YU84703A - Oralni rastvor aripiprazola - Google Patents

Oralni rastvor aripiprazola

Info

Publication number
YU84703A
YU84703A YU84703A YUP84703A YU84703A YU 84703 A YU84703 A YU 84703A YU 84703 A YU84703 A YU 84703A YU P84703 A YUP84703 A YU P84703A YU 84703 A YU84703 A YU 84703A
Authority
YU
Yugoslavia
Prior art keywords
oral solution
aripiprazole
acid
aripiprazole oral
solution
Prior art date
Application number
YU84703A
Other languages
English (en)
Inventor
Prakash Parab
Joyce Chou
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23099862&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=YU84703(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of YU84703A publication Critical patent/YU84703A/sh
Publication of RS52082B publication Critical patent/RS52082B/sr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Sadašnji pronalazak obezbeđuje farmaceutski rastvor pogodan za oralnu administraciju i uključuje aripiprazol, farmaceutski pogodni sistem rastvarača, jedno ili više sredstava za poboljšanje i/ili za maskiranje ukusa, i jedan ili više agenasa odabranih od grupe koja uključuje mlečnu kiselinu, sirćetnu kiselinu, vinsku kiselinu i limunsku kiselinu, pri čemu je pH navedenog rastvora između 2.5 i 4.5.[The present invention provides for a pharmaceutical solution suitable for oral administration comprising aripiprazole, a pharmaceutically suitable solvent system, one or more taste-enhancing/masking agents and one or more agents selected from the group consisting of lactic acid, acetic acid, tartaric acid and citric acid, wherein said solution has a pH from 2.5 to 4.5.
YU84703A 2001-04-25 2002-04-24 Oralni rastvor aripiprazola RS52082B (sr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US28671801P 2001-04-25 2001-04-25

Publications (2)

Publication Number Publication Date
YU84703A true YU84703A (sh) 2006-08-17
RS52082B RS52082B (sr) 2012-06-30

Family

ID=23099862

Country Status (37)

Country Link
US (1) US6977257B2 (sh)
EP (2) EP2436384B2 (sh)
JP (1) JP4401077B2 (sh)
KR (1) KR100909329B1 (sh)
CN (1) CN1512884B (sh)
AR (1) AR033168A1 (sh)
AT (1) ATE537831T1 (sh)
AU (1) AU2002254722B2 (sh)
BG (1) BG66177B1 (sh)
BR (1) BR0208986A (sh)
CA (1) CA2445276C (sh)
CY (1) CY1112606T1 (sh)
CZ (1) CZ306181B6 (sh)
DK (1) DK1381367T3 (sh)
EE (1) EE05581B1 (sh)
ES (1) ES2377855T3 (sh)
GE (1) GEP20053602B (sh)
HK (2) HK1058316A1 (sh)
HR (1) HRP20030870B1 (sh)
HU (1) HU230456B1 (sh)
IL (2) IL158202A0 (sh)
IS (1) IS2863B (sh)
MX (1) MXPA03009728A (sh)
MY (1) MY129350A (sh)
NO (1) NO324606B1 (sh)
NZ (1) NZ528550A (sh)
PE (1) PE20021086A1 (sh)
PL (1) PL206882B1 (sh)
PT (1) PT1381367E (sh)
RS (1) RS52082B (sh)
RU (1) RU2295960C2 (sh)
SK (1) SK287948B6 (sh)
TW (1) TWI337865B (sh)
UA (1) UA76144C2 (sh)
UY (1) UY27273A1 (sh)
WO (1) WO2002085366A1 (sh)
ZA (1) ZA200307797B (sh)

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Also Published As

Publication number Publication date
UA76144C2 (uk) 2006-07-17
HU230456B1 (hu) 2016-07-28
HRP20030870B1 (en) 2011-10-31
KR100909329B1 (ko) 2009-07-24
DK1381367T3 (da) 2012-04-10
AR033168A1 (es) 2003-12-03
US20020193438A1 (en) 2002-12-19
RS52082B (sr) 2012-06-30
HRP20030870A2 (en) 2004-06-30
CA2445276C (en) 2009-10-13
EP2436384A2 (en) 2012-04-04
EE200300523A (et) 2004-02-16
UY27273A1 (es) 2002-11-29
HUP0303946A3 (en) 2005-06-28
EP2436384A3 (en) 2012-09-19
BR0208986A (pt) 2004-04-20
ATE537831T1 (de) 2012-01-15
BG108216A (bg) 2004-12-30
BG66177B1 (bg) 2011-11-30
HK1058316A1 (en) 2004-05-14
PE20021086A1 (es) 2002-12-14
CY1112606T1 (el) 2016-02-10
RU2003132426A (ru) 2005-04-20
CZ306181B6 (cs) 2016-09-14
GEP20053602B (en) 2005-08-10
IS2863B (is) 2013-12-15
NO20034705D0 (no) 2003-10-21
MY129350A (en) 2007-03-30
CN1512884A (zh) 2004-07-14
ES2377855T3 (es) 2012-04-02
NO20034705L (no) 2003-11-28
IS6994A (is) 2003-10-14
TWI337865B (en) 2011-03-01
WO2002085366A1 (en) 2002-10-31
JP2004532225A (ja) 2004-10-21
CZ20032821A3 (cs) 2004-09-15
CN1512884B (zh) 2010-05-26
IL158202A (en) 2008-04-13
PL364666A1 (en) 2004-12-13
HK1168792A1 (en) 2013-01-11
HUP0303946A2 (hu) 2004-04-28
ZA200307797B (en) 2004-10-06
EP1381367B1 (en) 2011-12-21
SK287948B6 (sk) 2012-06-04
CA2445276A1 (en) 2002-10-31
EP1381367A1 (en) 2004-01-21
PT1381367E (pt) 2012-03-01
JP4401077B2 (ja) 2010-01-20
EP2436384B2 (en) 2018-05-23
AU2002254722B2 (en) 2006-11-09
IL158202A0 (en) 2004-05-12
SK12642003A3 (sk) 2004-07-07
EP1381367A4 (en) 2009-07-01
KR20030096332A (ko) 2003-12-24
EP2436384B1 (en) 2015-06-10
RU2295960C2 (ru) 2007-03-27
NZ528550A (en) 2005-03-24
MXPA03009728A (es) 2004-01-29
NO324606B1 (no) 2007-11-26
PL206882B1 (pl) 2010-10-29
EE05581B1 (et) 2012-10-15
US6977257B2 (en) 2005-12-20

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