HRP20180900T1 - Heterociklički amidi kao inhibitori kinaza - Google Patents

Heterociklički amidi kao inhibitori kinaza

Info

Publication number
HRP20180900T1
HRP20180900T1 HRP20180900TT HRP20180900T HRP20180900T1 HR P20180900 T1 HRP20180900 T1 HR P20180900T1 HR P20180900T T HRP20180900T T HR P20180900TT HR P20180900 T HRP20180900 T HR P20180900T HR P20180900 T1 HRP20180900 T1 HR P20180900T1
Authority
HR
Croatia
Prior art keywords
kinase inhibitors
heterocyclic amides
amides
heterocyclic
kinase
Prior art date
Application number
HRP20180900TT
Other languages
English (en)
Croatian (hr)
Inventor
Deepak BANDYOPADHYAY
Patrick M. Eidam
Peter J. GOUGH
Philip Anthony Harris
Jae U. Jeong
Jianxing Kang
Bryan Wayne KING
Ami Lakdawala Shah
Robert W. Marquis
Lara Kathryn LEISTER
Attiq Rahman
Joshi M. Ramanjulu
Clark A Sehon
JR. Robert SINGHAUS
Daohua Zhang
Original Assignee
Glaxosmithkline Intellectual Property Development Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Intellectual Property Development Limited filed Critical Glaxosmithkline Intellectual Property Development Limited
Publication of HRP20180900T1 publication Critical patent/HRP20180900T1/hr

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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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    • C07D223/06Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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HRP20180900TT 2013-02-15 2014-02-14 Heterociklički amidi kao inhibitori kinaza HRP20180900T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201361765664P 2013-02-15 2013-02-15
US201361790044P 2013-03-15 2013-03-15
EP14705891.1A EP2956452B1 (en) 2013-02-15 2014-02-14 Heterocyclic amides as kinase inhibitors
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