ATA276783A - Verfahren zur herstellung einer amorphen form des (6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl -2-methoxyiminoacetamido)-ceph-3-em-4-carbonsaeu e-1 acetoxyethylesters - Google Patents

Verfahren zur herstellung einer amorphen form des (6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl -2-methoxyiminoacetamido)-ceph-3-em-4-carbonsaeu e-1 acetoxyethylesters

Info

Publication number
ATA276783A
ATA276783A AT0276783A AT276783A ATA276783A AT A276783 A ATA276783 A AT A276783A AT 0276783 A AT0276783 A AT 0276783A AT 276783 A AT276783 A AT 276783A AT A276783 A ATA276783 A AT A276783A
Authority
AT
Austria
Prior art keywords
carbonsaeu
acetoxyethylesters
methoxyiminoacetamido
carbamoyloxymethyl
ceph
Prior art date
Application number
AT0276783A
Other languages
English (en)
Other versions
AT382154B (de
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10532012&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATA276783(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of ATA276783A publication Critical patent/ATA276783A/de
Application granted granted Critical
Publication of AT382154B publication Critical patent/AT382154B/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AT0276783A 1982-07-30 1983-07-29 Verfahren zur herstellung einer amorphen form des (6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl -2-methoxyiminoacetamido)-ceph-3-em-4-carbonsaeu e-1 acetoxyethylesters AT382154B (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8222019 1982-07-30

Publications (2)

Publication Number Publication Date
ATA276783A true ATA276783A (de) 1986-06-15
AT382154B AT382154B (de) 1987-01-26

Family

ID=10532012

Family Applications (1)

Application Number Title Priority Date Filing Date
AT0276783A AT382154B (de) 1982-07-30 1983-07-29 Verfahren zur herstellung einer amorphen form des (6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl -2-methoxyiminoacetamido)-ceph-3-em-4-carbonsaeu e-1 acetoxyethylesters

Country Status (41)

Country Link
US (4) US4562181A (de)
EP (1) EP0107276B1 (de)
JP (1) JPH0730084B2 (de)
KR (1) KR910000046B1 (de)
AT (1) AT382154B (de)
AU (1) AU566881B2 (de)
BE (1) BE897422A (de)
CA (1) CA1240313A (de)
CH (1) CH657134A5 (de)
CS (1) CS259515B2 (de)
CY (1) CY1434A (de)
CZ (1) CZ280528B6 (de)
DE (2) DE3327449A1 (de)
DK (2) DK164507C (de)
DO (1) DOP1990004773A (de)
EC (1) ECSP941098A (de)
ES (1) ES524590A0 (de)
FI (1) FI76093C (de)
FR (1) FR2531087B1 (de)
GB (1) GB2127401B (de)
GR (1) GR79349B (de)
HK (1) HK84288A (de)
HU (1) HU190603B (de)
IE (1) IE55748B1 (de)
IL (1) IL69375A (de)
IT (1) IT1168206B (de)
KE (1) KE3805A (de)
LU (1) LU84935A1 (de)
MY (1) MY8700058A (de)
NL (1) NL8302705A (de)
NO (1) NO163897C (de)
NZ (1) NZ205083A (de)
PL (1) PL156001B1 (de)
PT (1) PT77135B (de)
SE (1) SE453195B (de)
SG (1) SG26088G (de)
SK (1) SK403191A3 (de)
SU (1) SU1266471A3 (de)
YU (1) YU44680B (de)
ZA (1) ZA835579B (de)
ZW (1) ZW17383A1 (de)

