AP136A - Substituted:- 1,3-oxathiolanes with antiviral properties. - Google Patents

Substituted:- 1,3-oxathiolanes with antiviral properties. Download PDF

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Publication number
AP136A
AP136A APAP/P/1990/000163A AP9000163A AP136A AP 136 A AP136 A AP 136A AP 9000163 A AP9000163 A AP 9000163A AP 136 A AP136 A AP 136A
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AP
ARIPO
Prior art keywords
formula
compound
group
oxathiolane
hydroxymethyl
Prior art date
Application number
APAP/P/1990/000163A
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English (en)
Other versions
AP9000163A0 (en
Inventor
BELLEAY, (DECEASED) Bernard
Belleau, (Executor Of Estate) Pierette
Nghe Nguyen-Ba
Original Assignee
Iaf Biochem Int
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25678044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP136(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Iaf Biochem Int filed Critical Iaf Biochem Int
Publication of AP9000163A0 publication Critical patent/AP9000163A0/xx
Application granted granted Critical
Publication of AP136A publication Critical patent/AP136A/en
Priority claimed from CA002152269A external-priority patent/CA2152269C/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D327/02—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
    • C07D327/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
APAP/P/1990/000163A 1989-02-08 1990-02-08 Substituted:- 1,3-oxathiolanes with antiviral properties. AP136A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/308,101 US5047407A (en) 1989-02-08 1989-02-08 2-substituted-5-substituted-1,3-oxathiolanes with antiviral properties
CA002152269A CA2152269C (en) 1989-02-08 1992-12-21 Process for preparing substituted 1,3-oxathiolanes with antiviral properties

Publications (2)

Publication Number Publication Date
AP9000163A0 AP9000163A0 (en) 1990-04-30
AP136A true AP136A (en) 1991-08-05

Family

ID=25678044

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1990/000163A AP136A (en) 1989-02-08 1990-02-08 Substituted:- 1,3-oxathiolanes with antiviral properties.

Country Status (35)

Country Link
US (1) US5047407A (el)
EP (2) EP0382526B1 (el)
JP (4) JP2644357B2 (el)
KR (1) KR960007531B1 (el)
CN (1) CN1033640C (el)
AP (1) AP136A (el)
AT (2) ATE138065T1 (el)
AU (1) AU630913B2 (el)
CA (1) CA2009637C (el)
CY (1) CY2036A (el)
CZ (1) CZ282720B6 (el)
DE (3) DE69034119T2 (el)
DK (2) DK0711771T3 (el)
ES (2) ES2206476T3 (el)
FI (1) FI98065C (el)
GR (1) GR3019919T3 (el)
HK (2) HK51997A (el)
HR (1) HRP940040B1 (el)
HU (2) HU208134B (el)
IE (1) IE72184B1 (el)
IL (1) IL93318A (el)
LU (1) LU88809I2 (el)
MX (1) MX19437A (el)
NL (1) NL960025I2 (el)
NO (2) NO179518C (el)
NZ (1) NZ232421A (el)
OA (1) OA09193A (el)
PL (1) PL164785B1 (el)
PT (1) PT93094B (el)
RU (1) RU2092485C1 (el)
SG (2) SG77215A1 (el)
SI (1) SI9010243B (el)
SK (1) SK279175B6 (el)
YU (1) YU48840B (el)
ZA (1) ZA90943B (el)

Families Citing this family (149)

* Cited by examiner, † Cited by third party
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