PT925292E - Processos e intermediarios para a preparacao de derivados de cromanol substituido - Google Patents

Processos e intermediarios para a preparacao de derivados de cromanol substituido

Info

Publication number
PT925292E
PT925292E PT97934679T PT97934679T PT925292E PT 925292 E PT925292 E PT 925292E PT 97934679 T PT97934679 T PT 97934679T PT 97934679 T PT97934679 T PT 97934679T PT 925292 E PT925292 E PT 925292E
Authority
PT
Portugal
Prior art keywords
intermediaries
replaced
processes
preparation
chromanol derivatives
Prior art date
Application number
PT97934679T
Other languages
English (en)
Inventor
Anthony D Piscopio
Joel Michael Hawkins
Stephane Caron
Michael J Castaldi
Sarah E Kelly
Jeffrey W Raggon
Robert W Dugger
Sally G Ruggeri
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT925292E publication Critical patent/PT925292E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/50Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
PT97934679T 1996-09-16 1997-08-25 Processos e intermediarios para a preparacao de derivados de cromanol substituido PT925292E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16

Publications (1)

Publication Number Publication Date
PT925292E true PT925292E (pt) 2004-01-30

Family

ID=21831429

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97934679T PT925292E (pt) 1996-09-16 1997-08-25 Processos e intermediarios para a preparacao de derivados de cromanol substituido

Country Status (39)

Country Link
US (4) US6096906A (pt)
EP (1) EP0925292B1 (pt)
JP (1) JP3117730B2 (pt)
KR (1) KR100339164B1 (pt)
CN (1) CN1108298C (pt)
AP (1) AP726A (pt)
AT (1) ATE249452T1 (pt)
AU (1) AU713701B2 (pt)
BG (1) BG63542B1 (pt)
BR (1) BR9711482A (pt)
CA (1) CA2265043C (pt)
CO (1) CO4600635A1 (pt)
DE (1) DE69724801T2 (pt)
DK (1) DK0925292T3 (pt)
DZ (1) DZ2308A1 (pt)
EA (1) EA002204B1 (pt)
ES (1) ES2206738T3 (pt)
GT (3) GT199700104A (pt)
HN (1) HN1997000127A (pt)
HR (1) HRP970497B1 (pt)
ID (1) ID19613A (pt)
IL (1) IL128732A0 (pt)
IS (1) IS4980A (pt)
MA (1) MA24319A1 (pt)
NO (1) NO991254L (pt)
NZ (1) NZ334214A (pt)
OA (1) OA10995A (pt)
PA (1) PA8437901A1 (pt)
PE (1) PE109798A1 (pt)
PL (1) PL332351A1 (pt)
PT (1) PT925292E (pt)
SK (1) SK31399A3 (pt)
TN (1) TNSN97155A1 (pt)
TR (1) TR199900592T2 (pt)
TW (1) TW449579B (pt)
UA (1) UA58520C2 (pt)
WO (1) WO1998011085A1 (pt)
YU (1) YU13299A (pt)
ZA (1) ZA978291B (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
BR0206771A (pt) * 2001-01-30 2004-02-25 Pfizer Prod Inc Processos para a preparação de cidos cromanilbenzóicos
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
ES2551916T3 (es) 2007-07-23 2015-11-24 The Board Of Trustees Of The University Of Illinois Sistema para controlar la reactividad de los ácidos borónicos
WO2010036921A2 (en) 2008-09-26 2010-04-01 The Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
US8304513B2 (en) * 2009-09-02 2012-11-06 E I Du Pont De Nemours And Company Polyesters comprising fluorovinylether functionalized aromatic moieties
US8378061B2 (en) * 2009-09-02 2013-02-19 E.I. Du Pont De Nemours And Company Polyester films with improved oil repellency
TW201127822A (en) * 2009-09-02 2011-08-16 Du Pont Fluorinated 4-oxo-chroman-carboxylates
CN102612509A (zh) 2009-09-02 2012-07-25 纳幕尔杜邦公司 氟醚官能化的芳族二酯及其衍生物
CA2773142A1 (en) * 2009-09-02 2011-03-10 Neville Everton Drysdale Polyaramid comprising fluorovinylether functionalized aromatic moieties
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
US8557980B2 (en) 2010-02-18 2013-10-15 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
US10500178B2 (en) 2015-03-13 2019-12-10 The Board Of Trustees Of The Leland Stanford Junior University LTB4 inhibition to prevent and treat human lymphedema