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KR100363566B1 (ko) * 1998-11-20 2003-08-19 국제약품공업주식회사 무정형 세푸록심 악세틸의 제조방법
AT413647B (de) * 1998-11-26 2006-04-15 Sandoz Ag Verwendung eines copolymerisats aus 1-vinyl-2-pyrrolidon und vinylacetat zur herstellung von cefuroximaxetil-hältigen tabletten
EP1165051B1 (de) 1999-03-19 2003-07-09 Ranbaxy Laboratories, Ltd. Verfahren zur herstellung einer bioverfügbaren oralen darreichungsform von cefuroxim-axetil
IN191492B (de) * 1999-05-25 2003-12-06 Ranbaxy Lab Ltd
IN191236B (de) 1999-05-25 2003-10-11 Ranbaxy Lab Ltd
US6930983B2 (en) * 2000-03-15 2005-08-16 Texas Instruments Incorporated Integrated circuits, systems, apparatus, packets and processes utilizing path diversity for media over packet applications
CA2280925A1 (en) 1999-07-29 2001-01-29 Bernard Charles Sherman Stabilized cefuroxime axetil
IN191496B (de) * 1999-07-30 2003-12-06 Ranbaxy Lab Ltd
KR100342943B1 (ko) * 1999-08-04 2002-07-02 민경윤 비결정질 세푸록심 악세틸 고형분산체, 이의 제조 방법 및 이를 포함하는 경구투여용 조성물
JP2001131071A (ja) * 1999-10-29 2001-05-15 Meiji Seika Kaisha Ltd 非晶質および非晶質を含有する医薬組成物
KR100357816B1 (ko) * 2000-05-09 2002-10-18 보령제약 주식회사 무정형 세푸록심 악세틸의 제조 및 이의 분리방법
IN190849B (de) 2000-07-17 2003-08-23 Ranbaxy Lab Ltd
KR20020016052A (ko) * 2000-08-24 2002-03-04 최현식 무정형 세푸록심 악세틸의 제조방법
AT411996B (de) * 2000-09-11 2004-08-26 Sandoz Ag Verfahren zur herstellung von cefuroxim in der form seines n-butylammoniumsalzes
KR100399195B1 (ko) * 2001-03-17 2003-09-26 신풍제약주식회사 무정형 세푸록심 악세틸의 제조방법
ITMI20011766A1 (it) * 2001-08-10 2003-02-10 A & G Soluzioni Digitali S R L Dispositivo e metodo per la simulazione della presenza di una o piu' sorgenti di suoni in posizioni virtuali nello spazio acustico a tre dim
ITMI20011763A1 (it) * 2001-08-10 2003-02-10 Antibioticos Spa Processo di preparazione di cefuroxime axelite ad elevata purezza
DE60225026T2 (de) * 2001-09-10 2009-02-05 F. Hoffmann-La Roche Ag Ölige thixotrope zusammensetzungen
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KR100552567B1 (ko) * 2003-08-23 2006-02-15 한국유나이티드제약 주식회사 수분 흡수에 안정하고 빠르게 붕해되는 세푸록심 악세틸을포함하는 정제의 조성물 및 제조 방법
CN1909889B (zh) * 2004-01-09 2010-06-02 韩美药品株式会社 头孢呋辛酯颗粒及其制备方法
US7633033B2 (en) * 2004-01-09 2009-12-15 General Lasertronics Corporation Color sensing for laser decoating
CN100448879C (zh) * 2004-07-22 2009-01-07 北京化工大学 一种无定型头孢呋辛酯的制备方法
DE102005019458A1 (de) 2005-04-25 2006-10-26 Grünenthal GmbH Darreichungsform mit verbesserter Freisetzung von Cefuroximaxetil
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Also Published As

Publication number Publication date
ZA835579B (en) 1984-09-26
DK164507B (da) 1992-07-06
EP0107276B1 (de) 1987-10-07
CY1434A (en) 1988-09-02
DE3374010D1 (en) 1987-11-12
DK68392D0 (da) 1992-05-25
CZ403191A3 (en) 1993-05-12
SE8304208D0 (sv) 1983-07-29
FR2531087A1 (fr) 1984-02-03
DE3327449A1 (de) 1984-02-02
PL243228A1 (en) 1984-08-27
EP0107276A2 (de) 1984-05-02
YU44680B (en) 1990-12-31
KR840005454A (ko) 1984-11-12
FI832757A0 (fi) 1983-07-29
IE831804L (en) 1984-01-30
GB2127401A (en) 1984-04-11
JPH0730084B2 (ja) 1995-04-05
SG26088G (en) 1988-07-15
CH657134A5 (de) 1986-08-15
SK277896B6 (en) 1995-07-11
CZ280528B6 (cs) 1996-02-14
SU1266471A3 (ru) 1986-10-23
NO163897B (no) 1990-04-30
IL69375A (en) 1986-12-31
FI76093B (fi) 1988-05-31
US4994567A (en) 1991-02-19
SK403191A3 (en) 1995-07-11
IT8348789A0 (it) 1983-07-29
GB2127401B (en) 1986-04-16
ES8505689A1 (es) 1985-06-01
US4562181A (en) 1985-12-31
LU84935A1 (fr) 1983-11-23
BE897422A (fr) 1984-01-30
PT77135B (en) 1986-01-24
IT1168206B (it) 1987-05-20
FI832757A (fi) 1984-01-31
DK68392A (da) 1992-05-25
AU566881B2 (en) 1987-11-05
CS259515B2 (en) 1988-10-14
DOP1990004773A (es) 1999-02-09
AT382154B (de) 1987-01-26
JPS5944391A (ja) 1984-03-12
CS568783A2 (en) 1988-03-15
YU155883A (en) 1986-04-30
GR79349B (de) 1984-10-22
KR910000046B1 (ko) 1991-01-19
FI76093C (fi) 1988-09-09
DK349083A (da) 1984-01-31
IL69375A0 (en) 1983-11-30
GB8320518D0 (en) 1983-09-01
US5013833A (en) 1991-05-07
NO163897C (no) 1990-08-08
EP0107276A3 (en) 1985-03-06
KE3805A (en) 1988-06-03
ES524590A0 (es) 1985-06-01
CA1240313A (en) 1988-08-09
DK164507C (da) 1992-11-23
NO832773L (no) 1984-01-31
SE453195B (sv) 1988-01-18
DK349083D0 (da) 1983-07-29
PL156001B1 (pl) 1992-01-31
AU1741783A (en) 1984-02-02
US4820833A (en) 1989-04-11
SE8304208L (sv) 1984-01-31
PT77135A (en) 1983-08-01
ZW17383A1 (en) 1983-10-26
NZ205083A (en) 1986-03-14
ECSP941098A (es) 1995-01-16
HK84288A (en) 1988-10-28
MY8700058A (en) 1987-12-31
IE55748B1 (en) 1991-01-02
FR2531087B1 (fr) 1985-11-22
HU190603B (en) 1986-09-29
NL8302705A (nl) 1984-02-16

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