AU666902B2 - Biaryl substituted 4-amino-butyric acid amides - Google Patents

Biaryl substituted 4-amino-butyric acid amides Download PDF

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Publication number
AU666902B2
AU666902B2 AU31842/93A AU3184293A AU666902B2 AU 666902 B2 AU666902 B2 AU 666902B2 AU 31842/93 A AU31842/93 A AU 31842/93A AU 3184293 A AU3184293 A AU 3184293A AU 666902 B2 AU666902 B2 AU 666902B2
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Australia
Prior art keywords
lower alkyl
aryl
coor
amino
carboxyl
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Expired - Fee Related
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AU31842/93A
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AU3184293A (en
Inventor
Gary Ksander
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Novartis AG
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Ciba Geigy AG
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Publication of AU3184293A publication Critical patent/AU3184293A/en
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Anticipated expiration legal-status Critical
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/47—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom having the carbon atom of the carboxamide group bound to a hydrogen atom or to a carbon atom of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/04—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C235/12—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atom of at least one of the carboxamide groups bound to an acyclic carbon atom of a hydrocarbon radical substituted by carboxyl groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU31842/93A 1992-01-22 1993-01-15 Biaryl substituted 4-amino-butyric acid amides Expired - Fee Related AU666902B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US824132 1992-01-22
US07/824,132 US5217996A (en) 1992-01-22 1992-01-22 Biaryl substituted 4-amino-butyric acid amides

Publications (2)

Publication Number Publication Date
AU3184293A AU3184293A (en) 1993-07-29
AU666902B2 true AU666902B2 (en) 1996-02-29

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ID=25240671

Family Applications (1)

Application Number Title Priority Date Filing Date
AU31842/93A Expired - Fee Related AU666902B2 (en) 1992-01-22 1993-01-15 Biaryl substituted 4-amino-butyric acid amides

Country Status (14)

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US (2) US5217996A (show.php)
EP (1) EP0555175A1 (show.php)
JP (1) JPH05310664A (show.php)
KR (1) KR930016393A (show.php)
AU (1) AU666902B2 (show.php)
CA (1) CA2087652A1 (show.php)
FI (1) FI930195A7 (show.php)
HU (1) HUT63376A (show.php)
IL (1) IL104387A0 (show.php)
MX (1) MX9300310A (show.php)
NO (1) NO930193L (show.php)
NZ (1) NZ245716A (show.php)
TW (1) TW228513B (show.php)
ZA (1) ZA93421B (show.php)

Families Citing this family (138)

* Cited by examiner, † Cited by third party
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