ATE207489T1 - Benzimidazolderivate, deren herstellung und deren therapeutische anwendung - Google Patents

Benzimidazolderivate, deren herstellung und deren therapeutische anwendung

Info

Publication number
ATE207489T1
ATE207489T1 AT96303940T AT96303940T ATE207489T1 AT E207489 T1 ATE207489 T1 AT E207489T1 AT 96303940 T AT96303940 T AT 96303940T AT 96303940 T AT96303940 T AT 96303940T AT E207489 T1 ATE207489 T1 AT E207489T1
Authority
AT
Austria
Prior art keywords
ylmethyl
dioxothiazolidin
production
therapeutic use
benzimidazole derivatives
Prior art date
Application number
AT96303940T
Other languages
English (en)
Inventor
Takashi Fujita
Kunio Wada
Minoru Oguchi
Hiroaki Yanagisawa
Koichi Fujimoto
Toshihiko Fujiwara
Hiroyoshi Horikoshi
Takao Yoshioka
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26385935&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE207489(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sankyo Co filed Critical Sankyo Co
Application granted granted Critical
Publication of ATE207489T1 publication Critical patent/ATE207489T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/12—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT96303940T 1995-06-01 1996-05-31 Benzimidazolderivate, deren herstellung und deren therapeutische anwendung ATE207489T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP13509795 1995-06-01
JP4584596 1996-03-04

Publications (1)

Publication Number Publication Date
ATE207489T1 true ATE207489T1 (de) 2001-11-15

Family

ID=26385935

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96303940T ATE207489T1 (de) 1995-06-01 1996-05-31 Benzimidazolderivate, deren herstellung und deren therapeutische anwendung

Country Status (20)

Country Link
US (1) US5886014A (de)
EP (1) EP0745600B1 (de)
JP (2) JP2976885B2 (de)
KR (2) KR100485425B1 (de)
CN (1) CN1066729C (de)
AT (1) ATE207489T1 (de)
AU (1) AU712390B2 (de)
CA (1) CA2177858C (de)
CZ (1) CZ293016B6 (de)
DE (1) DE69616151T2 (de)
DK (1) DK0745600T3 (de)
ES (1) ES2164841T3 (de)
HU (1) HU225778B1 (de)
IL (1) IL118474A (de)
MX (1) MX9602122A (de)
NO (1) NO308744B1 (de)
NZ (1) NZ286716A (de)
PT (1) PT745600E (de)
RU (1) RU2125048C1 (de)
TW (1) TW449594B (de)

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IL118474A0 (en) 1996-09-12
MX9602122A (es) 1997-06-28
DE69616151D1 (de) 2001-11-29
JP3249490B2 (ja) 2002-01-21
TW449594B (en) 2001-08-11
EP0745600B1 (de) 2001-10-24
HK1002280A1 (en) 1998-08-14
HUP9601492A3 (en) 1998-10-28
JP2976885B2 (ja) 1999-11-10
NO308744B1 (no) 2000-10-23
HUP9601492A2 (hu) 1998-08-28
NO962239L (no) 1996-12-02
CN1066729C (zh) 2001-06-06
KR100485425B1 (ko) 2005-10-27
RU2125048C1 (ru) 1999-01-20
HU9601492D0 (en) 1996-07-29
NO962239D0 (no) 1996-05-31
HK1011683A1 (en) 1999-07-16
US5886014A (en) 1999-03-23
CZ156796A3 (en) 1996-12-11
JPH09295970A (ja) 1997-11-18
CN1157288A (zh) 1997-08-20
KR100493772B1 (ko) 2005-06-08
KR970001349A (ko) 1997-01-24
ES2164841T3 (es) 2002-03-01
HU225778B1 (en) 2007-08-28
PT745600E (pt) 2002-02-28
JP2000001487A (ja) 2000-01-07
CA2177858C (en) 2010-07-06
AU712390B2 (en) 1999-11-04
AU5462796A (en) 1996-12-12
CA2177858A1 (en) 1996-12-02
CZ293016B6 (cs) 2004-01-14
IL118474A (en) 2001-08-08
DE69616151T2 (de) 2002-07-11
DK0745600T3 (da) 2001-11-12
EP0745600A1 (de) 1996-12-04
NZ286716A (en) 1997-08-22

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