ZA201505267B - Heterocyclic amides as kinase inhibitors - Google Patents

Heterocyclic amides as kinase inhibitors

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Publication number
ZA201505267B
ZA201505267B ZA2015/05267A ZA201505267A ZA201505267B ZA 201505267 B ZA201505267 B ZA 201505267B ZA 2015/05267 A ZA2015/05267 A ZA 2015/05267A ZA 201505267 A ZA201505267 A ZA 201505267A ZA 201505267 B ZA201505267 B ZA 201505267B
Authority
ZA
South Africa
Prior art keywords
kinase inhibitors
heterocyclic amides
amides
heterocyclic
kinase
Prior art date
Application number
ZA2015/05267A
Other languages
English (en)
Inventor
Daohua Zhang
Jr Robert Singhaus
Clark A Sehon
Joshi M Ramanjulu
Attiq Rahman
Lara Kathryn Leister
Jr Robert W Marquis
Shah Ami Lakdawala
Jianxing Kang
Jae U Jeong
Philip Anthony Harris
Peter J Gough
Patrick M Eidam
Deepak Bandyopadhyay
Original Assignee
Glaxosmithkline Intellectual Property And Dev Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Intellectual Property And Dev Ltd filed Critical Glaxosmithkline Intellectual Property And Dev Ltd
Publication of ZA201505267B publication Critical patent/ZA201505267B/en

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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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