BG106508A - Alkylene diamine-substituted heterocycles - Google Patents
Alkylene diamine-substituted heterocyclesInfo
- Publication number
- BG106508A BG106508A BG106508A BG10650802A BG106508A BG 106508 A BG106508 A BG 106508A BG 106508 A BG106508 A BG 106508A BG 10650802 A BG10650802 A BG 10650802A BG 106508 A BG106508 A BG 106508A
- Authority
- BG
- Bulgaria
- Prior art keywords
- attached
- double bond
- adjacent ring
- atom
- single bond
- Prior art date
Links
- 125000000623 heterocyclic group Chemical class 0.000 title abstract 2
- 125000002947 alkylene group Chemical group 0.000 title 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 4
- 125000006413 ring segment Chemical group 0.000 abstract 4
- 229910052799 carbon Inorganic materials 0.000 abstract 3
- 229910052717 sulfur Inorganic materials 0.000 abstract 3
- 101710151321 Melanostatin Proteins 0.000 abstract 2
- 101150027439 NPY1 gene Proteins 0.000 abstract 2
- 102400000064 Neuropeptide Y Human genes 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- URPYMXQQVHTUDU-OFGSCBOVSA-N nucleopeptide y Chemical compound C([C@@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(N)=O)NC(=O)[C@H](CC=1NC=NC=1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CC=1C=CC(O)=CC=1)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](C)NC(=O)[C@H]1N(CCC1)C(=O)[C@H](C)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H](CCC(O)=O)NC(=O)CNC(=O)[C@H]1N(CCC1)C(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(O)=O)NC(=O)[C@H]1N(CCC1)C(=O)[C@H](CCCCN)NC(=O)[C@H](CO)NC(=O)[C@H]1N(CCC1)C(=O)[C@@H](N)CC=1C=CC(O)=CC=1)C1=CC=C(O)C=C1 URPYMXQQVHTUDU-OFGSCBOVSA-N 0.000 abstract 2
- 239000002464 receptor antagonist Substances 0.000 abstract 2
- 229940044551 receptor antagonist Drugs 0.000 abstract 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- 101000869592 Daucus carota Major allergen Dau c 1 Proteins 0.000 abstract 1
- 101000650136 Homo sapiens WAS/WASL-interacting protein family member 3 Proteins 0.000 abstract 1
- 101000585507 Solanum tuberosum Cytochrome b-c1 complex subunit 7 Proteins 0.000 abstract 1
- 102100027539 WAS/WASL-interacting protein family member 3 Human genes 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 238000007429 general method Methods 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 108090000765 processed proteins & peptides Proteins 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
- 125000000169 tricyclic heterocycle group Chemical group 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/73—Unsubstituted amino or imino radicals
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C07D215/46—Nitrogen atoms attached in position 4 with hydrocarbon radicals, substituted by nitrogen atoms, attached to said nitrogen atoms
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- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
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- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
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- Organic Chemistry (AREA)
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- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- General Health & Medical Sciences (AREA)
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- Neurosurgery (AREA)
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- Neurology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Pulmonology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Anesthesiology (AREA)
- Child & Adolescent Psychology (AREA)
- Rheumatology (AREA)
- Emergency Medicine (AREA)
- Vascular Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US15687099P | 1999-09-30 | 1999-09-30 | |
PCT/US2000/026886 WO2001023389A2 (en) | 1999-09-30 | 2000-09-29 | Certain alkylene diamine-substituted heterocycles |
Publications (1)
Publication Number | Publication Date |
---|---|
