AR052907A1 - Compuesto 14,15-deshidro-16-oxoparahercuamida y compuestos 2- desoxo de parahercuamida y marcfortina - Google Patents

Compuesto 14,15-deshidro-16-oxoparahercuamida y compuestos 2- desoxo de parahercuamida y marcfortina

Info

Publication number
AR052907A1
AR052907A1 ARP060100487A ARP060100487A AR052907A1 AR 052907 A1 AR052907 A1 AR 052907A1 AR P060100487 A ARP060100487 A AR P060100487A AR P060100487 A ARP060100487 A AR P060100487A AR 052907 A1 AR052907 A1 AR 052907A1
Authority
AR
Argentina
Prior art keywords
15alpha
14alpha
hydroxy
compound
compounds
Prior art date
Application number
ARP060100487A
Other languages
English (en)
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21695455&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR052907(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of AR052907A1 publication Critical patent/AR052907A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings

Abstract

Un compuesto que es 14,15-deshidro-16-oxoparahercuamiada B. Reivindicacion 2: Compuestos caracterizados porque están seleccionados del grupo constituido por: 15alfa-etil-14alfa-hidroxi-17- oxomarcfortina A; 14alfa-hidroxi-15alfa-vinil-17- oxomarcfortina A; 14alfa-hidroxi-15alfa-(1'-2'-dihidroxietil)-17-oxomarcfortina A; 14alfa- hidroxi-15alfa-hidroximetil-17-oxomarcfortina A; 15alfa-fluorometil-14alfa-hidroxi-17-oxomarcfortina A; 14,15-deshidro-15- metilmarcfortina A; 14alfa-hidroxi- 16,17-dioxo-15alfa-metilmarcfortina A; 14alfa-hidroxi-16-oxo-15alfa-metilparahercuamida B; 16,17- dioxomarcforina A; 16-oxoparahercuamida B (XVI); 14alfa-hidroxi-15alfa-17-oxomarcfortina.
ARP060100487A 1995-07-21 2006-02-10 Compuesto 14,15-deshidro-16-oxoparahercuamida y compuestos 2- desoxo de parahercuamida y marcfortina AR052907A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US132495P 1995-07-21 1995-07-21

Publications (1)

Publication Number Publication Date
AR052907A1 true AR052907A1 (es) 2007-04-11

Family

ID=21695455

Family Applications (10)

Application Number Title Priority Date Filing Date
ARP960103674A AR003466A1 (es) 1995-07-21 1996-07-19 Compuestos 14-hidroxi-2-desoxoparahercuamida b
ARP030100483A AR038429A2 (es) 1995-07-21 2003-02-13 Compuestos 15-alquil-16-hidroxilo de marcfortina
ARP030100485A AR038431A2 (es) 1995-07-21 2003-02-13 Derivados 2-desoxo-15-alquilo de marcfortina
ARP030100482A AR038428A2 (es) 1995-07-21 2003-02-13 Compuestos fluorados de marcfortina
ARP030100484A AR038430A2 (es) 1995-07-21 2003-02-13 Derivados de parahercuamida b
ARP030100486A AR038432A2 (es) 1995-07-21 2003-02-13 Derivados 1,2-dihidro de parahercuamida y marcfortina
ARP030100481A AR038427A2 (es) 1995-07-21 2003-02-13 Compuestos 15-alquil-14-hidroxilo de marcfortina y parahercuamida
ARP030100488A AR038434A2 (es) 1995-07-21 2003-02-13 Compuesto 14,15-dihidro-16-oxoparahercuamida y compuestos 2-desoxo de parahercuamida y marcfortina
ARP030100487A AR038433A2 (es) 1995-07-21 2003-02-13 Derivados 2-alquil-2-desoxo de parahercuamida y marcfortina
ARP060100487A AR052907A1 (es) 1995-07-21 2006-02-10 Compuesto 14,15-deshidro-16-oxoparahercuamida y compuestos 2- desoxo de parahercuamida y marcfortina

Family Applications Before (9)

Application Number Title Priority Date Filing Date
ARP960103674A AR003466A1 (es) 1995-07-21 1996-07-19 Compuestos 14-hidroxi-2-desoxoparahercuamida b
ARP030100483A AR038429A2 (es) 1995-07-21 2003-02-13 Compuestos 15-alquil-16-hidroxilo de marcfortina
ARP030100485A AR038431A2 (es) 1995-07-21 2003-02-13 Derivados 2-desoxo-15-alquilo de marcfortina
ARP030100482A AR038428A2 (es) 1995-07-21 2003-02-13 Compuestos fluorados de marcfortina
ARP030100484A AR038430A2 (es) 1995-07-21 2003-02-13 Derivados de parahercuamida b
ARP030100486A AR038432A2 (es) 1995-07-21 2003-02-13 Derivados 1,2-dihidro de parahercuamida y marcfortina
ARP030100481A AR038427A2 (es) 1995-07-21 2003-02-13 Compuestos 15-alquil-14-hidroxilo de marcfortina y parahercuamida
ARP030100488A AR038434A2 (es) 1995-07-21 2003-02-13 Compuesto 14,15-dihidro-16-oxoparahercuamida y compuestos 2-desoxo de parahercuamida y marcfortina
ARP030100487A AR038433A2 (es) 1995-07-21 2003-02-13 Derivados 2-alquil-2-desoxo de parahercuamida y marcfortina