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
ES2098547T3 (es) * 1992-01-23 1997-05-01 Pfizer Benzopirano y otros antagonistas de ltb4 relacionados.
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
JPH07507811A (ja) * 1992-10-21 1995-08-31 ファイザー・インク. 鏡像異性のシス−3−(4,6−ジヒドロキシクロマン−3−イル−メチル)安息香酸
KR950704309A (ko) * 1992-10-21 1995-11-17 알렌 제이. 스피겔 벤젠융합된 하이드록시 치환-사이클로알킬 및 헤테로사이클릭 고리 화합물의 설폰아미드 유도체(sulfonamide derivatives of benzenefused hydroxy substituted cycloalkyl and heterocyclic ring compounds)
MX9702734A (es) * 1994-10-13 1997-06-28 Pfizer Benzopirano y compuestos benzocondensados, su preparacion y su uso como antagonistas de leucotrieno b4 (ltb4).
KR100232341B1 (ko) * 1994-10-13 2000-07-01 디. 제이. 우드 류코트리엔 b4(ltb4) 길항물질로서의 벤조피란 및 벤조-축합된 화합물
US5539128A (en) * 1994-11-30 1996-07-23 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
GT199700104BA (es) 1999-03-28
UA58520C2 (uk) 2003-08-15
KR20000036136A (ko) 2000-06-26
TR199900592T2 (xx) 1999-06-21
NO991254L (no) 1999-05-14
CO4600635A1 (es) 1998-05-08
AU713701B2 (en) 1999-12-09
CN1230954A (zh) 1999-10-06
HRP970497A2 (en) 1998-08-31
CA2265043C (en) 2003-01-14
IS4980A (is) 1999-02-16
AP9701083A0 (en) 1997-10-31
SK31399A3 (en) 2000-05-16
WO1998011085A1 (en) 1998-03-19
US6288242B1 (en) 2001-09-11
PL332351A1 (en) 1999-09-13
US20020042526A1 (en) 2002-04-11
DE69724801T2 (de) 2004-06-17
CN1108298C (zh) 2003-05-14
ZA978291B (en) 1999-03-15
TNSN97155A1 (fr) 2005-03-15
BG63542B1 (bg) 2002-04-30
AU3781497A (en) 1998-04-02
AP726A (en) 1999-01-29
DE69724801D1 (de) 2003-10-16
ATE249452T1 (de) 2003-09-15
PE109798A1 (es) 1999-01-13
NO991254D0 (no) 1999-03-15
MA24319A1 (fr) 1998-04-01
JP3117730B2 (ja) 2000-12-18
KR100339164B1 (ko) 2002-06-01
ID19613A (id) 1998-07-23
DK0925292T3 (da) 2004-01-12
US20020099227A1 (en) 2002-07-25
JP2000502726A (ja) 2000-03-07
PA8437901A1 (es) 2000-05-24
US6444826B1 (en) 2002-09-03
YU13299A (sh) 2001-03-07
EP0925292A1 (en) 1999-06-30
GT199700104AA (es) 1999-03-28
NZ334214A (en) 2000-09-29
HRP970497B1 (en) 2002-06-30
DZ2308A1 (fr) 2002-12-28
US6355825B1 (en) 2002-03-12
EP0925292B1 (en) 2003-09-10
HN1997000127A (es) 1997-12-20
BR9711482A (pt) 1999-08-24
US6096906A (en) 2000-08-01
TW449579B (en) 2001-08-11
GT199700104A (es) 1999-03-02
CA2265043A1 (en) 1998-03-19
BG103231A (en) 1999-12-30
ES2206738T3 (es) 2004-05-16
OA10995A (en) 2001-11-06
EA199900204A1 (ru) 1999-08-26
EA002204B1 (ru) 2002-02-28
IL128732A0 (en) 2000-01-31

Similar Documents

Publication Publication Date Title
DE69716296D1 (de) Indan- oder dihydroindolderivate
BR9507179A (pt) Derivados de 3-aril-4-hidróxi-delta3-dihidrotiofena
DK0746310T3 (da) Præparat med styret afgivelse
MX9202290A (es) Nuevos derivados de tiopiranopirrol y procedimiento para su preparacion.
PT850948E (pt) Derivados propiofenona e processo para a preparacao dos mesmos
PT977748E (pt) Derivados benzopirano substituidos para o tratamento de inflamacao
AR002651A1 (es) Procedimiento integrado para la producción de 1-buteno
BR9708386A (pt) Derivados de 6-fenilpiridil-2-amina
PT831098E (pt) Intermediarios e processo para a preparacao de olanzapina
EE200000140A (et) Asendatud kromaani derivaadid
PT925292E (pt) Processos e intermediarios para a preparacao de derivados de cromanol substituido
PT888291E (pt) Novos processos para a preparacao de intermediarios pesticidas
BR9509793A (pt) Derivados de tiofeneno
EE200000144A (et) Asendatud kromaani derivaadid
MX21917A (es) Derivados de benzopirano y benzotiopirano y procedimiento para su preparacion.
PT1004583E (pt) Processos e intermediarios hidantoinicos para a sintese de secretagogos da hormona do crescimento
PT1028960E (pt) Processo para a preparacao de derivados de tiazolidinodiona
PT983249E (pt) Procesos e intermediarios para a preparacao de derivados de indazole substituidos
PT970080E (pt) Derivados de imino-aza-antraciclinona para o tartamento de amiloidoses
BR9506618A (pt) Derivados de difeniloxazolinas
PT1073627E (pt) Processos para a preparacao de intermediarios pesticidas
BR9509877A (pt) Novos derivados de pirimidinilóxi-e piridimidinilamino- etilfenil-dioxolano
DE29601701U1 (de) Sicherheitsbandage
BR9708310A (pt) Derivados de 2-tioxotetrahidropirimidin-4-ona
BR9708461A (pt) Derivados de butadieno e processos para sua preparação