Everton Drysdale Polyaramid comprising fluorovinylether functionalized aromatic moieties
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
US8557980B2 (en) 2010-02-18 2013-10-15 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
US10500178B2 (en) 2015-03-13 2019-12-10 The Board Of Trustees Of The Leland Stanford Junior University LTB4 inhibition to prevent and treat human lymphedema

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
ES2098547T3 (es) * 1992-01-23 1997-05-01 Pfizer Benzopirano y otros antagonistas de ltb4 relacionados.
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
JPH07507811A (ja) * 1992-10-21 1995-08-31 ファイザー・インク. 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸
KR950704309A (ko) * 1992-10-21 1995-11-17 알렌 제이. 스피겔 벤젠융합된 하이드록시 치환-사이클로알킬 및 헤테로사이클릭 고리 화합물의 설폰아미드 유도체(sulfonamide derivatives of benzenefused hydroxy substituted cycloalkyl and heterocyclic ring compounds)
MX9702734A (es) * 1994-10-13 1997-06-28 Pfizer Benzopirano y compuestos benzocondensados, su preparacion y su uso como antagonistas de leucotrieno b4 (ltb4).
KR100232341B1 (ko) * 1994-10-13 2000-07-01 디. 제이. 우드 류코트리엔 b4(ltb4) 길항물질로서의 벤조피란 및 벤조-축합된 화합물
US5539128A (en) * 1994-11-30 1996-07-23 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
UA58520C2 (uk) 2003-08-15
KR20000036136A (ko) 2000-06-26
TR199900592T2 (xx) 1999-06-21
NO991254L (no) 1999-05-14
CO4600635A1 (es) 1998-05-08
AU713701B2 (en) 1999-12-09
CN1230954A (zh) 1999-10-06
HRP970497A2 (en) 1998-08-31
CA2265043C (en) 2003-01-14
IS4980A (is) 1999-02-16
AP9701083A0 (en) 1997-10-31
SK31399A3 (en) 2000-05-16
WO1998011085A1 (en) 1998-03-19
US6288242B1 (en) 2001-09-11
PL332351A1 (en) 1999-09-13
US20020042526A1 (en) 2002-04-11
DE69724801T2 (de) 2004-06-17
CN1108298C (zh) 2003-05-14
ZA978291B (en) 1999-03-15
TNSN97155A1 (fr) 2005-03-15
BG63542B1 (bg) 2002-04-30
AU3781497A (en) 1998-04-02
AP726A (en) 1999-01-29
PT925292E (pt) 2004-01-30
DE69724801D1 (de) 2003-10-16
ATE249452T1 (de) 2003-09-15
PE109798A1 (es) 1999-01-13
NO991254D0 (no) 1999-03-15
MA24319A1 (fr) 1998-04-01
JP3117730B2 (ja) 2000-12-18
KR100339164B1 (ko) 2002-06-01
ID19613A (id) 1998-07-23
DK0925292T3 (da) 2004-01-12
US20020099227A1 (en) 2002-07-25
JP2000502726A (ja) 2000-03-07
PA8437901A1 (es) 2000-05-24
US6444826B1 (en) 2002-09-03
YU13299A (sh) 2001-03-07
EP0925292A1 (en) 1999-06-30
GT199700104AA (es) 1999-03-28
NZ334214A (en) 2000-09-29
HRP970497B1 (en) 2002-06-30
DZ2308A1 (fr) 2002-12-28
US6355825B1 (en) 2002-03-12
EP0925292B1 (en) 2003-09-10
HN1997000127A (es) 1997-12-20
BR9711482A (pt) 1999-08-24
US6096906A (en) 2000-08-01
TW449579B (en) 2001-08-11
GT199700104A (es) 1999-03-02
CA2265043A1 (en) 1998-03-19
BG103231A (en) 1999-12-30
ES2206738T3 (es) 2004-05-16
OA10995A (en) 2001-11-06
EA199900204A1 (ru) 1999-08-26
EA002204B1 (ru) 2002-02-28
IL128732A0 (en) 2000-01-31

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