Country Status (31)

Country Link
US (2) US5703078A (es)
EP (3) EP0871631B1 (es)
JP (2) JP4122447B2 (es)
KR (1) KR100428335B1 (es)
CN (2) CN1277830C (es)
AR (10) AR003466A1 (es)
AT (1) ATE311390T1 (es)
AU (1) AU699644B2 (es)
BR (7) BR9612975B8 (es)
CA (1) CA2225813C (es)
CO (1) CO4750664A1 (es)
CZ (1) CZ296008B6 (es)
DE (1) DE69635524T2 (es)
DK (2) DK1489082T3 (es)
ES (2) ES2249783T3 (es)
FI (2) FI115912B (es)
HK (2) HK1017883A1 (es)
HU (1) HU226296B1 (es)
ID (1) ID30373A (es)
MX (1) MX9800625A (es)
MY (1) MY113806A (es)
NO (1) NO324287B1 (es)
NZ (1) NZ311952A (es)
PL (1) PL185007B1 (es)
PT (1) PT1489082E (es)
RU (1) RU2162090C2 (es)
SI (1) SI0871631T1 (es)
SK (2) SK284833B6 (es)
TW (1) TW334436B (es)
WO (1) WO1997003988A1 (es)
ZA (1) ZA965908B (es)

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Also Published As

Publication number Publication date
EP0871631A1 (en) 1998-10-21
BR9612974B8 (pt) 2014-10-29
MY113806A (en) 2002-05-31
CN1277830C (zh) 2006-10-04
EP1489082B1 (en) 2013-11-20
BR9609812B8 (pt) 2014-10-29
KR100428335B1 (ko) 2004-06-16
FI118471B (fi) 2007-11-30
PT1489082E (pt) 2013-12-23
AR038434A2 (es) 2005-01-12
AR038432A2 (es) 2005-01-12
AR038433A2 (es) 2005-01-12
BR9612973B8 (pt) 2014-10-29
NO980255L (no) 1998-03-20
EP1400523A2 (en) 2004-03-24
SK5498A3 (en) 1998-08-05
BR9612944B8 (pt) 2014-10-29
JP2008007516A (ja) 2008-01-17
CZ11098A3 (cs) 1998-06-17
DK0871631T3 (da) 2006-03-13
CA2225813A1 (en) 1997-02-06
FI980112A0 (fi) 1998-01-20
SI0871631T1 (sl) 2006-04-30
CZ296008B6 (cs) 2005-12-14
AR038431A2 (es) 2005-01-12
EP0871631B1 (en) 2005-11-30
DK1489082T3 (da) 2013-12-09
HK1061242A1 (en) 2004-09-10
ZA965908B (en) 1997-01-12
US5703078A (en) 1997-12-30
ID30373A (id) 1997-01-23
ATE311390T1 (de) 2005-12-15
AR038427A2 (es) 2005-01-12
FI980112A (fi) 1998-01-20
FI20050238A (fi) 2005-03-04
HK1017883A1 (en) 1999-12-03
AR038429A2 (es) 2005-01-12
DE69635524D1 (de) 2006-01-05
PL185007B1 (pl) 2003-01-31
BR9612963B8 (pt) 2014-10-29
CN1125824C (zh) 2003-10-29
CO4750664A1 (es) 1999-03-31
EP1400523A3 (en) 2004-04-07
NO324287B1 (no) 2007-09-17
CN1191537A (zh) 1998-08-26
BR9612975B8 (pt) 2014-10-29
SK285248B6 (sk) 2006-09-07
JP4122447B2 (ja) 2008-07-23
MX9800625A (es) 1998-04-30
JPH11509550A (ja) 1999-08-24
EP1489082A1 (en) 2004-12-22
HUP9802221A3 (en) 2000-05-29
AR003466A1 (es) 1998-08-05
AR038430A2 (es) 2005-01-12
FI115912B (fi) 2005-08-15
RU2162090C2 (ru) 2001-01-20
NO980255D0 (no) 1998-01-20
BR9612972B8 (pt) 2014-10-29
AU699644B2 (en) 1998-12-10
CA2225813C (en) 2008-02-26
HU226296B1 (hu) 2008-08-28
AU6337396A (en) 1997-02-18
TW334436B (en) 1998-06-21
NZ311952A (en) 1999-03-29
HUP9802221A2 (hu) 1999-02-01
ES2439569T3 (es) 2014-01-23
ES2249783T3 (es) 2006-04-01
PL324574A1 (en) 1998-06-08
BR9609812A (pt) 1999-03-02
CN1495183A (zh) 2004-05-12
WO1997003988A1 (en) 1997-02-06
US5750695A (en) 1998-05-12
AR038428A2 (es) 2005-01-12
SK284833B6 (sk) 2005-12-01
DE69635524T2 (de) 2006-07-06

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