BG106508A true BG106508A (en) | 2003-02-28 |
Family
ID=22561438
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BG106508A BG106508A (en) | 1999-09-30 | 2002-03-11 | Alkylene diamine-substituted heterocycles |
Country Status (21)
Country | Link |
---|---|
US (3) | US6506762B1 (de) |
EP (1) | EP1224187B1 (de) |
JP (2) | JP2003510327A (de) |
KR (1) | KR20020043223A (de) |
CN (1) | CN1377356A (de) |
AT (1) | ATE318267T1 (de) |
AU (1) | AU7738000A (de) |
BG (1) | BG106508A (de) |
CA (1) | CA2379640C (de) |
CZ (1) | CZ20021086A3 (de) |
DE (1) | DE60026155T2 (de) |
EA (1) | EA200200424A1 (de) |
ES (1) | ES2258476T3 (de) |
HU (1) | HUP0202636A3 (de) |
IL (1) | IL148903A0 (de) |
NO (1) | NO20021358L (de) |
NZ (1) | NZ517575A (de) |
OA (1) | OA12050A (de) |
PL (1) | PL354784A1 (de) |
WO (1) | WO2001023389A2 (de) |
ZA (1) | ZA200202518B (de) |
Families Citing this family (151)
Publication number | Priority date | Publication date | Assignee | Title |
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-
2000
- 2000-09-29 EA EA200200424A patent/EA200200424A1/ru unknown
- 2000-09-29 EP EP00967133A patent/EP1224187B1/de not_active Expired - Lifetime
- 2000-09-29 KR KR1020027004150A patent/KR20020043223A/ko not_active Application Discontinuation
- 2000-09-29 HU HU0202636A patent/HUP0202636A3/hu unknown
- 2000-09-29 IL IL14890300A patent/IL148903A0/xx unknown
- 2000-09-29 AT AT00967133T patent/ATE318267T1/de not_active IP Right Cessation
- 2000-09-29 JP JP2001526541A patent/JP2003510327A/ja active Pending
- 2000-09-29 ES ES00967133T patent/ES2258476T3/es not_active Expired - Lifetime
- 2000-09-29 US US09/676,941 patent/US6506762B1/en not_active Expired - Fee Related
- 2000-09-29 AU AU77380/00A patent/AU7738000A/en not_active Abandoned
- 2000-09-29 NZ NZ517575A patent/NZ517575A/en unknown
- 2000-09-29 DE DE60026155T patent/DE60026155T2/de not_active Expired - Fee Related
- 2000-09-29 PL PL00354784A patent/PL354784A1/xx not_active Application Discontinuation
- 2000-09-29 CZ CZ20021086A patent/CZ20021086A3/cs unknown
- 2000-09-29 CA CA002379640A patent/CA2379640C/en not_active Expired - Fee Related
- 2000-09-29 OA OA1200200089A patent/OA12050A/en unknown
- 2000-09-29 WO PCT/US2000/026886 patent/WO2001023389A2/en active IP Right Grant
- 2000-09-29 CN CN00813704A patent/CN1377356A/zh active Pending
-
2002
- 2002-03-11 BG BG106508A patent/BG106508A/xx unknown
- 2002-03-19 NO NO20021358A patent/NO20021358L/no not_active Application Discontinuation
- 2002-03-28 ZA ZA200202518A patent/ZA200202518B/xx unknown
- 2002-11-08 US US10/291,446 patent/US6696445B2/en not_active Expired - Fee Related
-
2003
- 2003-11-10 US US10/705,446 patent/US7074929B2/en not_active Expired - Fee Related
-
2007
- 2007-08-22 JP JP2007215782A patent/JP2008007515A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
JP2008007515A (ja) | 2008-01-17 |
KR20020043223A (ko) | 2002-06-08 |
US6506762B1 (en) | 2003-01-14 |
CN1377356A (zh) | 2002-10-30 |
NO20021358D0 (no) | 2002-03-19 |
NZ517575A (en) | 2004-04-30 |
ES2258476T3 (es) | 2006-09-01 |
EA200200424A1 (ru) | 2002-12-26 |
AU7738000A (en) | 2001-04-30 |
NO20021358L (no) | 2002-05-27 |
WO2001023389A2 (en) | 2001-04-05 |
HUP0202636A3 (en) | 2004-06-28 |
ATE318267T1 (de) | 2006-03-15 |
IL148903A0 (en) | 2002-09-12 |
CZ20021086A3 (cs) | 2002-10-16 |
US7074929B2 (en) | 2006-07-11 |
US20030158197A1 (en) | 2003-08-21 |
OA12050A (en) | 2006-05-02 |
CA2379640C (en) | 2006-11-28 |
EP1224187A2 (de) | 2002-07-24 |
EP1224187B1 (de) | 2006-02-22 |
PL354784A1 (en) | 2004-02-23 |
ZA200202518B (en) | 2003-08-27 |
WO2001023389A3 (en) | 2002-05-10 |
HUP0202636A2 (hu) | 2002-12-28 |
DE60026155D1 (de) | 2006-04-27 |
CA2379640A1 (en) | 2001-04-05 |
DE60026155T2 (de) | 2006-08-10 |
US6696445B2 (en) | 2004-02-24 |
JP2003510327A (ja) | 2003-03-18 |
US20040229870A1 (en) | 2004-11-18 |
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