BG103189A - Substituted 6,5-heterobicyclic derivatives - Google Patents

Substituted 6,5-heterobicyclic derivatives

Info

Publication number
BG103189A
BG103189A BG103189A BG10318999A BG103189A BG 103189 A BG103189 A BG 103189A BG 103189 A BG103189 A BG 103189A BG 10318999 A BG10318999 A BG 10318999A BG 103189 A BG103189 A BG 103189A
Authority
BG
Bulgaria
Prior art keywords
nitrogen
carbon
substituted
compounds
heterobicyclic derivatives
Prior art date
Application number
BG103189A
Other languages
Bulgarian (bg)
English (en)
Inventor
Yuhpyng Chen
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21823717&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BG103189(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of BG103189A publication Critical patent/BG103189A/xx

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Addiction (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Virology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Communicable Diseases (AREA)
BG103189A 1996-08-28 1999-02-22 Substituted 6,5-heterobicyclic derivatives BG103189A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2503996P 1996-08-28 1996-08-28
PCT/IB1997/000922 WO1998008847A1 (en) 1996-08-28 1997-07-25 Substituted 6,5-hetero-bicyclic derivatives

Publications (1)

Publication Number Publication Date
BG103189A true BG103189A (en) 1999-09-30

Family

ID=21823717

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103189A BG103189A (en) 1996-08-28 1999-02-22 Substituted 6,5-heterobicyclic derivatives

Country Status (36)

Country Link
EP (1) EP0923582B1 (de)
JP (2) JP3621706B2 (de)
KR (1) KR20000035934A (de)
CN (1) CN1227554A (de)
AP (1) AP762A (de)
AR (1) AR015103A1 (de)
AT (1) ATE340176T1 (de)
AU (1) AU735401B2 (de)
BG (1) BG103189A (de)
BR (1) BR9711970A (de)
CA (1) CA2263566C (de)
CO (1) CO4600634A1 (de)
CZ (1) CZ68199A3 (de)
DE (1) DE69736711T2 (de)
DZ (1) DZ2300A1 (de)
EA (1) EA002769B1 (de)
ES (1) ES2273369T3 (de)
GT (1) GT199700095A (de)
HR (1) HRP970454B1 (de)
HU (1) HUP9903965A3 (de)
ID (1) ID18249A (de)
IL (1) IL127566A0 (de)
IS (1) IS4963A (de)
MA (1) MA26438A1 (de)
NO (1) NO313636B1 (de)
NZ (1) NZ333302A (de)
OA (1) OA10977A (de)
PA (1) PA8436201A1 (de)
PE (1) PE108898A1 (de)
PL (1) PL332040A1 (de)
SK (1) SK23399A3 (de)
TN (1) TNSN97145A1 (de)
TR (1) TR199900389T2 (de)
TW (1) TW575573B (de)
WO (1) WO1998008847A1 (de)
ZA (1) ZA977687B (de)

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US6313124B1 (en) 1997-07-23 2001-11-06 Dupont Pharmaceuticals Company Tetrazine bicyclic compounds
US6191131B1 (en) 1997-07-23 2001-02-20 Dupont Pharmaceuticals Company Azolo triazines and pyrimidines
US6060478A (en) * 1996-07-24 2000-05-09 Dupont Pharmaceuticals Azolo triazines and pyrimidines
US7094782B1 (en) 1996-07-24 2006-08-22 Bristol-Myers Squibb Company Azolo triazines and pyrimidines
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WO1998035967A2 (en) * 1997-02-18 1998-08-20 Neurocrine Biosciences, Inc. Biazacyclic crf antagonists
JP2002501493A (ja) 1997-04-22 2002-01-15 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ Crfアンタゴニストのチオフェノピリジン類
HRP980375A2 (en) * 1997-07-03 1999-04-30 Argyrios Georgios Arvanitis Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders
EP1344779B1 (de) * 1998-01-28 2005-08-10 Bristol-Myers Squibb Pharma Company Azolo-Pyrimidine
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
AU3375999A (en) 1998-04-02 1999-10-25 Neurogen Corporation Aminoalkyl substituted 5,6,7,8-tetrahydro-9h pyrimidino(2,3-b)indole and 5,6,7,8-tetrahydro-9h-pyrimidino(4,5-b)indole derivatives: crf1 specific ligands
US6472402B1 (en) 1998-04-02 2002-10-29 Neurogen Corporation Aminoalkyl substituted 5,6,7,8-Tetrahydro-9H-Pyridino [2,3-B]indole derivatives
WO1999051608A1 (en) * 1998-04-03 1999-10-14 Du Pont Pharmaceuticals Company THIAZOLO[4,5-d]PYRIMIDINES AND PYRIDINES AS CORTICOTROPIN RELEASING FACTOR (CRF) ANTAGONISTS
CA2334671A1 (en) 1998-06-09 1999-12-16 Neurogen Corporation Pyrido[2,3-b]indolizine derivatives and aza analogues thereof; crf1 specific ligands
US6509338B1 (en) 1998-06-22 2003-01-21 Bristol-Myers Squibb Company Pyrazolo[1,5-A]triazine corticotropin releasing factor antagonists
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