LT3342771T - Heterocikliniai amidai kaip kinazės inhibitoriai - Google Patents

Heterocikliniai amidai kaip kinazės inhibitoriai

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Publication number
LT3342771T
LT3342771T LTEP18155836.2T LT18155836T LT3342771T LT 3342771 T LT3342771 T LT 3342771T LT 18155836 T LT18155836 T LT 18155836T LT 3342771 T LT3342771 T LT 3342771T
Authority
LT
Lithuania
Prior art keywords
amids
heterocyclic
kinase inhibitors
kinase
inhibitors
Prior art date
Application number
LTEP18155836.2T
Other languages
English (en)
Inventor
Deepak BANDYOPADHYAY
Patrick M. Eidam
Peter J. GOUGH
Philip Anthony Harris
Jae U. Jeong
Jianxing Kang
Bryan Wayne KING
Ami Lakdawala Shah
Marquis, Jr.
Lara Kathryn LEISTER
Attiq Rahman
Joshi M. Ramanjulu
Clark A. Sehon
Singhaus, Jr.
Daohua Zhang
Original Assignee
Glaxosmithkline Intellectual Property Development Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Intellectual Property Development Ltd filed Critical Glaxosmithkline Intellectual Property Development Ltd
Publication of LT3342771T publication Critical patent/LT3342771T/lt

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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