AU2006239929B2 - Dipeptidyl peptidase-IV inhibitors - Google Patents

Dipeptidyl peptidase-IV inhibitors Download PDF

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Publication number
AU2006239929B2
AU2006239929B2 AU2006239929A AU2006239929A AU2006239929B2 AU 2006239929 B2 AU2006239929 B2 AU 2006239929B2 AU 2006239929 A AU2006239929 A AU 2006239929A AU 2006239929 A AU2006239929 A AU 2006239929A AU 2006239929 B2 AU2006239929 B2 AU 2006239929B2
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AU
Australia
Prior art keywords
alkyl
mixture
title compound
afford
pct
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AU2006239929A
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AU2006239929A1 (en
Inventor
Jurgen Boer
Michael Essers
Tim Feuerstein
Fritz-Frieder Frickel
Matthias Hochguertel
Heiko Kroth
Bert Nolte
Frank Richter
Matthias Schneider
Christoph Steeneck
Arthur Taveras
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Alantos Pharmaceuticals Holding Inc
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Alantos Pharmaceuticals Holding Inc
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Application filed by Alantos Pharmaceuticals Holding Inc filed Critical Alantos Pharmaceuticals Holding Inc
Publication of AU2006239929A1 publication Critical patent/AU2006239929A1/en
Priority to AU2010201511A priority Critical patent/AU2010201511B2/en
Application granted granted Critical
Publication of AU2006239929B2 publication Critical patent/AU2006239929B2/en
Anticipated expiration legal-status Critical
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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AU2006239929A 2005-04-22 2006-04-21 Dipeptidyl peptidase-IV inhibitors Ceased AU2006239929B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2010201511A AU2010201511B2 (en) 2005-04-22 2010-04-15 Dipeptidyl peptidase-IV inhibitors

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US67415105P 2005-04-22 2005-04-22
US60/674,151 2005-04-22
PCT/US2006/015200 WO2006116157A2 (en) 2005-04-22 2006-04-21 Dipeptidyl peptidase-iv inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
AU2010201511A Division AU2010201511B2 (en) 2005-04-22 2010-04-15 Dipeptidyl peptidase-IV inhibitors

Publications (2)

Publication Number Publication Date
AU2006239929A1 AU2006239929A1 (en) 2006-11-02
AU2006239929B2 true AU2006239929B2 (en) 2011-11-03

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AU2006239929A Ceased AU2006239929B2 (en) 2005-04-22 2006-04-21 Dipeptidyl peptidase-IV inhibitors
AU2010201511A Ceased AU2010201511B2 (en) 2005-04-22 2010-04-15 Dipeptidyl peptidase-IV inhibitors

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AU2010201511A Ceased AU2010201511B2 (en) 2005-04-22 2010-04-15 Dipeptidyl peptidase-IV inhibitors

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US (3) US7553861B2 (OSRAM)
EP (1) EP1888562B1 (OSRAM)
JP (2) JP4568361B2 (OSRAM)
KR (1) KR20080000665A (OSRAM)
CN (1) CN101277949A (OSRAM)
AP (1) AP2007004234A0 (OSRAM)
AU (2) AU2006239929B2 (OSRAM)
BR (1) BRPI0608469A2 (OSRAM)
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ZA (1) ZA200708179B (OSRAM)

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